Sfoglia per Autore
Development of Novel Peptide-based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs)
2017-01-01 Previti, Santo; Ettari, Roberta; Sandro, Cosconati; Giorgio, Amendola; Khawla, Chouchene; Annika, Wagner; Ute A., Hellmich; Kathrin, Ulrich; R., Luise Krauth Siegel; Peter R., Wich; Ira, Schmid; Tanja, Schirmeister; Jiri, Gut; Philip J., Rosenthal; Grasso, Silvana; Zappala', Maria
Identification of 2-thioxoimidazolidin-4-one derivatives as novel noncovalent proteasome and immunoproteasome inhibitors
2018-01-01 Maccari, R.; Ettari, R.; Adornato, I.; Naß, A.; Wolber, G.; Bitto, A.; Mannino, F.; Aliquo', Federica; Bruno, G.; Nicolò, F.; Previti, S.; Grasso, S.; Zappalà, M.; Ottanà, R.
Immunoproteasome-selective and non-selective inhibitors: A promising approach for the treatment of multiple myeloma.
2018-01-01 Ettari, Roberta; Zappala', Maria; Grasso, Silvana; Musolino, Caterina; Innao, Vanessa; Allegra, Alessandro
Development of novel irreversible rhodesain inhibitors as antitrypanosomal agents.
2019-01-01 Maiorana, Santina; Ettari, Roberta; Previti, Santo; Cosconati, Sandro; Zappala', Maria
Development of pyridin-2-one derivatives as non-covalent inhibitors of immunoproteasome
2019-01-01 Maiorana, Santina; Ettari, Roberta; Lavecchia, Antonio; Zappala', Maria
Development of novel peptide-based Michael acceptors as antitrypanosomal agents
2019-01-01 Maiorana, Santina; Ettari, Roberta; Cosconati, Sandro; Zappala', Maria
Design, synthesis and biological evaluation of novel rhodesain inhibitors for the treatment of Human African Trypanosomiasis
2019-01-01 Maiorana, S.; Ettari, R.; Previti, S.; Cosconati, S.; Zappalà, M.
Composti antitumorali
2019-01-01 Corsi, L.; Alessandrini, A.; Bennaud, C.; Ettari, R.
Non-covalent immunoproteasome inhibitors induce cell cycle arrest in multiple myeloma cells
2019-01-01 Ettari, R.; Pallio, G.; Pizzino, G.; Irrera, N.; Zappalà, M.; Maiorana, S.; Di Chio, C.; Altavilla, D.; Squadrito, F.; Bitto, A.
Formaldehyde exposure and acute myeloid leukemia: A review of the literature
2019-01-01 Allegra, Alessandro; Spatari, Giovanna; Mattioli, Stefano; Curti, Stefania; Innao, Vanessa; Ettari, Roberta; Allegra, Andrea Gaetano; Giorgianni, Concetto; Gangemi, Sebastiano; Musolino, Caterina
Role of the microbiota in hematologic malignancies.
2019-01-01 Allegra, A.; Innao, V.; Allegra, A. G.; Ettari, R.; Pugliese, M.; Pulvirenti, N.; Musolino, C.
Drug combination studies of curcumin and genistein against rhodesain of Trypanosoma brucei rhodesiense
2019-01-01 Ettari, Roberta; Previti, Santo; Maiorana, Santina; Allegra, Alessandro; Schirmeister, Tanja; Grasso, Silvana; Zappala', Maria
Development of novel amides as noncovalent inhibitors of immunoproteasome
2019-01-01 Ettari, Roberta; Cerchia, Carmen; Maiorana, Santina; Guccione, Manuela; Novellino, Ettore; Bitto, Alessandra; Grasso, Silvana; Lavecchia, Antonio; Zappala', Maria
Exploiting Curcumin Synergy With Natural Products Using Quantitative Analysis of Dose–Effect Relationships in an Experimental In Vitro Model of Osteoarthritis
2019-01-01 D'Ascola, Angela; Irrera, Natasha; Ettari, Roberta; Bitto, Alessandra; Pallio, Giovanni; Mannino, Federica; Atteritano, Marco; Campo, Giuseppe M.; Minutoli, Letteria; Arcoraci, Vincenzo; Squadrito, Violetta; Picciolo, Giacomo; Squadrito, Francesco; Altavilla, Domenica
Optimization Strategy of Novel Peptide-Based Michael Acceptors for the Treatment of Human African Trypanosomiasis
2019-01-01 Ettari, Roberta; Previti, Santo; Maiorana, Santina; Amendola, Giorgio; Wagner, Annika; Cosconati, Sandro; Schirmeister, Tanja; Hellmich, Ute A.; Zappala', Maria
Development of novel benzodiazepine-based peptidomimetics as inhibitors of rhodesain of Trypanosoma brucei rhodesiense
2020-01-01 DI CHIO, Carla; Previti, Santo; Cosconati, Sandro; Zappala', Maria; Ettari, Roberta
Discovery of novel peptidomimetics containing a benzodiazepine scaffold as inhibitors of rhodesain of Trypanosoma brucei rhodesiense
2020-01-01 DI CHIO, Carla; Previti, Santo; Amendola, Giorgio; Cosconati, Sandro; Zappala', Maria; Ettari, Roberta
Discovery of novel antitrypanosomal agents: design, synthesis of novel benzodiazepine-based peptidomimetics targeting rhodesain, the main cysteine protease of Trypanosoma brucei rhodesiense
2020-01-01 DI CHIO, Carla; Zappala', Maria; Ettari, Roberta
Development of Novel Benzodiazepine-Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense
2020-01-01 DI CHIO, Carla; Previti, Santo; Amendola, Giorgio; Cosconati, Sandro; Schirmeister, Tanja; Zappala', Maria; Ettari, Roberta
Peptidyl Vinyl Ketone Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment
2020-01-01 Maiorana, Santina; Ettari, Roberta; Previti, Santo; Amendola, Giorgio; Wagner, Annika; Cosconati, Sandro; Hellmich, Ute A.; Schirmeister, Tanja; Zappala', Maria
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Development of Novel Peptide-based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs) | 1-gen-2017 | Previti, Santo; Ettari, Roberta; Sandro, Cosconati; Giorgio, Amendola; Khawla, Chouchene; Annika, Wagner; Ute A., Hellmich; Kathrin, Ulrich; R., Luise Krauth Siegel; Peter R., Wich; Ira, Schmid; Tanja, Schirmeister; Jiri, Gut; Philip J., Rosenthal; Grasso, Silvana; Zappala', Maria | |
Identification of 2-thioxoimidazolidin-4-one derivatives as novel noncovalent proteasome and immunoproteasome inhibitors | 1-gen-2018 | Maccari, R.; Ettari, R.; Adornato, I.; Naß, A.; Wolber, G.; Bitto, A.; Mannino, F.; Aliquo', Federica; Bruno, G.; Nicolò, F.; Previti, S.; Grasso, S.; Zappalà, M.; Ottanà, R. | |
Immunoproteasome-selective and non-selective inhibitors: A promising approach for the treatment of multiple myeloma. | 1-gen-2018 | Ettari, Roberta; Zappala', Maria; Grasso, Silvana; Musolino, Caterina; Innao, Vanessa; Allegra, Alessandro | |
Development of novel irreversible rhodesain inhibitors as antitrypanosomal agents. | 1-gen-2019 | Maiorana, Santina; Ettari, Roberta; Previti, Santo; Cosconati, Sandro; Zappala', Maria | |
Development of pyridin-2-one derivatives as non-covalent inhibitors of immunoproteasome | 1-gen-2019 | Maiorana, Santina; Ettari, Roberta; Lavecchia, Antonio; Zappala', Maria | |
Development of novel peptide-based Michael acceptors as antitrypanosomal agents | 1-gen-2019 | Maiorana, Santina; Ettari, Roberta; Cosconati, Sandro; Zappala', Maria | |
Design, synthesis and biological evaluation of novel rhodesain inhibitors for the treatment of Human African Trypanosomiasis | 1-gen-2019 | Maiorana, S.; Ettari, R.; Previti, S.; Cosconati, S.; Zappalà, M. | |
Composti antitumorali | 1-gen-2019 | Corsi, L.; Alessandrini, A.; Bennaud, C.; Ettari, R. | |
Non-covalent immunoproteasome inhibitors induce cell cycle arrest in multiple myeloma cells | 1-gen-2019 | Ettari, R.; Pallio, G.; Pizzino, G.; Irrera, N.; Zappalà, M.; Maiorana, S.; Di Chio, C.; Altavilla, D.; Squadrito, F.; Bitto, A. | |
Formaldehyde exposure and acute myeloid leukemia: A review of the literature | 1-gen-2019 | Allegra, Alessandro; Spatari, Giovanna; Mattioli, Stefano; Curti, Stefania; Innao, Vanessa; Ettari, Roberta; Allegra, Andrea Gaetano; Giorgianni, Concetto; Gangemi, Sebastiano; Musolino, Caterina | |
Role of the microbiota in hematologic malignancies. | 1-gen-2019 | Allegra, A.; Innao, V.; Allegra, A. G.; Ettari, R.; Pugliese, M.; Pulvirenti, N.; Musolino, C. | |
Drug combination studies of curcumin and genistein against rhodesain of Trypanosoma brucei rhodesiense | 1-gen-2019 | Ettari, Roberta; Previti, Santo; Maiorana, Santina; Allegra, Alessandro; Schirmeister, Tanja; Grasso, Silvana; Zappala', Maria | |
Development of novel amides as noncovalent inhibitors of immunoproteasome | 1-gen-2019 | Ettari, Roberta; Cerchia, Carmen; Maiorana, Santina; Guccione, Manuela; Novellino, Ettore; Bitto, Alessandra; Grasso, Silvana; Lavecchia, Antonio; Zappala', Maria | |
Exploiting Curcumin Synergy With Natural Products Using Quantitative Analysis of Dose–Effect Relationships in an Experimental In Vitro Model of Osteoarthritis | 1-gen-2019 | D'Ascola, Angela; Irrera, Natasha; Ettari, Roberta; Bitto, Alessandra; Pallio, Giovanni; Mannino, Federica; Atteritano, Marco; Campo, Giuseppe M.; Minutoli, Letteria; Arcoraci, Vincenzo; Squadrito, Violetta; Picciolo, Giacomo; Squadrito, Francesco; Altavilla, Domenica | |
Optimization Strategy of Novel Peptide-Based Michael Acceptors for the Treatment of Human African Trypanosomiasis | 1-gen-2019 | Ettari, Roberta; Previti, Santo; Maiorana, Santina; Amendola, Giorgio; Wagner, Annika; Cosconati, Sandro; Schirmeister, Tanja; Hellmich, Ute A.; Zappala', Maria | |
Development of novel benzodiazepine-based peptidomimetics as inhibitors of rhodesain of Trypanosoma brucei rhodesiense | 1-gen-2020 | DI CHIO, Carla; Previti, Santo; Cosconati, Sandro; Zappala', Maria; Ettari, Roberta | |
Discovery of novel peptidomimetics containing a benzodiazepine scaffold as inhibitors of rhodesain of Trypanosoma brucei rhodesiense | 1-gen-2020 | DI CHIO, Carla; Previti, Santo; Amendola, Giorgio; Cosconati, Sandro; Zappala', Maria; Ettari, Roberta | |
Discovery of novel antitrypanosomal agents: design, synthesis of novel benzodiazepine-based peptidomimetics targeting rhodesain, the main cysteine protease of Trypanosoma brucei rhodesiense | 1-gen-2020 | DI CHIO, Carla; Zappala', Maria; Ettari, Roberta | |
Development of Novel Benzodiazepine-Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense | 1-gen-2020 | DI CHIO, Carla; Previti, Santo; Amendola, Giorgio; Cosconati, Sandro; Schirmeister, Tanja; Zappala', Maria; Ettari, Roberta | |
Peptidyl Vinyl Ketone Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment | 1-gen-2020 | Maiorana, Santina; Ettari, Roberta; Previti, Santo; Amendola, Giorgio; Wagner, Annika; Cosconati, Sandro; Hellmich, Ute A.; Schirmeister, Tanja; Zappala', Maria |
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