Sfoglia per Autore  

Opzioni
Mostrati risultati da 1 a 15 di 15
Titolo Data di pubblicazione Autore(i) File
Direct and chemoselective synthesis α,α-difluoromethylketones under transfer of (CHF2) unit 1-gen-2019 Citarella, A.; Miele, M.; Micale, N.; Pace, V.
Direct and chemoselective transfer of the difluoromethyl (CHF2) unit into carbon-electrophiles under nucleophilic regime 1-gen-2019 Citarella, A.; Miele, M.; Micale, N.; Pace, V.
Hydroxamic Acid-Based Histone Deacetylase (HDAC) Inhibitors Bearing a Pyrazole Scaffold and a Cinnamoyl Linker 1-gen-2019 Zagni, Chiara; Citarella, Andrea; Oussama, Mahjoub; Rescifina, Antonio; Maugeri, Alessandro; Navarra, Michele; Scala, Angela; Piperno, Anna; Micale, Nicola
Direct and Chemoselective Synthesis of Tertiary Difluoroketones via Weinreb Amide Homologation with a CHF2-Carbene Equivalent 1-gen-2019 Miele, M.; Citarella, A.; Micale, N.; Holzer, W.; Pace, V.
Chemoselective Homologation-Deoxygenation Strategy Enabling the Direct Conversion of Carbonyls into (n+1)-Halomethyl-Alkanes 1-gen-2020 Miele, Margherita; Citarella, Andrea; Langer, Thierry; Urban, Ernst; Zehl, Martin; Holzer, Wolfgang; Ielo, Laura; Pace, Vittorio
Peptide-based α,α-Difluoromethyl Ketone as new inhibitor of Pathogenic Coronavirus Mpro 1-gen-2020 Citarella, Andrea; Gentile, Davide; Rescifina, Antonio; Pace, Vittorio; Piperno, Anna; Micale, Nicola
Peptidyl fluoromethyl ketones and their applications in medicinal chemistry 1-gen-2020 Micale, Nicola; Citarella, Andrea
Hydrogels for the Delivery of Plant-Derived (Poly)Phenols 1-gen-2020 Micale, Nicola; Citarella, Andrea; Molonia, Maria Sofia; Speciale, Antonio; Cimino, Francesco; Saija, Antonella; Cristani, Mariateresa
Fluorine-based pseudopeptides from halocarbene transfer reaction: synthesis and biological perspectives 1-gen-2020 Citarella, Andrea; Miele, Margherita; Pace, Vittorio; Micale, Nicola
Pseudo-Dipeptide Bearing ,-Difluoromethyl Ketone Moiety as ElectrophilicWarhead with Activity against Coronaviruses 1-gen-2021 Citarella, Andrea; Gentile, Davide; Rescifina, Antonio; Piperno, Anna; Mognetti, Barbara; Gribaudo, Giorgio; Sciortino, Maria Teresa; Holzer, Wolfgang; Pace, Vittorio; Micale, Nicola
SARS-CoV-2 Mpro: A Potential Target for Peptidomimetics and Small-Molecule Inhibitors 1-gen-2021 Citarella, Andrea; Scala, Angela; Piperno, Anna; Micale, Nicola
Natural product-based hybrids as potential candidates for the treatment of cancer: Focus on curcumin and resveratrol 1-gen-2021 Micale, N.; Molonia, M. S.; Citarella, A.; Cimino, F.; Saija, A.; Cristani, M.; Speciale, A.
NUCLEOPHILIC α-SUBSTITUTED ORGANOMETALLIC REAGENTS IN HOMOLOGATION CHEMISTRY: SYNTHETIC APPLICATIONS AND BIOLOGICAL PERSPECTIVES 13-gen-2021 Citarella, Andrea
Synthesis, computational investigation and biological evaluation of α,α-difluoromethyl ketones embodying pyrazole and isoxazole nuclei as COX inhibitors 1-gen-2022 Citarella, Andrea; Ielo, Laura; Stagno, Claudio; Cristani, Mariateresa; Muscara', Claudia; Pace, Vittorio; Micale, Nicola
Novel Class of Proteasome Inhibitors: In Silico and In Vitro Evaluation of Diverse Chloro(trifluoromethyl)aziridines 1-gen-2022 Ielo, Laura; Patamia, Vincenzo; Citarella, Andrea; Efferth, Thomas; Shahhamzehei, Nasim; Schirmeister, Tanja; Stagno, Claudio; Langer, Thierry; Rescifina, Antonio; Micale, Nicola; Pace, Vittorio
Mostrati risultati da 1 a 15 di 15
Legenda icone

  •  file ad accesso aperto
  •  file disponibili sulla rete interna
  •  file disponibili agli utenti autorizzati
  •  file disponibili solo agli amministratori
  •  file sotto embargo
  •  nessun file disponibile