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Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases 1-gen-2018 De Luca, Laura; Mancuso, Francesca; Ferro, Stefania; Buemi, Maria Rosa; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria
Simulated human digestion of N1-aryl-2-arylthioacetamidobenzimidazoles and their activity against Herpes-simplex virus 1 in vitro 1-gen-2019 Mandalari, Giuseppina; Bisignano, Carlo; Smeriglio, Antonella; Denaro, Marcella; Musarra-Pizzo, Maria; Pennisi, Rosamaria; Mancuso, Francesca; Ferro, Stefania; Trombetta, Domenico; Monforte, Anna Maria; Sciortino, Maria Teresa; De Luca, Laura
Seeking new approach for therapeutic treatment of cholera disease via inhibition of bacterial carbonic anhydrases: experimental and theoretical studies for sixteen benzenesulfonamide derivatives 1-gen-2019 Gitto, R.; De Luca, L.; Mancuso, Francesca; Del Prete, S.; Vullo, D.; Supuran, CLAUDIU TRANDAFIR; Capasso, C.
Exploring structural properties of potent human carbonic anhydrase inhibitors bearing a 4-(cycloalkylamino-1-carbonyl)benzenesulfonamide moiety 1-gen-2019 Buemi, Maria Rosa; Di Fiore, Anna; De Luca, Laura; Angeli, Andrea; Mancuso, Francesca; Ferro, Stefania; Monti, Simona Maria; Buonanno, Martina; Russo, Emilio; De Sarro, Giovanbattista; De Simone, Giuseppina; Supuran, Claudiu T; Gitto, Rosaria
P158-DEVELOPMENT OF FLEXIBLE ARYLSULFONAMIDES AS POTENTIAL MULTITARGET ANTICANCER AGENTS 1-gen-2020 Bucolo, Federica; Mancuso, Francesca; DE LUCA, Laura; Angeli, Andrea; Supuran, Claudiu T.; Gitto, Rosaria
Transition‐Metal‐Mediated versus Tetrazine‐Triggered Bioorthogonal Release Reactions: Direct Comparison and Combinations Thereof 1-gen-2020 Mancuso, Francesca; Rahm, Michal; Dzijak, Rastislav; Mertlíková‐kaiserová, Helena; Vrabel, Milan
In Silico-Guided Identification of New Potent Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae 1-gen-2020 Mancuso, Francesca; De Luca, Laura; Angeli, Andrea; Berrino, Emanuela; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria
Synthesis, computational studies and assessment of in vitro inhibitory activity of umbelliferon-based compounds against tumour-associated carbonic anhydrase isoforms IX and XII 1-gen-2020 Mancuso, Francesca; De Luca, Laura; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria
Looking toward the Rim of the Active Site Cavity of Druggable Human Carbonic Anhydrase Isoforms 1-gen-2020 Mancuso, F.; Di Fiore, A.; De Luca, L.; Angeli, A.; Monti, S. M.; De Simone, G.; Supuran, C. T.; Gitto, R.
Effetto in vitro di derivati di 1-(1H-indol-3-il) etanone e propan-1-one su Candida spp. and Aspergillus niger 1-gen-2021 Gervasi, Teresa; Ginestra, Giovanna; Mancuso, Francesca; Barreca, Davide; DE LUCA, Laura; Mandalari, Giuseppina
The In Vitro Potential of 1-(1H-indol-3-yl) Derivatives against Candida spp. and Aspergillus niger as Tyrosinase Inhibitors 1-gen-2021 Gervasi, Teresa; Ginestra, Giovanna; Mancuso, Francesca; Barreca, Davide; De Luca, Laura; Mandalari, Giuseppina
The In Vitro Potential of 1-(1H-indol-3-yl) Derivatives against Candida spp. and Aspergillus niger as Tyrosinase Inhibitors 1-gen-2021 Gervasi, T.; Ginestra, G.; Mancuso, F.; Barreca, D.; De Luca, L.; Mandalari, G.
4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae 1-gen-2021 Mancuso, F.; De Luca, L.; Bucolo, F.; Vrabel, M.; Angeli, A.; Capasso, C.; Supuran, C. T.; Gitto, R.
Targeting Carbonic Anhydrases (CAs): Rational Design, Synthesis, Structural Studies and Biochemical Evaluation 8-gen-2021 Mancuso, Francesca
Tetraamino-dihydroxy-tetraoxacalix[4]arene as a versatile paraquat receptor 1-gen-2022 Crisafulli, Daniele; Mancuso, Francesca; Milone, Marco; Irto, Anna; Cigala, Rosalia Maria; Lando, Gabriele; Pisagatti, Ilenia; Notti, Anna; Gattuso, Giuseppe
One oxacalix[4]arene, seven protonated species: a macrocyclic receptor for paraquat 1-gen-2022 Crisafulli, Daniele; Mancuso, Francesca; Milone, Marco; Irto, Anna; Cigala, Rosalia Maria; Lando, Gabriele; Pisagatti, Ilenia; Notti, Anna; Gattuso, Giuseppe
The in vitro potential of novel carbonic anhydrase Inhibitors against candida spp 1-gen-2022 Gitto, Rosaria; Mancuso, Francesca; Bucolo, Federica; Gervasi, Teresa; Ginestra, Giovanna; DE LUCA, Laura; Mandalari, Giuseppina
Proton transfer mediated recognition of amines by ionizable macrocyclic receptors 1-gen-2022 Gattuso, Giuseppe; Crisafulli, Daniele; Milone, Marco; Mancuso, Francesca; Pisagatti, Ilenia; Notti, Anna; Parisi, Melchiorre F.
Tetracationic-to-dianionic tetraamino-dihydroxy-tetraoxacalix[4]arene: A paraquat receptor for all seasons 1-gen-2022 Mancuso, Francesca; Crisafulli, Daniele; Milone, Marco; Irto, Anna; Cigala, Rosalia Maria; Lando, Gabriele; Pisagatti, Ilenia; Notti, Anna; Gattuso, Giuseppe
Synthesis and biological evaluation of sulfonamide-based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae 1-gen-2022 Mancuso, F.; Angeli, A.; De Luca, V.; Bucolo, F.; De Luca, L.; Capasso, C.; Supuran, C. T.; Gitto, R.
Mostrati risultati da 1 a 20 di 23
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