Sfoglia per Autore
Synthesis and antitumor activity evaluation of Delta(2)-1,2,4- oxadiazoline derivatives
1996-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Rao, A; Zappala', Maria
Substituent effects on the enantioselective retention of anti- HIV 5-aryl-Delta(2)-1,2,4-oxadiazolines on R,R-DACH-DNB chiral stationary phase
1996-01-01 Altomare, C; Cellamare, S; Carotti, A; Barreca, Ml; Chimirri, Alba; Monforte, Anna Maria; Gasparrini, F; Villani, C; Cirilli, M; Mazza, F.
Anti-HIV agents .4. Synthesis and in vitro anti-HIV activity of novel 1-(2,6-difluorophenyl)-1H,3H-thiazolo[3,4- a]benzimidazoles
1996-01-01 Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Scopelliti, R.
Electronic and conformational properties of 2,3-benzodiazepine derivatives
1996-01-01 Pelaggi, Mr; Girlanda, Raffaello; Chimirri, Alba; Gitto, Rosaria
Azirino[1,2-d][1,4]benzodiazepine derivatives and related 1,4- benzodiazepines as anticonvulsant agents in DBA/2 mice
1996-01-01 Desarro, G; Chimirri, Alba; Zappala', Maria; Guisti, P; Lipartiti, M; DE SARRO, Angelina
Separation of the enantiomers of anticonvulsant tricyclic pyrroloimidazolones by enantioselective HPLC. A chiral recognition model and a chiroptical study
1996-01-01 Caccamese, S; Principato, G; Chimirri, Alba; Grasso, Silvana
1-fluoromethyl-1-methyl-1H,3H-thiazolo-[3,4-a]benzimidazole
1996-01-01 BRUNO G; CHIMIRRI A; MONFORTE AM; F. NICOLO'; SCOPELLITI R
Structural features and anti-human immunodeficiency virus (HIV) activity of the isomers of 1-(2',6'-difluorophenyl)-1H,3H- thiazolo[3,4-a]benzimidazole, a potent non-nucleoside HIV-1 reverse transcriptase inhibitor
1997-01-01 Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Witvrouw, M.; Jonckeere, H.; Balzarini, J.; Declercq, E.
Anti-HIV agents. V. Synthesis, structure and in vitro anti-HIV activity of novel 1H,3H-naphtho[2 ',3 ': 4,5]imidazo[1,2- c]thiazoles
1997-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A.; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Scopelliti, R.
1-aryl-3,5-dihydro-4H-2,3-benzodiazepin-4-ones: Novel AMPA receptor antagonists
1997-01-01 Chimirri, Alba; DE SARRO, G; DE SARRO, Angelina; Gitto, Rosaria; Grasso, Silvana; Quartarone, S; Zappala', Maria; Giusti, P; Libri, V; Constanti, A; Chapman, Ag
1-Aryl-1H,3H-thiazolo[3,4-a]benzimidazole derivatives
1997-01-01 Bruno, Giuseppe; Chimirri, Alba; Monforte, Anna Maria; Nicolo', Francesco; Scopelliti, R.
Synthesis and structural characteristics of novel 5H- thiazolo[2,3-d][1,5]benzothiazepine derivatives
1997-01-01 Bruno, Giuseppe; Chimirri, Alba; Gitto, Rosaria; Grasso, Silvana; Nicolo', Francesco; Scopelliti, R; Zappala', Maria
Anticonvulsant activity of azirino[1,2-d][1,4]benzodiazepines and related 1,4-benzodiazepines in mice
1997-01-01 DE SARRO, G; Chimirri, Alba; Mckernan, R; Quirk, K; Giusti, P; DE SARRO, Angelina
Relationship between anticonvulsant activity and plasma level of some 2,3-benzodiazepines in genetically epilepsy-prone rats
1998-01-01 DE SARRO, G; Rizzo, M; Sinopoli, Va; Gitto, Rosaria; DE SARRO, Angelina; Zappala', Maria; Chimirri, Alba
Selective induction of apoptosis in multidrug resistant HL60R cells by the thiazolobenzimidazole derivative TBZ.
1998-01-01 Grimaudo, S.; Tolomeo, M.; Chimirri, Alba; Zappala', Maria; Gancitano, R. A.; D'Alessandro, N.
3,5-dihydro-4H-2,3-benzodiazepine-4-thiones: A new class of AMPA receptor antagonists
1998-01-01 Chimirri, Alba; DE SARRO, G; DE SARRO, Angelina; Gitto, Rosaria; Quartarone, S; Zappala', Maria; Constanti, A; Libri, V.
High-performance liquid chromatographic determination of new 2,3-benzodiazepines
1998-01-01 Rizzo, M; Sinopoli, Va; Gitto, Rosaria; Zappala', Maria; DE SARRO, G; Chimirri, Alba
Synthesis, structure and in vitro anti-human immunodeficiency virus activity of novel 3-methyl-1H,3H-thiazolo[3,4- a]benzimidazoles
1998-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Pannecouque, C; Witvrouw, M; DE CLERCQ, E.
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system
1999-01-01 Chimirri, Alba; DE CLERCQ, E.; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Pannecouque, C.; Rao, A.; Witvrouw, M.; Zappala', Maria
Synthesis and anticonvulsant activity of triazolo[4,5-c][2,3]benzodiazepines
1999-01-01 Chimirri, Alba; Bevacqua, F; Gitto, Rosaria; Quartarone, S; Zappala', Maria; DE SARRO, Angelina; G., DE SARRO; M., Rizzo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and antitumor activity evaluation of Delta(2)-1,2,4- oxadiazoline derivatives | 1-gen-1996 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Rao, A; Zappala', Maria | |
Substituent effects on the enantioselective retention of anti- HIV 5-aryl-Delta(2)-1,2,4-oxadiazolines on R,R-DACH-DNB chiral stationary phase | 1-gen-1996 | Altomare, C; Cellamare, S; Carotti, A; Barreca, Ml; Chimirri, Alba; Monforte, Anna Maria; Gasparrini, F; Villani, C; Cirilli, M; Mazza, F. | |
Anti-HIV agents .4. Synthesis and in vitro anti-HIV activity of novel 1-(2,6-difluorophenyl)-1H,3H-thiazolo[3,4- a]benzimidazoles | 1-gen-1996 | Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Scopelliti, R. | |
Electronic and conformational properties of 2,3-benzodiazepine derivatives | 1-gen-1996 | Pelaggi, Mr; Girlanda, Raffaello; Chimirri, Alba; Gitto, Rosaria | |
Azirino[1,2-d][1,4]benzodiazepine derivatives and related 1,4- benzodiazepines as anticonvulsant agents in DBA/2 mice | 1-gen-1996 | Desarro, G; Chimirri, Alba; Zappala', Maria; Guisti, P; Lipartiti, M; DE SARRO, Angelina | |
Separation of the enantiomers of anticonvulsant tricyclic pyrroloimidazolones by enantioselective HPLC. A chiral recognition model and a chiroptical study | 1-gen-1996 | Caccamese, S; Principato, G; Chimirri, Alba; Grasso, Silvana | |
1-fluoromethyl-1-methyl-1H,3H-thiazolo-[3,4-a]benzimidazole | 1-gen-1996 | BRUNO G; CHIMIRRI A; MONFORTE AM; F. NICOLO'; SCOPELLITI R | |
Structural features and anti-human immunodeficiency virus (HIV) activity of the isomers of 1-(2',6'-difluorophenyl)-1H,3H- thiazolo[3,4-a]benzimidazole, a potent non-nucleoside HIV-1 reverse transcriptase inhibitor | 1-gen-1997 | Chimirri, Alba; Grasso, Silvana; Molica, C; Monforte, Anna Maria; Monforte, Pietro; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Witvrouw, M.; Jonckeere, H.; Balzarini, J.; Declercq, E. | |
Anti-HIV agents. V. Synthesis, structure and in vitro anti-HIV activity of novel 1H,3H-naphtho[2 ',3 ': 4,5]imidazo[1,2- c]thiazoles | 1-gen-1997 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A.; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Scopelliti, R. | |
1-aryl-3,5-dihydro-4H-2,3-benzodiazepin-4-ones: Novel AMPA receptor antagonists | 1-gen-1997 | Chimirri, Alba; DE SARRO, G; DE SARRO, Angelina; Gitto, Rosaria; Grasso, Silvana; Quartarone, S; Zappala', Maria; Giusti, P; Libri, V; Constanti, A; Chapman, Ag | |
1-Aryl-1H,3H-thiazolo[3,4-a]benzimidazole derivatives | 1-gen-1997 | Bruno, Giuseppe; Chimirri, Alba; Monforte, Anna Maria; Nicolo', Francesco; Scopelliti, R. | |
Synthesis and structural characteristics of novel 5H- thiazolo[2,3-d][1,5]benzothiazepine derivatives | 1-gen-1997 | Bruno, Giuseppe; Chimirri, Alba; Gitto, Rosaria; Grasso, Silvana; Nicolo', Francesco; Scopelliti, R; Zappala', Maria | |
Anticonvulsant activity of azirino[1,2-d][1,4]benzodiazepines and related 1,4-benzodiazepines in mice | 1-gen-1997 | DE SARRO, G; Chimirri, Alba; Mckernan, R; Quirk, K; Giusti, P; DE SARRO, Angelina | |
Relationship between anticonvulsant activity and plasma level of some 2,3-benzodiazepines in genetically epilepsy-prone rats | 1-gen-1998 | DE SARRO, G; Rizzo, M; Sinopoli, Va; Gitto, Rosaria; DE SARRO, Angelina; Zappala', Maria; Chimirri, Alba | |
Selective induction of apoptosis in multidrug resistant HL60R cells by the thiazolobenzimidazole derivative TBZ. | 1-gen-1998 | Grimaudo, S.; Tolomeo, M.; Chimirri, Alba; Zappala', Maria; Gancitano, R. A.; D'Alessandro, N. | |
3,5-dihydro-4H-2,3-benzodiazepine-4-thiones: A new class of AMPA receptor antagonists | 1-gen-1998 | Chimirri, Alba; DE SARRO, G; DE SARRO, Angelina; Gitto, Rosaria; Quartarone, S; Zappala', Maria; Constanti, A; Libri, V. | |
High-performance liquid chromatographic determination of new 2,3-benzodiazepines | 1-gen-1998 | Rizzo, M; Sinopoli, Va; Gitto, Rosaria; Zappala', Maria; DE SARRO, G; Chimirri, Alba | |
Synthesis, structure and in vitro anti-human immunodeficiency virus activity of novel 3-methyl-1H,3H-thiazolo[3,4- a]benzimidazoles | 1-gen-1998 | Chimirri, Alba; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Rao, A; Zappala', Maria; Bruno, Giuseppe; Nicolo', Francesco; Pannecouque, C; Witvrouw, M; DE CLERCQ, E. | |
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system | 1-gen-1999 | Chimirri, Alba; DE CLERCQ, E.; Grasso, Silvana; Monforte, Anna Maria; Monforte, Pietro; Pannecouque, C.; Rao, A.; Witvrouw, M.; Zappala', Maria | |
Synthesis and anticonvulsant activity of triazolo[4,5-c][2,3]benzodiazepines | 1-gen-1999 | Chimirri, Alba; Bevacqua, F; Gitto, Rosaria; Quartarone, S; Zappala', Maria; DE SARRO, Angelina; G., DE SARRO; M., Rizzo |
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