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Non-covalent immunoproteasome inhibitors induce cell cycle arrest in multiple myeloma cells 1-gen-2019 Ettari, R.; Pallio, G.; Pizzino, G.; Irrera, N.; Zappalà, M.; Maiorana, S.; Di Chio, C.; Altavilla, D.; Squadrito, F.; Bitto, A.
Development of novel benzodiazepine-based peptidomimetics as inhibitors of rhodesain of Trypanosoma brucei rhodesiense 1-gen-2020 DI CHIO, Carla; Previti, Santo; Cosconati, Sandro; Zappala', Maria; Ettari, Roberta
Discovery of novel peptidomimetics containing a benzodiazepine scaffold as inhibitors of rhodesain of Trypanosoma brucei rhodesiense 1-gen-2020 DI CHIO, Carla; Previti, Santo; Amendola, Giorgio; Cosconati, Sandro; Zappala', Maria; Ettari, Roberta
Discovery of novel antitrypanosomal agents: design, synthesis of novel benzodiazepine-based peptidomimetics targeting rhodesain, the main cysteine protease of Trypanosoma brucei rhodesiense 1-gen-2020 DI CHIO, Carla; Zappala', Maria; Ettari, Roberta
Drug synergism: studies of combination of RK-52 and curcumin against rhodesain of Trypanosoma brucei rhodesiense 1-gen-2020 Ettari, R.; Previti, S.; Di Chio, C.; Maiorana, S.; Allegra, A.; Schirmeister, T.; Zappalà, M.
Development of Novel Benzodiazepine-Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense 1-gen-2020 DI CHIO, Carla; Previti, Santo; Amendola, Giorgio; Cosconati, Sandro; Schirmeister, Tanja; Zappala', Maria; Ettari, Roberta
Development of peptidyl Michael acceptors for S3 pocket investigation of rhodesain, cysteine protease of Trypanosoma brucei rhodesiense 1-gen-2021 Previti, Santo; Ettari, Roberta; DI CHIO, Carla; Cosconati, Sandro; Amendola, Giorgio; Schirmeister, Tanja; Zappala', Maria
Development of novel dipeptide nitriles as inhibitors of rhodesain of Trypanosoma brucei hodesiense 1-gen-2021 Di Chio, C.; Previti, S.; Ravichandran, R.; Cosconati, S.; Schirmeister, T.; Zappalà, Maria; Ettari, R.
Design and NMR conformational analysis in solution of β5i-selective inhibitors of immunoproteasome 1-gen-2021 Rotondo, Archimede; Zappala', Maria; Previti, Santo; DI CHIO, Carla; Allegra, Alessandro; Ettari, Roberta
Lead discovery of SARS-CoV-2 main protease inhibitors through covalent docking-based virtual screening 1-gen-2021 Amendola, Giorgio; Ettari, Roberta; Previti, Santo; DI CHIO, Carla; Messere, Anna; Di Maro, Salvatore; Hammerschmidt, Stefan J.; Zimmer, Collin; Zimmermann, Robert A.; Schirmeister, Tanja; Zappala', Maria; Sandro Cosconati, And
Falcipain-2 and Falcipain-3 Inhibitors as Promising Antimalarial Agents 1-gen-2021 Ettari, Roberta; Previti, Santo; Di Chio, Carla; Zappala', Maria
Design, synthesis and biological evaluation of novel bioactive molecules for the treatment of protozoan and human diseases 18-nov-2021 DI CHIO, Carla
Synthesis and cytotoxicity of diarylpentanoids against sensitive CCRF-CEM and multidrug-resistant CEM/ADR5000 leukemia cells 1-gen-2022 DI CHIO, Carla; Zhou, Min; Efferth, Thomas; Schirmeister, Tanja; Zappala', Maria; Ettari, Roberta
Development of Urea-Bond-Containing Michael Acceptors as Antitrypanosomal Agents Targeting Rhodesain 1-gen-2022 Previti, Santo; Ettari, Roberta; Calcaterra, Elsa; DI CHIO, Carla; Ravichandran, Rahul; Zimmer, Collin; Hammerschmidt, Stefan; Wagner, Annika; Bogacz, Marta; Cosconati, Sandro; Schirmeister, Tanja; Zappala', Maria
Development of novel dipeptide nitriles as inhibitors of rhodesain of Trypanosoma brucei rhodesiense 1-gen-2022 DI CHIO, Carla; Previti, Santo; Amendola, Giorgio; Ravichandran, Rahul; Wagner, Annika; Cosconati, Sandro; A Hellmich, Ute; Schirmeister, Tanja; Zappalà, Maria; Ettari, Roberta
Drug combination studies of the dipeptide nitrile CD24 with curcumin: a new strategy to synergistically inhibit rhodesain of trypanosoma brucei rhodesiense 1-gen-2022 DI CHIO, Carla; Previti, Santo; DE LUCA, Fabiola; Bogacz, Marta; Zimmer, Collin; Wagner, Annika; Schirmeister, Tanja; Zappala', Maria; Ettari, Roberta
Dual inhibition of parasitic targets: a valuable strategy to treat malaria and neglected tropical diseases 1-gen-2022 Previti, Santo; DI CHIO, Carla; Ettari, Roberta; Zappala', Maria
Development of reduced peptide bond pseudopeptide Michael acceptors for the treatment of Human African Trypanosomiasis 1-gen-2022 Previti, Santo; Ettari, Roberta; DI CHIO, Carla; Ravichandran, Rahul; Bogacz, Marta; Hellmich, Ute A.; Schirmeister, Tanja; Cosconati, Sandro; Zappala', Maria
Development of isoquinolinone derivatives as immunoproteasome inhibitors. 1-gen-2022 Ettari, R.; Iraci, N.; Di Chio, C.; Previti, S.; Danze', M.; Zappala', M
Drug combination studies of PS-1 and quercetin against rhodesain of Trypanosoma brucei rhodesiense 1-gen-2022 DI CHIO, Carla; Previti, Santo; DE LUCA, Fabiola; Allegra, Alessandro; Zappala', Maria; Ettari, Roberta
Mostrati risultati da 1 a 20 di 26
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