Sfoglia per Autore
Progettazione e sintesi di antagonisti non competitivi del recettore NR2B/NMDA
2009-01-01 Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Scicchitano, F; Maierù, Mt; Gitto, Rosaria
Searching for NR2B/NMDA Receptor Antagonists As Neuroprotective Agents
2009-01-01 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Bruno, Giuseppe; De Sarro, G; Chimirri, Alba
Nuovi ligandi del recettore NR2B/NMDA a struttura indolica
2009-01-01 Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Chimirri, Alba
Synthesis, biological evaluation and docking studies of NR2B/NMDA receptor antagonists
2010-01-01 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Scicchitano, F; De Sarro, G; Costa, LARA TANIA; Ciranna, L; Chimirri, Alba
New indole derivatives as promising ligands for ifenprodil site of NR2B/NMDA receptors
2010-01-01 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; De Sarro, G; Chimirri, Alba
SYNTHESIS AND BIOLOGICAL CHARACTERIZATION OF 3-SUBSTITUTED-1H-INDOLES AS LIGANDS OF GLUN2B-CONTAINING N-METHYL-D-ASPARTATE RECEPTORS
2011-01-01 Buemi, Mariarosa; Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Giovambattista De, Sarro; Lucia, Ciranna; Chimirri, Alba
SYNTHESIS AND BIOLOGICAL CHARACTERIZATION OF NEW NR2B/NMDA RECEPTOR LIGANDS
2011-01-01 Buemi, Mariarosa
DISCOVERY OF NEW INDOLE DERIVATES AS NEUROPROTECTIVE AGENTS
2011-01-01 Buemi, Mariarosa; Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; R., Alajarin; J., ALVAREZ BUILLA; R., Citraro; Chimirri, Alba
Synthesis and Biological Characterization of 3-Substituted-1H-indoles as Ligands of GluN2B-Containing N-Methyl-d-aspartate Receptors
2011-01-01 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Russo, E; De Sarro, G; Costa, LARA TANIA; Ciranna, L; Prezzavento, O; Arena, E; Ronsisvalle, S; Bruno, Giuseppe; Chimirri, Alba
Rational Design and synthesis of new GluN2B/NMDA receptor ligands as neuroprotective agents.
2012-01-01 Buemi, Mariarosa
Identification of 3-substituted-1H-indoles as ligands of GluN2B containing N-methyl-D-aspartate receptors
2012-01-01 Ferro, Stefania; Buemi, Mariarosa; Gitto, Rosaria; DE LUCA, Laura; Russo, E.; Ciranna, L.; Chimirri, Alba
Synthesis and Biological Characterization of 3-Substituted-1H-indoles as Ligands of GluN2B-containing N-Methyl-D-Aspartate Receptors. Part. 2.
2012-01-01 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Russo, E; De Sarro, G; Chisari, M; Ciranna, L; Chimirri, Alba
Design, Synthesis and Biostructural Characterization of Carbonic Anhydrase Inhibitors
2013-01-01 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Vullo, D; Supuran, Ct; Brynda, J; Rezacova, P; Pospisilova, K; Damiano, F; Chimirri, Alba
Indole derivatives as dual-effective agents for the treatment of neurodegenerative diseases: Synthesis, biological evaluation, and molecular modeling studies
2013-01-01 Maria Rosa, Buemi; Laura, De Luca; Alba, Chimirri; Stefania, Ferro; Rosaria, Gitto; Julio, Alvarez-Builla; Ramon, Alajarin
Design and optimization of isoquinoline-sulfonamides as potent and selective inhibitors of human carbonic anhydrase VII
2014-01-01 Bruno, Elvira; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Ceruso, Mariangela; Supuran, Claudiu T.; Gitto, Rosaria
Synthesis, Modelling and Biological Characterization of 3-Substituted-1H-indoles as Ligands of GluN2B-containing N-Methyl-d-Aspartate Receptors
2014-01-01 Rosaria Gitto;Laura De Luca;Stefania Ferro;Emilio Russo;Giovambattista De Sarro;Mariangela Chisari;Lucia Ciranna;Julio Alvarez-Builla;Ramon Alajarin;Maria Rosa Buemi;Alba Chimirri
Targeting GluN2B-containing N-Methyl-D-aspartate receptors: design, synthesis, and binding affinity evaluation of novel 3-substituted indoles.
2014-01-01 Buemi MR;De Luca L;Ferro S;Gitto R
From NMDA receptor antagonists to discovery of selective σ2 receptor ligands
2014-01-01 Rosaria Gitto;Laura De Luca;Stefania Ferro;Angela Scala;Simone Ronsisvalle;Carmela Parenti;Orazio Prezzavento;Maria Rosa Buemi;Alba Chimirri
Serendipitous discovery of indole derivatives as potent tyrosinase inhibitors
2015-01-01 Gitto, Rosaria; Buemi, Mariarosa; DE LUCA, Laura; Certo, Giovanna; Germano', Maria Paola; Rapisarda, Antonio; Ferro, Stefania
Synthesis and biological characterization of novel potent arylsulfonamides as human carbonic anhydrase inhibitors (hCAIs) targeting central nervous system
2015-01-01 Bruno, Elvira; Buemi, Mariarosa; DE LUCA, Laura; Ferro, Stefania; Ceruso, Mariangela; Supuran, Claudiu T.; Gitto, Rosaria
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Progettazione e sintesi di antagonisti non competitivi del recettore NR2B/NMDA | 1-gen-2009 | Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Scicchitano, F; Maierù, Mt; Gitto, Rosaria | |
Searching for NR2B/NMDA Receptor Antagonists As Neuroprotective Agents | 1-gen-2009 | Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Bruno, Giuseppe; De Sarro, G; Chimirri, Alba | |
Nuovi ligandi del recettore NR2B/NMDA a struttura indolica | 1-gen-2009 | Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Chimirri, Alba | |
Synthesis, biological evaluation and docking studies of NR2B/NMDA receptor antagonists | 1-gen-2010 | Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Scicchitano, F; De Sarro, G; Costa, LARA TANIA; Ciranna, L; Chimirri, Alba | |
New indole derivatives as promising ligands for ifenprodil site of NR2B/NMDA receptors | 1-gen-2010 | Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; De Sarro, G; Chimirri, Alba | |
SYNTHESIS AND BIOLOGICAL CHARACTERIZATION OF 3-SUBSTITUTED-1H-INDOLES AS LIGANDS OF GLUN2B-CONTAINING N-METHYL-D-ASPARTATE RECEPTORS | 1-gen-2011 | Buemi, Mariarosa; Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Giovambattista De, Sarro; Lucia, Ciranna; Chimirri, Alba | |
SYNTHESIS AND BIOLOGICAL CHARACTERIZATION OF NEW NR2B/NMDA RECEPTOR LIGANDS | 1-gen-2011 | Buemi, Mariarosa | |
DISCOVERY OF NEW INDOLE DERIVATES AS NEUROPROTECTIVE AGENTS | 1-gen-2011 | Buemi, Mariarosa; Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; R., Alajarin; J., ALVAREZ BUILLA; R., Citraro; Chimirri, Alba | |
Synthesis and Biological Characterization of 3-Substituted-1H-indoles as Ligands of GluN2B-Containing N-Methyl-d-aspartate Receptors | 1-gen-2011 | Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Russo, E; De Sarro, G; Costa, LARA TANIA; Ciranna, L; Prezzavento, O; Arena, E; Ronsisvalle, S; Bruno, Giuseppe; Chimirri, Alba | |
Rational Design and synthesis of new GluN2B/NMDA receptor ligands as neuroprotective agents. | 1-gen-2012 | Buemi, Mariarosa | |
Identification of 3-substituted-1H-indoles as ligands of GluN2B containing N-methyl-D-aspartate receptors | 1-gen-2012 | Ferro, Stefania; Buemi, Mariarosa; Gitto, Rosaria; DE LUCA, Laura; Russo, E.; Ciranna, L.; Chimirri, Alba | |
Synthesis and Biological Characterization of 3-Substituted-1H-indoles as Ligands of GluN2B-containing N-Methyl-D-Aspartate Receptors. Part. 2. | 1-gen-2012 | Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Russo, E; De Sarro, G; Chisari, M; Ciranna, L; Chimirri, Alba | |
Design, Synthesis and Biostructural Characterization of Carbonic Anhydrase Inhibitors | 1-gen-2013 | Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Vullo, D; Supuran, Ct; Brynda, J; Rezacova, P; Pospisilova, K; Damiano, F; Chimirri, Alba | |
Indole derivatives as dual-effective agents for the treatment of neurodegenerative diseases: Synthesis, biological evaluation, and molecular modeling studies | 1-gen-2013 | Maria Rosa, Buemi; Laura, De Luca; Alba, Chimirri; Stefania, Ferro; Rosaria, Gitto; Julio, Alvarez-Builla; Ramon, Alajarin | |
Design and optimization of isoquinoline-sulfonamides as potent and selective inhibitors of human carbonic anhydrase VII | 1-gen-2014 | Bruno, Elvira; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Ceruso, Mariangela; Supuran, Claudiu T.; Gitto, Rosaria | |
Synthesis, Modelling and Biological Characterization of 3-Substituted-1H-indoles as Ligands of GluN2B-containing N-Methyl-d-Aspartate Receptors | 1-gen-2014 | Rosaria Gitto;Laura De Luca;Stefania Ferro;Emilio Russo;Giovambattista De Sarro;Mariangela Chisari;Lucia Ciranna;Julio Alvarez-Builla;Ramon Alajarin;Maria Rosa Buemi;Alba Chimirri | |
Targeting GluN2B-containing N-Methyl-D-aspartate receptors: design, synthesis, and binding affinity evaluation of novel 3-substituted indoles. | 1-gen-2014 | Buemi MR;De Luca L;Ferro S;Gitto R | |
From NMDA receptor antagonists to discovery of selective σ2 receptor ligands | 1-gen-2014 | Rosaria Gitto;Laura De Luca;Stefania Ferro;Angela Scala;Simone Ronsisvalle;Carmela Parenti;Orazio Prezzavento;Maria Rosa Buemi;Alba Chimirri | |
Serendipitous discovery of indole derivatives as potent tyrosinase inhibitors | 1-gen-2015 | Gitto, Rosaria; Buemi, Mariarosa; DE LUCA, Laura; Certo, Giovanna; Germano', Maria Paola; Rapisarda, Antonio; Ferro, Stefania | |
Synthesis and biological characterization of novel potent arylsulfonamides as human carbonic anhydrase inhibitors (hCAIs) targeting central nervous system | 1-gen-2015 | Bruno, Elvira; Buemi, Mariarosa; DE LUCA, Laura; Ferro, Stefania; Ceruso, Mariangela; Supuran, Claudiu T.; Gitto, Rosaria |
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