CITARELLA, Andrea
CITARELLA, Andrea
Dipartimento di Scienze biomediche, odontoiatriche e delle immagini morfologiche e funzionali
Chemoselective Homologation-Deoxygenation Strategy Enabling the Direct Conversion of Carbonyls into (n+1)-Halomethyl-Alkanes
2020-01-01 Miele, Margherita; Citarella, Andrea; Langer, Thierry; Urban, Ernst; Zehl, Martin; Holzer, Wolfgang; Ielo, Laura; Pace, Vittorio
Direct and Chemoselective Synthesis of Tertiary Difluoroketones via Weinreb Amide Homologation with a CHF2-Carbene Equivalent
2019-01-01 Miele, M.; Citarella, A.; Micale, N.; Holzer, W.; Pace, V.
Direct and chemoselective synthesis α,α-difluoromethylketones under transfer of (CHF2) unit
2019-01-01 Citarella, A.; Miele, M.; Micale, N.; Pace, V.
Direct and chemoselective transfer of the difluoromethyl (CHF2) unit into carbon-electrophiles under nucleophilic regime
2019-01-01 Citarella, A.; Miele, M.; Micale, N.; Pace, V.
Fluorine-based pseudopeptides from halocarbene transfer reaction: synthesis and biological perspectives
2020-01-01 Citarella, Andrea; Miele, Margherita; Pace, Vittorio; Micale, Nicola
Hydrogels for the Delivery of Plant-Derived (Poly)Phenols
2020-01-01 Micale, Nicola; Citarella, Andrea; Molonia, Maria Sofia; Speciale, Antonio; Cimino, Francesco; Saija, Antonella; Cristani, Mariateresa
Hydroxamic Acid-Based Histone Deacetylase (HDAC) Inhibitors Bearing a Pyrazole Scaffold and a Cinnamoyl Linker
2019-01-01 Zagni, Chiara; Citarella, Andrea; Oussama, Mahjoub; Rescifina, Antonio; Maugeri, Alessandro; Navarra, Michele; Scala, Angela; Piperno, Anna; Micale, Nicola
Natural product-based hybrids as potential candidates for the treatment of cancer: Focus on curcumin and resveratrol
2021-01-01 Micale, N.; Molonia, M. S.; Citarella, A.; Cimino, F.; Saija, A.; Cristani, M.; Speciale, A.
Novel Class of Proteasome Inhibitors: In Silico and In Vitro Evaluation of Diverse Chloro(trifluoromethyl)aziridines
2022-01-01 Ielo, Laura; Patamia, Vincenzo; Citarella, Andrea; Efferth, Thomas; Shahhamzehei, Nasim; Schirmeister, Tanja; Stagno, Claudio; Langer, Thierry; Rescifina, Antonio; Micale, Nicola; Pace, Vittorio
NUCLEOPHILIC α-SUBSTITUTED ORGANOMETALLIC REAGENTS IN HOMOLOGATION CHEMISTRY: SYNTHETIC APPLICATIONS AND BIOLOGICAL PERSPECTIVES
2021-01-13 Citarella, Andrea
Peptide-based α,α-Difluoromethyl Ketone as new inhibitor of Pathogenic Coronavirus Mpro
2020-01-01 Citarella, Andrea; Gentile, Davide; Rescifina, Antonio; Pace, Vittorio; Piperno, Anna; Micale, Nicola
Peptidyl fluoromethyl ketones and their applications in medicinal chemistry
2020-01-01 Micale, Nicola; Citarella, Andrea
Pseudo-Dipeptide Bearing ,-Difluoromethyl Ketone Moiety as ElectrophilicWarhead with Activity against Coronaviruses
2021-01-01 Citarella, Andrea; Gentile, Davide; Rescifina, Antonio; Piperno, Anna; Mognetti, Barbara; Gribaudo, Giorgio; Sciortino, Maria Teresa; Holzer, Wolfgang; Pace, Vittorio; Micale, Nicola
SARS-CoV-2 Mpro: A Potential Target for Peptidomimetics and Small-Molecule Inhibitors
2021-01-01 Citarella, Andrea; Scala, Angela; Piperno, Anna; Micale, Nicola
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells
2024-01-01 Citarella, Andrea; Petrella, Serena; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Damia, Giovanna; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele
Synthesis, computational investigation and biological evaluation of α,α-difluoromethyl ketones embodying pyrazole and isoxazole nuclei as COX inhibitors
2022-01-01 Citarella, Andrea; Ielo, Laura; Stagno, Claudio; Cristani, Mariateresa; Muscara, Claudia; Pace, Vittorio; Micale, Nicola
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Chemoselective Homologation-Deoxygenation Strategy Enabling the Direct Conversion of Carbonyls into (n+1)-Halomethyl-Alkanes | 1-gen-2020 | Miele, Margherita; Citarella, Andrea; Langer, Thierry; Urban, Ernst; Zehl, Martin; Holzer, Wolfgang; Ielo, Laura; Pace, Vittorio | |
| Direct and Chemoselective Synthesis of Tertiary Difluoroketones via Weinreb Amide Homologation with a CHF2-Carbene Equivalent | 1-gen-2019 | Miele, M.; Citarella, A.; Micale, N.; Holzer, W.; Pace, V. | |
| Direct and chemoselective synthesis α,α-difluoromethylketones under transfer of (CHF2) unit | 1-gen-2019 | Citarella, A.; Miele, M.; Micale, N.; Pace, V. | |
| Direct and chemoselective transfer of the difluoromethyl (CHF2) unit into carbon-electrophiles under nucleophilic regime | 1-gen-2019 | Citarella, A.; Miele, M.; Micale, N.; Pace, V. | |
| Fluorine-based pseudopeptides from halocarbene transfer reaction: synthesis and biological perspectives | 1-gen-2020 | Citarella, Andrea; Miele, Margherita; Pace, Vittorio; Micale, Nicola | |
| Hydrogels for the Delivery of Plant-Derived (Poly)Phenols | 1-gen-2020 | Micale, Nicola; Citarella, Andrea; Molonia, Maria Sofia; Speciale, Antonio; Cimino, Francesco; Saija, Antonella; Cristani, Mariateresa | |
| Hydroxamic Acid-Based Histone Deacetylase (HDAC) Inhibitors Bearing a Pyrazole Scaffold and a Cinnamoyl Linker | 1-gen-2019 | Zagni, Chiara; Citarella, Andrea; Oussama, Mahjoub; Rescifina, Antonio; Maugeri, Alessandro; Navarra, Michele; Scala, Angela; Piperno, Anna; Micale, Nicola | |
| Natural product-based hybrids as potential candidates for the treatment of cancer: Focus on curcumin and resveratrol | 1-gen-2021 | Micale, N.; Molonia, M. S.; Citarella, A.; Cimino, F.; Saija, A.; Cristani, M.; Speciale, A. | |
| Novel Class of Proteasome Inhibitors: In Silico and In Vitro Evaluation of Diverse Chloro(trifluoromethyl)aziridines | 1-gen-2022 | Ielo, Laura; Patamia, Vincenzo; Citarella, Andrea; Efferth, Thomas; Shahhamzehei, Nasim; Schirmeister, Tanja; Stagno, Claudio; Langer, Thierry; Rescifina, Antonio; Micale, Nicola; Pace, Vittorio | |
| NUCLEOPHILIC α-SUBSTITUTED ORGANOMETALLIC REAGENTS IN HOMOLOGATION CHEMISTRY: SYNTHETIC APPLICATIONS AND BIOLOGICAL PERSPECTIVES | 13-gen-2021 | Citarella, Andrea | |
| Peptide-based α,α-Difluoromethyl Ketone as new inhibitor of Pathogenic Coronavirus Mpro | 1-gen-2020 | Citarella, Andrea; Gentile, Davide; Rescifina, Antonio; Pace, Vittorio; Piperno, Anna; Micale, Nicola | |
| Peptidyl fluoromethyl ketones and their applications in medicinal chemistry | 1-gen-2020 | Micale, Nicola; Citarella, Andrea | |
| Pseudo-Dipeptide Bearing ,-Difluoromethyl Ketone Moiety as ElectrophilicWarhead with Activity against Coronaviruses | 1-gen-2021 | Citarella, Andrea; Gentile, Davide; Rescifina, Antonio; Piperno, Anna; Mognetti, Barbara; Gribaudo, Giorgio; Sciortino, Maria Teresa; Holzer, Wolfgang; Pace, Vittorio; Micale, Nicola | |
| SARS-CoV-2 Mpro: A Potential Target for Peptidomimetics and Small-Molecule Inhibitors | 1-gen-2021 | Citarella, Andrea; Scala, Angela; Piperno, Anna; Micale, Nicola | |
| Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells | 1-gen-2024 | Citarella, Andrea; Petrella, Serena; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Damia, Giovanna; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele | |
| Synthesis, computational investigation and biological evaluation of α,α-difluoromethyl ketones embodying pyrazole and isoxazole nuclei as COX inhibitors | 1-gen-2022 | Citarella, Andrea; Ielo, Laura; Stagno, Claudio; Cristani, Mariateresa; Muscara, Claudia; Pace, Vittorio; Micale, Nicola |