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Titolo Data di pubblicazione Autore(i) File
Design, synthesis and biological evaluation of novel dipeptide-like rhodesain inhibitors containing a conformationally constrained 3-bromoisoxazoline warhead 1-gen-2015 Ettari, Roberta; Previti, Santo; Pinto, A.; Tamborini, L.; Cullia, G.; Pietra, V. La; Marinelli, L.; Novellino, E.; De Micheli, C.; Conti, P.; Grasso, Silvana; Zappala', Maria
NMR conformational analysis in solution of a potent class of cysteine proteases inhibitors 1-gen-2015 Rotondo, Archimede; Ettari, Roberta; Grasso, Silvana; Zappala', Maria
Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation 1-gen-2015 Ettari, Roberta; Pinto, Andrea; Previti, Santo; Tamborini, Lucia; Angelo, Ilenia C.; Pietra, Valeria La; Marinelli, Luciana; Novellino, Ettore; Schirmeister, Tanja; Zappala', Maria; Grasso, Silvana; De Micheli, Carlo; Conti, Paola
Synthesis and pharmacological evaluation of α4β2 nicotinic ligands with a 3-fluoropyrrolidine nucleus 1-gen-2015 Tamborini, Lucia; Pinto, Andrea; Ettari, Roberta; Gotti, Cecilia; Fasoli, Francesca; Conti, Paola; De Micheli, Carlo
Mechanism and Site of Inhibition of AMPA Receptors: Substitution of One and Two Methyl groups at the 4-Aminophenyl Ring of 2,3-Benzodiazepine and Implications in the “E” Site 1-gen-2015 Wang, C.; Wu, A.; Shen, Y. C; Ettari, Roberta; Grasso, Silvana; Niu, L.
Identification of novel 5 arylidene-3-phenyl-2 thioxoimidazolidin-4-ones as inhibitors of the chymotrypsin-like activities of the constitutive and immuno-proteasomes 1-gen-2016 Adornato, Ilenia; Ettari, Roberta; Maccari, Rosanna; Kaffy, Julia; Ottana', Rosaria; Grasso, Silvana
Development of novel amides as non covalent inhibitors of immunoproteasome 1-gen-2016 Ettari, Roberta; Previti, Santo; Maiorana, Santina; Guccione, Manuela; Ongeri, S.; Zappala', Maria; Grasso, Silvana
Development of novel 1,4-benzodiazepines as antitrypanosomal agents 1-gen-2016 Previti, Santo; Ettari, Roberta; Maiorana, Santina; Cosconati, S.; Schirmeister, T.; Grasso, Silvana; Zappala', Maria
Identification of noncovalent proteasome inhibitors with high selectivity for chymotrypsin-like activity by a multistep structure-based virtual screening 1-gen-2016 Di Giovanni, Carmen; Ettari, Roberta; Sarno, Serena; Rotondo, Archimede; Bitto, Alessandra; Squadrito, Francesco; Altavilla, Domenica; Schirmeister, Tanja; Novellino, Ettore; Grasso, Silvana; Zappala', Maria; Lavecchia, Antonio
A novel 2,3-benzodiazepine-4-one derivative AMPA antagonist inhibits G2/M transition and induces apoptosis in human leukemia Jurkat T cell line 1-gen-2016 Parenti, S.; Casagrande, G.; Montanari, M.; Espahbodinia, Milad; Ettari, Roberta; Grande, A.; Corsi, L.
The Inhibition of Cysteine Proteases Rhodesain and TbCatB: A Valuable Approach to Treat Human African Trypanosomiasis 1-gen-2016 Ettari, Roberta; Previti, Santo; Tamborini, Lucia; Cullia, Gregorio; Grasso, Silvana; Zappala', Maria
G-Protein-Coupled Receptor Kinase 2 (GRK2) Inhibitors: Current Trends and Future Perspectives 1-gen-2016 Guccione, Manuela; Ettari, Roberta; Taliani, Sabrina; Da Settimo, Federico; Zappala', Maria; Grasso, Silvana
Synthesis and biological evaluation of novel peptidomimetics as rhodesain inhibitors 1-gen-2016 Ettari, Roberta; Previti, Santo; Cosconati, S.; Kesselring, J.; Schirmeister, T.; Grasso, Silvana; Zappala', Maria
Development of novel 1,4-benzodiazepine-based Michael acceptors as antitrypanosomal agents 1-gen-2016 Ettari, Roberta; Previti, Santo; Cosconati, Sandro; Maiorana, Santina; Schirmeister, Tanja; Grasso, Silvana; Zappala', Maria
Immunoproteasome-selective inhibitors: a promising strategy to treat hematologic malignancies, autoimmune and inflammatory diseases 1-gen-2016 Ettari, Roberta; Previti, Santo; Bitto, Alessandra; Grasso, Silvana; Zappala', Maria
Development of novel peptide-based Michael acceptors targeting rhodesain and falcipain-2 for the treatment of neglected tropical diseases (NTDs) 1-gen-2017 Previti, Santo; Ettari, Roberta; Grasso, Silvana; Zappala', Maria
Development of novel peptide-based Michael acceptors targeting rhodesain for the treatment of human african trypanosomiasis 1-gen-2017 Previti, Santo; Ettari, Roberta; Cosconati, Sandro; Schirmeister, Tanja; Rhosental, Philip J; Zappala', Maria; Grasso, Silvana
Development of novel Michael acceptors targeting rhodesain as antitrypanosomal agents 1-gen-2017 Previti, Santo; Ettari, Roberta; Cosconati, Sandro; Schirmeister, Tanja; Rosenthal, Philip J.; Grasso, Silvana; Zappala', Maria
BAY 11-7082 inhibits the NF-κB and NLRP3 inflammasome pathways and protects against IMQ-induced psoriasis 1-gen-2017 Irrera, Natasha; Vaccaro, Mario; Bitto, Alessandra; Pallio, Giovanni; Pizzino, Carmelo Gabriele; Lentini, Maria; Arcoraci, Vincenzo; Minutoli, Letteria; Scuruchi, Michele; Cutroneo, Giuseppina; Anastasi, Giuseppe Pio; Ettari, Roberta; Squadrito, Francesco; Altavilla, Domenica
Development of novel N-3-bromoisoxazolin-5-yl substituted 2,3-benzodiazepines as noncompetitive AMPAR antagonists 1-gen-2017 ESPAHBODINIA, MILAD; ETTARI, Roberta; Wen, Wei; Wu, Andrew; Shen, Yu Chuan; Niu, Li; GRASSO, Silvana; ZAPPALA', Maria
Mostrati risultati da 61 a 80 di 137
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