Sfoglia per Autore
DEVELOPMENT OF NOVEL PEPTIDOMIMETICS CONTAINIG A VINYL SULFONE MOIETY AS PROTEASOME INHIBITORS
2010-01-01 Ettari, Roberta; Bonaccorso, Cinzia; Micale, Nicola; Tanja, Schirmeister; Grasso, Silvana; Zappala', Maria
Constrained peptidomimetics as antiplasmodial falcipain-2 inhibitors
2010-01-01 Bova, Floriana; Ettari, Roberta; Micale, Nicola; Carnovale, Caterina; Tanja, Schirmeister; Christoph, Gelhaus; Matthias, Leippe; Grasso, Silvana; Zappala', Maria
Novel peptidomimetics as antiplasmodial falcipain-2 inhibitors
2010-01-01 Bova, Floriana; Ettari, Roberta; Tanja, Schirmeister; Grasso, Silvana; Zappala', Maria; Micale, Nicola
Synthesis of novel peptidomimetics as inhibitors of protozoan cysteine proteases falcipain-2 and rhodesain
2010-01-01 R. Ettari; M. Zappalà; N. Micale; T. Schirmeister; C. Gelhaus; M. Leippe; A. Evers; S. Grasso.
Design and synthesis of novel isoxazole-based HDAC inhibitors
2010-01-01 Paola, Conti; Lucia, Tamborini; Andrea, Pinto; Laura, Sola; Ettari, Roberta; Ciro, Mercurio; Carlo De, Micheli
Falcipain-2 inhibitors
2010-01-01 Ettari, Roberta; Bova, Floriana; Zappala', Maria; Grasso, Silvana; Micale, Nicola
Design, synthesis and molecular modeling studies on peptidomimetic vinyl esters as falcipan-2 inhibitors
2011-01-01 Ettari, Roberta; Micale, Nicola; Bova, Floriana; Giovanni, Grazioso; Tanja, Schirmeister; Grasso, Silvana; Zappala', Maria
Design, synthesis and biological evaluation of peptidomimetics boronic acids targeting 20S proteasome
2011-01-01 Ettari, Roberta; Micale, Nicola; Bonaccorso, Cinzia; T., Schirmeister; Zappala', Maria; Grasso, Silvana
Mechanism of Inhibition of the GluA2 AMPA Receptor Channel Opening: The Role of 4-Methyl versus 4-Carbonyl Group on the Diazepine Ring of 2,3-Benzodiazepine Derivatives
2011-01-01 Mark, Ritz; Congzhou, Wang; Micale, Nicola; Ettari, Roberta; Li, Niu
Glutamate Binding-Site Ligands of NMDA Receptors
2011-01-01 C. Bonaccorso; N. Micale; R. Ettari; S. Grasso; M. Zappalà
Effect of mammalian SERCA inhibitors on Plasmodium falciparum growth in vitro
2011-01-01 Serena, Pulcini; Stefan, Paula; Chengguo, Xing; Ettari, Roberta; Henry M., Staines; Sanjeev, Krishna
Development of Novel Peptidomimetics Containing a VinylSulfone Moiety as Proteasome Inhibitors
2011-01-01 Ettari, Roberta; Bonaccorso, Cinzia; Micale, Nicola; Cornelia, Heindl; Tanja, Schirmeister; Calabro', Maria; Grasso, Silvana; Zappala', Maria
Peptidomimetics containing a vinyl ketone warhead as falcipain-2 inhibitors
2011-01-01 Ettari, Roberta; Zappala', Maria; Micale, Nicola; Giovanni, Grazioso; Giofre', Salvatore Vincenzo; Tanja, Schirmeister; Grasso, Silvana
Formation of 3-Aminofuran-2-(5H)-ones and 3-Amino-1H-pyrrole-2,5-diones by Rearrangement of Isoxazolidines
2011-01-01 Iannazzo, Daniela; Carnovale, Caterina; Giofre', Salvatore Vincenzo; Ettari, Roberta; Romeo, Giovanni; Romeo, Roberto; Giuseppe, Lanza; Ugo, Chiacchio
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF PEPTIDOMIMETIC FALCIPAIN-2 INHIBITORS AS ANTIMALARIAL AGENTS
2012-01-01 Micale, Nicola; Ettari, Roberta; T., Schirmeister; G., Grazioso; Grasso, Silvana; Zappala', Maria
Novel peptidomimetic inhibitors, containing a 1,4-benzodiazepine scaffold, for treatment of neglected tropical diseases
2012-01-01 Ettari, Roberta; A., Pinto; L., Tamborini; I. C., Angelo; Grasso, Silvana; C., De Micheli
Synthesis and Molecular Modeling Studies of Derivatives of a Highly Potent Peptidomimetic Vinyl Ester as Falcipain-2 Inhibitors
2012-01-01 Ettari, Roberta; Micale, Nicola; Giovanni, Grazioso; Bova, Floriana; Tanja, Schirmeister; Grasso, Silvana; Zappala', Maria
Development of peptidomimetic boronates as proteasome inhibitors
2012-01-01 Micale, Nicola; Ettari, Roberta; C., Di Giovanni; A., Lavecchia; Scarbaci, Kety; V., Troiano; Grasso, Silvana; E., Novellino; T., Schirmeister; Zappala', Maria
Mechanism of falcipain-2 inhibition by α,β-unsaturated benzo[1,4]diazepin-2-one methyl ester
2012-01-01 Grazioso, G; Legnani, L; Toma, L; Ettari, Roberta; Micale, Nicola; De Micheli, C.
Identification of a new series of non-covalent proteasome inhibitors with selectivity for β5-subunits
2013-01-01 Scarbaci, Kety; Troiano, V.; Micale, Nicola; Ettari, Roberta; Lavecchia, A.; Di Giovanni, C.; Grasso, Silvana; Novellino, E.; Schirmeister, T.; Zappala', Maria
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
DEVELOPMENT OF NOVEL PEPTIDOMIMETICS CONTAINIG A VINYL SULFONE MOIETY AS PROTEASOME INHIBITORS | 1-gen-2010 | Ettari, Roberta; Bonaccorso, Cinzia; Micale, Nicola; Tanja, Schirmeister; Grasso, Silvana; Zappala', Maria | |
Constrained peptidomimetics as antiplasmodial falcipain-2 inhibitors | 1-gen-2010 | Bova, Floriana; Ettari, Roberta; Micale, Nicola; Carnovale, Caterina; Tanja, Schirmeister; Christoph, Gelhaus; Matthias, Leippe; Grasso, Silvana; Zappala', Maria | |
Novel peptidomimetics as antiplasmodial falcipain-2 inhibitors | 1-gen-2010 | Bova, Floriana; Ettari, Roberta; Tanja, Schirmeister; Grasso, Silvana; Zappala', Maria; Micale, Nicola | |
Synthesis of novel peptidomimetics as inhibitors of protozoan cysteine proteases falcipain-2 and rhodesain | 1-gen-2010 | R. Ettari; M. Zappalà; N. Micale; T. Schirmeister; C. Gelhaus; M. Leippe; A. Evers; S. Grasso. | |
Design and synthesis of novel isoxazole-based HDAC inhibitors | 1-gen-2010 | Paola, Conti; Lucia, Tamborini; Andrea, Pinto; Laura, Sola; Ettari, Roberta; Ciro, Mercurio; Carlo De, Micheli | |
Falcipain-2 inhibitors | 1-gen-2010 | Ettari, Roberta; Bova, Floriana; Zappala', Maria; Grasso, Silvana; Micale, Nicola | |
Design, synthesis and molecular modeling studies on peptidomimetic vinyl esters as falcipan-2 inhibitors | 1-gen-2011 | Ettari, Roberta; Micale, Nicola; Bova, Floriana; Giovanni, Grazioso; Tanja, Schirmeister; Grasso, Silvana; Zappala', Maria | |
Design, synthesis and biological evaluation of peptidomimetics boronic acids targeting 20S proteasome | 1-gen-2011 | Ettari, Roberta; Micale, Nicola; Bonaccorso, Cinzia; T., Schirmeister; Zappala', Maria; Grasso, Silvana | |
Mechanism of Inhibition of the GluA2 AMPA Receptor Channel Opening: The Role of 4-Methyl versus 4-Carbonyl Group on the Diazepine Ring of 2,3-Benzodiazepine Derivatives | 1-gen-2011 | Mark, Ritz; Congzhou, Wang; Micale, Nicola; Ettari, Roberta; Li, Niu | |
Glutamate Binding-Site Ligands of NMDA Receptors | 1-gen-2011 | C. Bonaccorso; N. Micale; R. Ettari; S. Grasso; M. Zappalà | |
Effect of mammalian SERCA inhibitors on Plasmodium falciparum growth in vitro | 1-gen-2011 | Serena, Pulcini; Stefan, Paula; Chengguo, Xing; Ettari, Roberta; Henry M., Staines; Sanjeev, Krishna | |
Development of Novel Peptidomimetics Containing a VinylSulfone Moiety as Proteasome Inhibitors | 1-gen-2011 | Ettari, Roberta; Bonaccorso, Cinzia; Micale, Nicola; Cornelia, Heindl; Tanja, Schirmeister; Calabro', Maria; Grasso, Silvana; Zappala', Maria | |
Peptidomimetics containing a vinyl ketone warhead as falcipain-2 inhibitors | 1-gen-2011 | Ettari, Roberta; Zappala', Maria; Micale, Nicola; Giovanni, Grazioso; Giofre', Salvatore Vincenzo; Tanja, Schirmeister; Grasso, Silvana | |
Formation of 3-Aminofuran-2-(5H)-ones and 3-Amino-1H-pyrrole-2,5-diones by Rearrangement of Isoxazolidines | 1-gen-2011 | Iannazzo, Daniela; Carnovale, Caterina; Giofre', Salvatore Vincenzo; Ettari, Roberta; Romeo, Giovanni; Romeo, Roberto; Giuseppe, Lanza; Ugo, Chiacchio | |
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF PEPTIDOMIMETIC FALCIPAIN-2 INHIBITORS AS ANTIMALARIAL AGENTS | 1-gen-2012 | Micale, Nicola; Ettari, Roberta; T., Schirmeister; G., Grazioso; Grasso, Silvana; Zappala', Maria | |
Novel peptidomimetic inhibitors, containing a 1,4-benzodiazepine scaffold, for treatment of neglected tropical diseases | 1-gen-2012 | Ettari, Roberta; A., Pinto; L., Tamborini; I. C., Angelo; Grasso, Silvana; C., De Micheli | |
Synthesis and Molecular Modeling Studies of Derivatives of a Highly Potent Peptidomimetic Vinyl Ester as Falcipain-2 Inhibitors | 1-gen-2012 | Ettari, Roberta; Micale, Nicola; Giovanni, Grazioso; Bova, Floriana; Tanja, Schirmeister; Grasso, Silvana; Zappala', Maria | |
Development of peptidomimetic boronates as proteasome inhibitors | 1-gen-2012 | Micale, Nicola; Ettari, Roberta; C., Di Giovanni; A., Lavecchia; Scarbaci, Kety; V., Troiano; Grasso, Silvana; E., Novellino; T., Schirmeister; Zappala', Maria | |
Mechanism of falcipain-2 inhibition by α,β-unsaturated benzo[1,4]diazepin-2-one methyl ester | 1-gen-2012 | Grazioso, G; Legnani, L; Toma, L; Ettari, Roberta; Micale, Nicola; De Micheli, C. | |
Identification of a new series of non-covalent proteasome inhibitors with selectivity for β5-subunits | 1-gen-2013 | Scarbaci, Kety; Troiano, V.; Micale, Nicola; Ettari, Roberta; Lavecchia, A.; Di Giovanni, C.; Grasso, Silvana; Novellino, E.; Schirmeister, T.; Zappala', Maria |
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