Sfoglia per Autore
New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists
2005-01-01 A., Pellicanò; Micale, Nicola; Grasso, Silvana; Zappala', Maria; C., DE MICHELI; G., Ferreri; G., DE SARRO; F. S., Menniti
Novel peptidomimetic cysteine protease inhibitors as antimalarial agents
2005-01-01 Micale, Nicola; Ettari, Roberta; Grasso, Silvana; Zappala', Maria; Chishti, A. H.; Kozikowski, A. P.
New 2,3-benzodiazepines as noncompetitive AMPA receptor antagonists.
2005-01-01 Grasso, Silvana; Zappala', Maria; G., Postorino; A., Pellicano'; Micale, Nicola; C., DE MICHELI; G., Grazioso; F. S., Menniti
Ligandi non competitivi del recettore AMPA del glutammato: sintesi e valutazione in vitro.
2005-01-01 A., Pellicanò; Zappala', Maria; G., Postorino; Micale, Nicola; Grasso, Silvana; F. S., Menniti
Synthesis of 2-semicarbazonomethyl-4,5-methylenedioxyphenylacetic acids as anticonvulsant agents
2005-01-01 Micale, Nicola; Zappala', Maria; G., Zuccala'; F. S., Menniti; G., Ferreri; G., DE SARRO; Grasso, Silvana
Novel 2H-isoquinolin-3-ones cysteine protease inhibitors as potential antimalarial agents
2006-01-01 G., Postorino; T., Impala'; Micale, Nicola; Grasso, Silvana; Zappala', Maria; A. H., Chishti
Reazioni di cross metathesis: applicazione alla sintesi di peptidomimetici potenziali inibitori di falcipaina-2
2006-01-01 Ettari, Roberta; E., Nizi; M. E., DI FRANCESCO; Micale, Nicola; Grasso, Silvana; Zappala', Maria
Synthesis of constrained dipeptide mimics containing the benzodiazepine scaffold
2006-01-01 Micale, Nicola; Ettari, Roberta; Grasso, Silvana; Zappala', Maria; A. P., Kozikowski
New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists
2006-01-01 Zappala', Maria; A., Pellicano'; Micale, Nicola; F. S., Menniti; G., Ferreri; G., DE SARRO; Grasso, Silvana; C., DE MICHELI
Novel peptidomimetic cysteine protease inhibitors as potential antimalarial agents
2006-01-01 Micale, Nicola; Kozikowski, Alan P.; Ettari, Roberta; Grasso, Silvana; Zappala', Maria; Jeong, Jong Jin; Kumar, Ajay; Hanspal, Manjit; Chishti, Athar H.
2,3-Benzodiazepine-based noncompetitive AMPAR antagonists: design, synthesis, binding affinity and mechanism of inhibition of the GluR2Qflip homomeric receptor channel
2006-01-01 Grasso, Silvana; Zappala', Maria; Micale, Nicola; G., Postorino; A., Pellicano'; S., Colleoni; A., Cagnotto; T., Mennini; M., Ritz; G., Li; L., Niu
Synthesis, chiral resolution and enantiopharmacology of a potent 2,3-benzodiazepine as noncompetitive AMPA receptor antagonist
2006-01-01 Zappala', Maria; G., Postorino; Micale, Nicola; S., Caccamese; N., Parrinello; G., Grazioso; G., Roda; F. S., Menniti; G., DE SARRO; Grasso, Silvana
Synthesis of novel 3-alkylcarbamoyl-2-aryl-1,2-dihydro-6,7-methylenedioxy-3H-quinazolin-4-ones as anticonvulsant agents
2006-01-01 N. MICALE; G. POSTORINO; GRASSO S.; M. ZAPPALA'; G. ZUCCALA'; G. FERRERI; G. DE SARRO
Enantioselective recognition of 2,3-benzodiazepin-4-one derivatives with anticonvulsant activity on several polysaccharide chiral stationary phases
2006-01-01 CALABRO ML; RANERI D; TOMMASINI S; FICARRA R; ALCARO S; GALLELLI A; MICALE N; ZAPPALA M; FICARRA P.
Chloro-substituted Hoveyda-Grubbs ruthenium carbene: investigation of electronic effects
2007-01-01 Ettari, Roberta; Micale, Nicola
Strategie per lo sviluppo di peptidomimetici: design di inbitori di cistein-proteasi
2007-01-01 Micale, Nicola
Cross-metathesis reactions applications to the synthesis of peptidomimetics as potent falcipain-2 inhibitors
2007-01-01 Ettari, Roberta; E., Nizi; M. E., DI FRANCESCO; R., Vi; K, ; T., Schirmeister; Micale, Nicola; Grasso, Silvana; Zappala', Maria
Development of nonpeptidic vinyl and allyl phosphonates as active-site-directed inhibitors of falcipain-2
2007-01-01 Grasso, Silvana; Ettari, Roberta; Zappala', Maria; Micale, Nicola; E., Nizi; M. E., DI FRANCESCO; R., Vicik; T., Schirmeister
Synthesis of Peptidomimetics with the Benzodiazepine Nucleus as beta-turn mimic
2007-01-01 Micale, Nicola; Ettari, Roberta
Synthesis of Peptidomimetics with the Benzodiazepine Nucleus as beta-turn mimic
2007-01-01 Micale, Nicola; Ettari, R.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists | 1-gen-2005 | A., Pellicanò; Micale, Nicola; Grasso, Silvana; Zappala', Maria; C., DE MICHELI; G., Ferreri; G., DE SARRO; F. S., Menniti | |
Novel peptidomimetic cysteine protease inhibitors as antimalarial agents | 1-gen-2005 | Micale, Nicola; Ettari, Roberta; Grasso, Silvana; Zappala', Maria; Chishti, A. H.; Kozikowski, A. P. | |
New 2,3-benzodiazepines as noncompetitive AMPA receptor antagonists. | 1-gen-2005 | Grasso, Silvana; Zappala', Maria; G., Postorino; A., Pellicano'; Micale, Nicola; C., DE MICHELI; G., Grazioso; F. S., Menniti | |
Ligandi non competitivi del recettore AMPA del glutammato: sintesi e valutazione in vitro. | 1-gen-2005 | A., Pellicanò; Zappala', Maria; G., Postorino; Micale, Nicola; Grasso, Silvana; F. S., Menniti | |
Synthesis of 2-semicarbazonomethyl-4,5-methylenedioxyphenylacetic acids as anticonvulsant agents | 1-gen-2005 | Micale, Nicola; Zappala', Maria; G., Zuccala'; F. S., Menniti; G., Ferreri; G., DE SARRO; Grasso, Silvana | |
Novel 2H-isoquinolin-3-ones cysteine protease inhibitors as potential antimalarial agents | 1-gen-2006 | G., Postorino; T., Impala'; Micale, Nicola; Grasso, Silvana; Zappala', Maria; A. H., Chishti | |
Reazioni di cross metathesis: applicazione alla sintesi di peptidomimetici potenziali inibitori di falcipaina-2 | 1-gen-2006 | Ettari, Roberta; E., Nizi; M. E., DI FRANCESCO; Micale, Nicola; Grasso, Silvana; Zappala', Maria | |
Synthesis of constrained dipeptide mimics containing the benzodiazepine scaffold | 1-gen-2006 | Micale, Nicola; Ettari, Roberta; Grasso, Silvana; Zappala', Maria; A. P., Kozikowski | |
New 7,8-ethylenedioxy-2,3-benzodiazepines as noncompetitive AMPA receptor antagonists | 1-gen-2006 | Zappala', Maria; A., Pellicano'; Micale, Nicola; F. S., Menniti; G., Ferreri; G., DE SARRO; Grasso, Silvana; C., DE MICHELI | |
Novel peptidomimetic cysteine protease inhibitors as potential antimalarial agents | 1-gen-2006 | Micale, Nicola; Kozikowski, Alan P.; Ettari, Roberta; Grasso, Silvana; Zappala', Maria; Jeong, Jong Jin; Kumar, Ajay; Hanspal, Manjit; Chishti, Athar H. | |
2,3-Benzodiazepine-based noncompetitive AMPAR antagonists: design, synthesis, binding affinity and mechanism of inhibition of the GluR2Qflip homomeric receptor channel | 1-gen-2006 | Grasso, Silvana; Zappala', Maria; Micale, Nicola; G., Postorino; A., Pellicano'; S., Colleoni; A., Cagnotto; T., Mennini; M., Ritz; G., Li; L., Niu | |
Synthesis, chiral resolution and enantiopharmacology of a potent 2,3-benzodiazepine as noncompetitive AMPA receptor antagonist | 1-gen-2006 | Zappala', Maria; G., Postorino; Micale, Nicola; S., Caccamese; N., Parrinello; G., Grazioso; G., Roda; F. S., Menniti; G., DE SARRO; Grasso, Silvana | |
Synthesis of novel 3-alkylcarbamoyl-2-aryl-1,2-dihydro-6,7-methylenedioxy-3H-quinazolin-4-ones as anticonvulsant agents | 1-gen-2006 | N. MICALE; G. POSTORINO; GRASSO S.; M. ZAPPALA'; G. ZUCCALA'; G. FERRERI; G. DE SARRO | |
Enantioselective recognition of 2,3-benzodiazepin-4-one derivatives with anticonvulsant activity on several polysaccharide chiral stationary phases | 1-gen-2006 | CALABRO ML; RANERI D; TOMMASINI S; FICARRA R; ALCARO S; GALLELLI A; MICALE N; ZAPPALA M; FICARRA P. | |
Chloro-substituted Hoveyda-Grubbs ruthenium carbene: investigation of electronic effects | 1-gen-2007 | Ettari, Roberta; Micale, Nicola | |
Strategie per lo sviluppo di peptidomimetici: design di inbitori di cistein-proteasi | 1-gen-2007 | Micale, Nicola | |
Cross-metathesis reactions applications to the synthesis of peptidomimetics as potent falcipain-2 inhibitors | 1-gen-2007 | Ettari, Roberta; E., Nizi; M. E., DI FRANCESCO; R., Vi; K, ; T., Schirmeister; Micale, Nicola; Grasso, Silvana; Zappala', Maria | |
Development of nonpeptidic vinyl and allyl phosphonates as active-site-directed inhibitors of falcipain-2 | 1-gen-2007 | Grasso, Silvana; Ettari, Roberta; Zappala', Maria; Micale, Nicola; E., Nizi; M. E., DI FRANCESCO; R., Vicik; T., Schirmeister | |
Synthesis of Peptidomimetics with the Benzodiazepine Nucleus as beta-turn mimic | 1-gen-2007 | Micale, Nicola; Ettari, Roberta | |
Synthesis of Peptidomimetics with the Benzodiazepine Nucleus as beta-turn mimic | 1-gen-2007 | Micale, Nicola; Ettari, R. |
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