Sfoglia per Autore
Progettazione, Sintesi e SAR di analoghi 1,3-diidro-benzimidazoloni come nuovi agenti anti-HIV
2007-01-01 Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; Barreca, M. L.; DE CLERCQ, E.; Chimirri, Alba; Monforte, Anna Maria
Structure-Based Pharmacophore Identification of New Chemical Scaffolds as Non –Nucleoside riverse Transcriptase Inhibitors
2007-01-01 DE LUCA, Laura; Barreca, Ml; Iraci, Nunzio; Ferro, Stefania; Monforte, Am; Maga, G; Chimirri, A.
Structure-based pharmacophore identification of new chemical scaffolds as non-nucleoside reverse transcriptase inhibitors
2007-01-01 Barreca, Maria Letizia; DE LUCA, Laura; Iraci, Nunzio; Rao, A; Ferro, Stefania; Maga, G; Chimirri, Alba
Discovery of novel benzimidazolones as potent non-nucleoside reverse transcriptase inhibitors active against wild-type and mutant HIV-1 strains.
2007-01-01 Barreca, Ml; Rao, A; DE LUCA, Laura; Iraci, Nunzio; Monforte, Anna Maria; Maga, G; DE CLERCQ, E; Pannecouque, C; Balzarini, J; Chimirri, Alba
MOLECULAR MODELING STUDIES AND SYNTHESIS FOR THE DISCOVERY OF HIV-1 IN-LEDGF/P75 INTERACTION INHIBITORS
2008-01-01 Ferro, Stefania; DE LUCA, Laura; BARRECA M., L; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
Synthesis and SAR of new 1,3-dihydro-benzimidazolone analogues as non-nucleoside reverse transcriptase inhibitors (NNRTIs)
2008-01-01 Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; DE CLERCQ, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria
HIV-1-IN Strand-Transfer Inhibitors: phenyl ring exploration and synthesis of 1H-benzylindole derivative through fluorine substitutions
2008-01-01 Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Iraci, Nunzio; DE GRAZIA, Sara; Debyser, Z; Witvrouw, M; Chimirri, Alba
A refined pharmacophore model and optimization of 1H-benzylindole HIV-1 integrase inhibitors
2008-01-01 DE LUCA, Laura; Barreca, Ml; Ferro, Stefania; Iraci, Nunzio; Debyser, Z; Witvrouw, M; Chimirri, Alba
Improvement of water solubility of non-competitive AMPA receptor antagonists by complexation with beta-cyclodextrin
2008-01-01 STANCANELLI R; CRUPI V; DE LUCA L; FICARRA P; FICARRA R; GITTO R; GUARDO M; IRACI N; MAJOLINO D; TOMMASINI S; VENUTI V
INTEGRASE STRAND TRANSFER INHIBITORS (INSTIs): SYNTHESIS AND ANTIVIRAL EFFETCS OF CHLORO-FLUORO SUBSTITUTIONS
2008-01-01 Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; MARIA LETIZIA, Barreca; Iraci, Nunzio; Frauke, Christ; Zeger, Debyser; Chimirri, Alba
Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside riverse transcriptase inhibitors
2008-01-01 Monforte, Anna Maria; Rao, A; Logoteta, Patrizia; Ferro, Stefania; DE LUCA, Laura; Barreca, Maria Letizia; Iraci, Nunzio; Maga, G; DE CLERCQ, E; Pannecouque, C; Chimirri, Alba
A refined pharmacophore model for HIV-1 integrase inhibitors: Optimization of potency in the 1H-benzylindole series
2008-01-01 DE LUCA, Laura; Barreca, Maria Letizia; Ferro, Stefania; Iraci, Nunzio; Michiels, M; Christ, F; Debyser, Z; Witvrouw, M; Chimirri, Alba
Design, synthesis and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents
2009-01-01 Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; De Clercq, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria
A structure-based approach to ligand discovery for inhibition of HIV-1 IN-LEDGF/p75 interaction: a new target for anti-AIDS therapy
2009-01-01 DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; Gitto, Rosaria; Monforte, Anna Maria; Iraci, Nunzio; Barreca, Ml; Debyser, Z; Chimirri, Alba
From 3D-pharmacophore models to synthetic route towards anti-HIV agents
2009-01-01 Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; DE GRAZIA, Sara; Iraci, Nunzio; Barreca, Ml; Debyser, Z.
Novel targets for HIV therapy: small molecules blocking IN-LEDGF/p75 interaction
2009-01-01 Ferro, Stefania; DE LUCA, Laura; Agnello, Stefano; Barreca, Ml; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
Design, Synthesis and SAR of New Potent HIV-1 RT Inhibitors”. Antiviral Research
2009-01-01 Chimirri, Alba; De Clercq, E; Maga, G; Logoteta, Patrizia; Ferro, Stefania; DE LUCA, Laura; Iraci, Nunzio; Pannecouque, C; Monforte, Anna Maria
Discovery of HIV-1 Integrase and cellular cofactor LEDGF/p75 interaction inhibitors
2009-01-01 Ferro, Stefania; Agnello, Stefano; DE LUCA, Laura; Barreca, Ml; Iraci, N; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
Design, synthesis, and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents
2009-01-01 Monforte AM; Logoteta P; Ferro S; De Luca L; Iraci N; Maga G; De Clercq E; Pannecouque C; Chimirri A
Induced-Fit Docking Approach Provides Insight into the Binding Mode and Mechanism of Action of HIV-1 Integrase Inhibitors
2009-01-01 Barreca, Maria Letizia; Iraci, Nunzio; DE LUCA, Laura; Chimirri, Alba
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Progettazione, Sintesi e SAR di analoghi 1,3-diidro-benzimidazoloni come nuovi agenti anti-HIV | 1-gen-2007 | Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; Barreca, M. L.; DE CLERCQ, E.; Chimirri, Alba; Monforte, Anna Maria | |
Structure-Based Pharmacophore Identification of New Chemical Scaffolds as Non –Nucleoside riverse Transcriptase Inhibitors | 1-gen-2007 | DE LUCA, Laura; Barreca, Ml; Iraci, Nunzio; Ferro, Stefania; Monforte, Am; Maga, G; Chimirri, A. | |
Structure-based pharmacophore identification of new chemical scaffolds as non-nucleoside reverse transcriptase inhibitors | 1-gen-2007 | Barreca, Maria Letizia; DE LUCA, Laura; Iraci, Nunzio; Rao, A; Ferro, Stefania; Maga, G; Chimirri, Alba | |
Discovery of novel benzimidazolones as potent non-nucleoside reverse transcriptase inhibitors active against wild-type and mutant HIV-1 strains. | 1-gen-2007 | Barreca, Ml; Rao, A; DE LUCA, Laura; Iraci, Nunzio; Monforte, Anna Maria; Maga, G; DE CLERCQ, E; Pannecouque, C; Balzarini, J; Chimirri, Alba | |
MOLECULAR MODELING STUDIES AND SYNTHESIS FOR THE DISCOVERY OF HIV-1 IN-LEDGF/P75 INTERACTION INHIBITORS | 1-gen-2008 | Ferro, Stefania; DE LUCA, Laura; BARRECA M., L; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba | |
Synthesis and SAR of new 1,3-dihydro-benzimidazolone analogues as non-nucleoside reverse transcriptase inhibitors (NNRTIs) | 1-gen-2008 | Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; DE CLERCQ, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria | |
HIV-1-IN Strand-Transfer Inhibitors: phenyl ring exploration and synthesis of 1H-benzylindole derivative through fluorine substitutions | 1-gen-2008 | Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Iraci, Nunzio; DE GRAZIA, Sara; Debyser, Z; Witvrouw, M; Chimirri, Alba | |
A refined pharmacophore model and optimization of 1H-benzylindole HIV-1 integrase inhibitors | 1-gen-2008 | DE LUCA, Laura; Barreca, Ml; Ferro, Stefania; Iraci, Nunzio; Debyser, Z; Witvrouw, M; Chimirri, Alba | |
Improvement of water solubility of non-competitive AMPA receptor antagonists by complexation with beta-cyclodextrin | 1-gen-2008 | STANCANELLI R; CRUPI V; DE LUCA L; FICARRA P; FICARRA R; GITTO R; GUARDO M; IRACI N; MAJOLINO D; TOMMASINI S; VENUTI V | |
INTEGRASE STRAND TRANSFER INHIBITORS (INSTIs): SYNTHESIS AND ANTIVIRAL EFFETCS OF CHLORO-FLUORO SUBSTITUTIONS | 1-gen-2008 | Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; MARIA LETIZIA, Barreca; Iraci, Nunzio; Frauke, Christ; Zeger, Debyser; Chimirri, Alba | |
Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside riverse transcriptase inhibitors | 1-gen-2008 | Monforte, Anna Maria; Rao, A; Logoteta, Patrizia; Ferro, Stefania; DE LUCA, Laura; Barreca, Maria Letizia; Iraci, Nunzio; Maga, G; DE CLERCQ, E; Pannecouque, C; Chimirri, Alba | |
A refined pharmacophore model for HIV-1 integrase inhibitors: Optimization of potency in the 1H-benzylindole series | 1-gen-2008 | DE LUCA, Laura; Barreca, Maria Letizia; Ferro, Stefania; Iraci, Nunzio; Michiels, M; Christ, F; Debyser, Z; Witvrouw, M; Chimirri, Alba | |
Design, synthesis and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents | 1-gen-2009 | Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; De Clercq, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria | |
A structure-based approach to ligand discovery for inhibition of HIV-1 IN-LEDGF/p75 interaction: a new target for anti-AIDS therapy | 1-gen-2009 | DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; Gitto, Rosaria; Monforte, Anna Maria; Iraci, Nunzio; Barreca, Ml; Debyser, Z; Chimirri, Alba | |
From 3D-pharmacophore models to synthetic route towards anti-HIV agents | 1-gen-2009 | Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; DE GRAZIA, Sara; Iraci, Nunzio; Barreca, Ml; Debyser, Z. | |
Novel targets for HIV therapy: small molecules blocking IN-LEDGF/p75 interaction | 1-gen-2009 | Ferro, Stefania; DE LUCA, Laura; Agnello, Stefano; Barreca, Ml; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba | |
Design, Synthesis and SAR of New Potent HIV-1 RT Inhibitors”. Antiviral Research | 1-gen-2009 | Chimirri, Alba; De Clercq, E; Maga, G; Logoteta, Patrizia; Ferro, Stefania; DE LUCA, Laura; Iraci, Nunzio; Pannecouque, C; Monforte, Anna Maria | |
Discovery of HIV-1 Integrase and cellular cofactor LEDGF/p75 interaction inhibitors | 1-gen-2009 | Ferro, Stefania; Agnello, Stefano; DE LUCA, Laura; Barreca, Ml; Iraci, N; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba | |
Design, synthesis, and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents | 1-gen-2009 | Monforte AM; Logoteta P; Ferro S; De Luca L; Iraci N; Maga G; De Clercq E; Pannecouque C; Chimirri A | |
Induced-Fit Docking Approach Provides Insight into the Binding Mode and Mechanism of Action of HIV-1 Integrase Inhibitors | 1-gen-2009 | Barreca, Maria Letizia; Iraci, Nunzio; DE LUCA, Laura; Chimirri, Alba |
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