Sfoglia per Autore
Synthesis and antitumor activity evaluation of Delta(2)-1,2,4- oxadiazoline derivatives
1996-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Rao, A; Zappala', Maria
Synthesis and in vitro antitumor activity evaluation of 9- substituted 1,2,3,4-tetrahydrocarbazoles
1996-01-01 Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Rizzo, M.
1-fluoromethyl-1-methyl-1H,3H-thiazolo-[3,4-a]benzimidazole
1996-01-01 BRUNO G; CHIMIRRI A; MONFORTE AM; F. NICOLO'; SCOPELLITI R
Substituent effects on the enantioselective retention of anti- HIV 5-aryl-Delta(2)-1,2,4-oxadiazolines on R,R-DACH-DNB chiral stationary phase
1996-01-01 Altomare, C; Cellamare, S; Carotti, A; Barreca, Ml; Chimirri, Alba; Monforte, Anna Maria; Gasparrini, F; Villani, C; Cirilli, M; Mazza, F.
Anti-HIV agents .4. Synthesis and in vitro anti-HIV activity of novel 1-(2,6-difluorophenyl)-1H,3H-thiazolo[3,4- a]benzimidazoles
1996-01-01 Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Scopelliti, R.
1-[3,5-bis(trifluoromethyl)phenyl]-1H,3H-thiazolo[3,4- a]benzimidazole
1996-01-01 Bruno, Giuseppe; Monforte, Anna Maria; Nicolo', Francesco; Scopelliti, R; Zappala', Maria
Structural features and anti-human immunodeficiency virus (HIV) activity of the isomers of 1-(2',6'-difluorophenyl)-1H,3H- thiazolo[3,4-a]benzimidazole, a potent non-nucleoside HIV-1 reverse transcriptase inhibitor
1997-01-01 Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Witvrouw, M.; Jonckeere, H.; Balzarini, J.; Declercq, E.
1-Aryl-1H,3H-thiazolo[3,4-a]benzimidazole derivatives
1997-01-01 Bruno, Giuseppe; Chimirri, Alba; Monforte, Anna Maria; Nicolo', Francesco; Scopelliti, R.
Anti-HIV agents. V. Synthesis, structure and in vitro anti-HIV activity of novel 1H,3H-naphtho[2 ',3 ': 4,5]imidazo[1,2- c]thiazoles
1997-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A.; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Scopelliti, R.
TBZ-analoghi inibitori non nucleosidici della HIV-RT
1998-01-01 A., Chimirri; E., DE CLERQ; Grasso, Silvana; Monforte, Anna Maria; P., Monforte; A., Rao; Zappala', Maria
Synthesis, structure and in vitro anti-human immunodeficiency virus activity of novel 3-methyl-1H,3H-thiazolo[3,4- a]benzimidazoles
1998-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Pannecouque, C; Witvrouw, M; DE CLERCQ, E.
Synthesis and biological activity of novel non-nucleoside HIV-1 RT inhibitors
1998-01-01 A., Chimirri; E., DE CLERCQ; Grasso, Silvana; Monforte, Anna Maria; P., Monforte; C., Pannecoque; A., Rao; M., Witrouw; Zappala', Maria
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system
1999-01-01 Chimirri, Alba; DE CLERCQ, E.; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Pannecouque, C.; Rao, A.; Witvrouw, M.; Zappala', Maria
Synthesis and anti-HIV activity of TBZ structurally-related 1,2-substituted benzimidazoles
1999-01-01 Chimirri, A.; Monforte, Anna Maria; P., Monforte; L., Musumeci; A., Rao; Zappala', Maria; C., Pannecouque; M., Witvrouw; E., DE CLERCQ
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system
1999-01-01 Chimirri, Alba; E., DE CLERCQ; Grasso, Silvana; Monforte, Anna Maria; P., Monforte; C., Pannecouque; A., Rao; M., Witvrouw; Zappala', Maria
Synthesis and anti-HIV activity of TBZ structurally-related 1,2-substituted benzimidazoles
1999-01-01 A., Chimirri; Monforte, Anna Maria; P., Monforte; L., Musumeci; A., Rao; Zappala', Maria; C., Pannecouque; M., Witvrouw; E., DE CLERCQ
Comparative molecular field analysis (CoMFA) and docking studies of non-nucleoside HIV-1 RT inhibitors (NNIs)
1999-01-01 Barreca, Maria Letizia; Carotti, A; Carrieri, A; Chimirri, Alba; Monforte, Anna Maria; Calace, Mp; Rao, Angela
Synthesis and biological activity of novel 1H,3H-thiazolo[3,4- a] benzimidazoles: non-nucleoside human immunodeficiency virus type 1 reverse transcriptase inhibitors
1999-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Rao, Angela; Zappala', Maria; Monforte, Anna Maria; Pannecouque, C; Witvrouw, M; Balzarini, J; DE CLERCQ, E.
Synthesis, structural features and anti-HIV activity of TBZ analogues.
1999-01-01 A., Chimirri; Monforte, Anna Maria; P., Monforte; L., Musumeci; A., Rao; Zappala', Maria; M., Witvrouw; E., DE CLERCQ
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system
1999-01-01 A., Chimirri; E., DE CLERCQ; Grasso, Silvana; Monforte, Anna Maria; P., Monforte; C., Pannecouque; A., Rao; M., Witvrouw; Zappala', Maria
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and antitumor activity evaluation of Delta(2)-1,2,4- oxadiazoline derivatives | 1-gen-1996 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Rao, A; Zappala', Maria | |
Synthesis and in vitro antitumor activity evaluation of 9- substituted 1,2,3,4-tetrahydrocarbazoles | 1-gen-1996 | Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Rizzo, M. | |
1-fluoromethyl-1-methyl-1H,3H-thiazolo-[3,4-a]benzimidazole | 1-gen-1996 | BRUNO G; CHIMIRRI A; MONFORTE AM; F. NICOLO'; SCOPELLITI R | |
Substituent effects on the enantioselective retention of anti- HIV 5-aryl-Delta(2)-1,2,4-oxadiazolines on R,R-DACH-DNB chiral stationary phase | 1-gen-1996 | Altomare, C; Cellamare, S; Carotti, A; Barreca, Ml; Chimirri, Alba; Monforte, Anna Maria; Gasparrini, F; Villani, C; Cirilli, M; Mazza, F. | |
Anti-HIV agents .4. Synthesis and in vitro anti-HIV activity of novel 1-(2,6-difluorophenyl)-1H,3H-thiazolo[3,4- a]benzimidazoles | 1-gen-1996 | Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Scopelliti, R. | |
1-[3,5-bis(trifluoromethyl)phenyl]-1H,3H-thiazolo[3,4- a]benzimidazole | 1-gen-1996 | Bruno, Giuseppe; Monforte, Anna Maria; Nicolo', Francesco; Scopelliti, R; Zappala', Maria | |
Structural features and anti-human immunodeficiency virus (HIV) activity of the isomers of 1-(2',6'-difluorophenyl)-1H,3H- thiazolo[3,4-a]benzimidazole, a potent non-nucleoside HIV-1 reverse transcriptase inhibitor | 1-gen-1997 | Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Witvrouw, M.; Jonckeere, H.; Balzarini, J.; Declercq, E. | |
1-Aryl-1H,3H-thiazolo[3,4-a]benzimidazole derivatives | 1-gen-1997 | Bruno, Giuseppe; Chimirri, Alba; Monforte, Anna Maria; Nicolo', Francesco; Scopelliti, R. | |
Anti-HIV agents. V. Synthesis, structure and in vitro anti-HIV activity of novel 1H,3H-naphtho[2 ',3 ': 4,5]imidazo[1,2- c]thiazoles | 1-gen-1997 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A.; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Scopelliti, R. | |
TBZ-analoghi inibitori non nucleosidici della HIV-RT | 1-gen-1998 | A., Chimirri; E., DE CLERQ; Grasso, Silvana; Monforte, Anna Maria; P., Monforte; A., Rao; Zappala', Maria | |
Synthesis, structure and in vitro anti-human immunodeficiency virus activity of novel 3-methyl-1H,3H-thiazolo[3,4- a]benzimidazoles | 1-gen-1998 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Pannecouque, C; Witvrouw, M; DE CLERCQ, E. | |
Synthesis and biological activity of novel non-nucleoside HIV-1 RT inhibitors | 1-gen-1998 | A., Chimirri; E., DE CLERCQ; Grasso, Silvana; Monforte, Anna Maria; P., Monforte; C., Pannecoque; A., Rao; M., Witrouw; Zappala', Maria | |
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system | 1-gen-1999 | Chimirri, Alba; DE CLERCQ, E.; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Pannecouque, C.; Rao, A.; Witvrouw, M.; Zappala', Maria | |
Synthesis and anti-HIV activity of TBZ structurally-related 1,2-substituted benzimidazoles | 1-gen-1999 | Chimirri, A.; Monforte, Anna Maria; P., Monforte; L., Musumeci; A., Rao; Zappala', Maria; C., Pannecouque; M., Witvrouw; E., DE CLERCQ | |
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system | 1-gen-1999 | Chimirri, Alba; E., DE CLERCQ; Grasso, Silvana; Monforte, Anna Maria; P., Monforte; C., Pannecouque; A., Rao; M., Witvrouw; Zappala', Maria | |
Synthesis and anti-HIV activity of TBZ structurally-related 1,2-substituted benzimidazoles | 1-gen-1999 | A., Chimirri; Monforte, Anna Maria; P., Monforte; L., Musumeci; A., Rao; Zappala', Maria; C., Pannecouque; M., Witvrouw; E., DE CLERCQ | |
Comparative molecular field analysis (CoMFA) and docking studies of non-nucleoside HIV-1 RT inhibitors (NNIs) | 1-gen-1999 | Barreca, Maria Letizia; Carotti, A; Carrieri, A; Chimirri, Alba; Monforte, Anna Maria; Calace, Mp; Rao, Angela | |
Synthesis and biological activity of novel 1H,3H-thiazolo[3,4- a] benzimidazoles: non-nucleoside human immunodeficiency virus type 1 reverse transcriptase inhibitors | 1-gen-1999 | Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Rao, Angela; Zappala', Maria; Monforte, Anna Maria; Pannecouque, C; Witvrouw, M; Balzarini, J; DE CLERCQ, E. | |
Synthesis, structural features and anti-HIV activity of TBZ analogues. | 1-gen-1999 | A., Chimirri; Monforte, Anna Maria; P., Monforte; L., Musumeci; A., Rao; Zappala', Maria; M., Witvrouw; E., DE CLERCQ | |
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system | 1-gen-1999 | A., Chimirri; E., DE CLERCQ; Grasso, Silvana; Monforte, Anna Maria; P., Monforte; C., Pannecouque; A., Rao; M., Witvrouw; Zappala', Maria |
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