Sfoglia per Autore
Synthesis and characterization of isomeric 2,3,3A,4-tetrahydro-1H-pyrrolo[1,2-A]benzimidazol-1-ones from 1,2-phenylenediamines and 3-acylpropionic acids
1988-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Romeo, Giovanni; Zappala', Maria
A simple, one-pot synthesis of novel 1H,3H-thiazolo[3,4-A]benzimidazoles
1988-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Romeo, Giovanni; Zappala', Maria
Compounds with potential anti-tumor activity VII. Synthesis and anti-tumor activity of 1-aryl-N,N'-di(1,3,4-thiadiazol-2-yl)methylenediamines
1990-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Fenech, Giovanna; Zappala', Maria; Monforte, Anna Maria
Anti-HIV agents II. Synthesis and in vitro anti-HIV activity of novel 1H,3H-thiazolo[3,4-a]benzimidazoles.
1991-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria
ANTI-HIV AGENTS .1. SYNTHESIS AND INVITRO ANTI-HIV EVALUATION OF NOVEL 1H,3H-THIAZOLO[3,4-A]BENZIMIDAZOLES
1991-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria
1H,3H-Thiazolo[3,4-a]benzimidazoles and pharmaceutical compositions containing them
1992-01-01 Monforte, Pietro; Monforte, Anna Maria; Zappala', Maria; Romeo, Giovanni; Grasso, Silvana; Chimirri, Alba
Sintesi ed attività anti-HIV di 1H,3H-tiazolo[3,4-a]benzimidazoli-sostituiti
1993-01-01 Monforte, Pietro; Monforte, Anna Maria; Zappala', Maria; Romeo, Giovanni; Grasso, Silvana; Chimirri, Alba
1-Phenyl-substituted 1H,3H-thiazolo[3,4-a]benzimidazoles and pharmaceutical compositions containing them
1993-01-01 Monforte, Pietro; Monforte, Anna Maria; Zappala', Maria; Romeo, Giovanni; Grasso, Silvana; Chimirri, Alba
Pyrrolo[1',2':1,2]imidazo[4,5-b]pyridines, pyrrolo[2',1':2,3]imidazo[4,5-c]pyridines and pyrrolo[2,1-f]purines as potential benzodiazepine receptor ligands.
1993-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Zappala', Maria; Genchi, G.
ANTI-HIV AGENTS .3. SYNTHESIS AND IN-VITRO ANTI-HIV ACTIVITY OF NOVEL 1H,3H-THIAZOLO[3,4-A]IMIDAZO[4,5-B]PYRIDINES
1994-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria
STRUCTURE-ACTIVITY-RELATIONSHIPS OF ANTITUMOR THIAZOLO[3,4- A]BENZIMIDAZOLE DERIVATIVES
1994-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Carotti, A.
SYNTHESIS AND IN-VITRO ANTI-HIV ACTIVITY OF NOVEL DELTA(2)- 1,2,4-OXADIAZOLINE DERIVATIVES
1994-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Carotti, A.
NOVEL PYRROLO- AND THIAZOLO-IMIDAZOLES
1995-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria
SYNTHESIS AND ANTIHYPERTENSIVE ACTIVITY EVALUATION OF INDOLE- DERIVATIVES N-ACETAMIDO SUBSTITUTED
1995-01-01 Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Monforte, Maria Teresa; Trovato, Ada
Synthesis and in vitro antitumor activity evaluation of 9- substituted 1,2,3,4-tetrahydrocarbazoles
1996-01-01 Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Rizzo, M.
Anti-HIV agents .4. Synthesis and in vitro anti-HIV activity of novel 1-(2,6-difluorophenyl)-1H,3H-thiazolo[3,4- a]benzimidazoles
1996-01-01 Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Scopelliti, R.
Structural features and anti-human immunodeficiency virus (HIV) activity of the isomers of 1-(2',6'-difluorophenyl)-1H,3H- thiazolo[3,4-a]benzimidazole, a potent non-nucleoside HIV-1 reverse transcriptase inhibitor
1997-01-01 Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Witvrouw, M.; Jonckeere, H.; Balzarini, J.; Declercq, E.
Anti-HIV agents. V. Synthesis, structure and in vitro anti-HIV activity of novel 1H,3H-naphtho[2 ',3 ': 4,5]imidazo[1,2- c]thiazoles
1997-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A.; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Scopelliti, R.
Synthesis, structure and in vitro anti-human immunodeficiency virus activity of novel 3-methyl-1H,3H-thiazolo[3,4- a]benzimidazoles
1998-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Pannecouque, C; Witvrouw, M; DE CLERCQ, E.
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system
1999-01-01 Chimirri, Alba; DE CLERCQ, E.; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Pannecouque, C.; Rao, A.; Witvrouw, M.; Zappala', Maria
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and characterization of isomeric 2,3,3A,4-tetrahydro-1H-pyrrolo[1,2-A]benzimidazol-1-ones from 1,2-phenylenediamines and 3-acylpropionic acids | 1-gen-1988 | Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Romeo, Giovanni; Zappala', Maria | |
A simple, one-pot synthesis of novel 1H,3H-thiazolo[3,4-A]benzimidazoles | 1-gen-1988 | Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Romeo, Giovanni; Zappala', Maria | |
Compounds with potential anti-tumor activity VII. Synthesis and anti-tumor activity of 1-aryl-N,N'-di(1,3,4-thiadiazol-2-yl)methylenediamines | 1-gen-1990 | Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Fenech, Giovanna; Zappala', Maria; Monforte, Anna Maria | |
Anti-HIV agents II. Synthesis and in vitro anti-HIV activity of novel 1H,3H-thiazolo[3,4-a]benzimidazoles. | 1-gen-1991 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria | |
ANTI-HIV AGENTS .1. SYNTHESIS AND INVITRO ANTI-HIV EVALUATION OF NOVEL 1H,3H-THIAZOLO[3,4-A]BENZIMIDAZOLES | 1-gen-1991 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria | |
1H,3H-Thiazolo[3,4-a]benzimidazoles and pharmaceutical compositions containing them | 1-gen-1992 | Monforte, Pietro; Monforte, Anna Maria; Zappala', Maria; Romeo, Giovanni; Grasso, Silvana; Chimirri, Alba | |
Sintesi ed attività anti-HIV di 1H,3H-tiazolo[3,4-a]benzimidazoli-sostituiti | 1-gen-1993 | Monforte, Pietro; Monforte, Anna Maria; Zappala', Maria; Romeo, Giovanni; Grasso, Silvana; Chimirri, Alba | |
1-Phenyl-substituted 1H,3H-thiazolo[3,4-a]benzimidazoles and pharmaceutical compositions containing them | 1-gen-1993 | Monforte, Pietro; Monforte, Anna Maria; Zappala', Maria; Romeo, Giovanni; Grasso, Silvana; Chimirri, Alba | |
Pyrrolo[1',2':1,2]imidazo[4,5-b]pyridines, pyrrolo[2',1':2,3]imidazo[4,5-c]pyridines and pyrrolo[2,1-f]purines as potential benzodiazepine receptor ligands. | 1-gen-1993 | Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Zappala', Maria; Genchi, G. | |
ANTI-HIV AGENTS .3. SYNTHESIS AND IN-VITRO ANTI-HIV ACTIVITY OF NOVEL 1H,3H-THIAZOLO[3,4-A]IMIDAZO[4,5-B]PYRIDINES | 1-gen-1994 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria | |
STRUCTURE-ACTIVITY-RELATIONSHIPS OF ANTITUMOR THIAZOLO[3,4- A]BENZIMIDAZOLE DERIVATIVES | 1-gen-1994 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Carotti, A. | |
SYNTHESIS AND IN-VITRO ANTI-HIV ACTIVITY OF NOVEL DELTA(2)- 1,2,4-OXADIAZOLINE DERIVATIVES | 1-gen-1994 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Carotti, A. | |
NOVEL PYRROLO- AND THIAZOLO-IMIDAZOLES | 1-gen-1995 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria | |
SYNTHESIS AND ANTIHYPERTENSIVE ACTIVITY EVALUATION OF INDOLE- DERIVATIVES N-ACETAMIDO SUBSTITUTED | 1-gen-1995 | Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Monforte, Maria Teresa; Trovato, Ada | |
Synthesis and in vitro antitumor activity evaluation of 9- substituted 1,2,3,4-tetrahydrocarbazoles | 1-gen-1996 | Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Rizzo, M. | |
Anti-HIV agents .4. Synthesis and in vitro anti-HIV activity of novel 1-(2,6-difluorophenyl)-1H,3H-thiazolo[3,4- a]benzimidazoles | 1-gen-1996 | Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Scopelliti, R. | |
Structural features and anti-human immunodeficiency virus (HIV) activity of the isomers of 1-(2',6'-difluorophenyl)-1H,3H- thiazolo[3,4-a]benzimidazole, a potent non-nucleoside HIV-1 reverse transcriptase inhibitor | 1-gen-1997 | Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Witvrouw, M.; Jonckeere, H.; Balzarini, J.; Declercq, E. | |
Anti-HIV agents. V. Synthesis, structure and in vitro anti-HIV activity of novel 1H,3H-naphtho[2 ',3 ': 4,5]imidazo[1,2- c]thiazoles | 1-gen-1997 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A.; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Scopelliti, R. | |
Synthesis, structure and in vitro anti-human immunodeficiency virus activity of novel 3-methyl-1H,3H-thiazolo[3,4- a]benzimidazoles | 1-gen-1998 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Pannecouque, C; Witvrouw, M; DE CLERCQ, E. | |
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system | 1-gen-1999 | Chimirri, Alba; DE CLERCQ, E.; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Pannecouque, C.; Rao, A.; Witvrouw, M.; Zappala', Maria |
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