Sfoglia per Autore
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system
1999-01-01 Chimirri, Alba; E., DE CLERCQ; Grasso, Silvana; Monforte, Anna Maria; P., Monforte; C., Pannecouque; A., Rao; M., Witvrouw; Zappala', Maria
Synthesis and anticonvulsant activity of new 11H-triazolo[4,5- c] [2,3]benzodiazepines
1999-01-01 Chimirri, Alba; Bevacqua, F; Gitto, Rosaria; Quartarone, S; Zappala', Maria; DE SARRO, Angelina; Maciocco, L; Biggio, G; DE SARRO, G.
Synthesis and structural features of 11H-tetrazolo[1,5-c][2,3]benzodiazepines
1999-01-01 Chimirri, Alba; Zappala', Maria; Gitto, Rosaria; Quartarone, S.; Bevacqua, F.
Anticonvulsant activity and plasma level of 2,3-benzodiazepin-4-ones (CFMs) in genetically epilepsy prone rats
1999-01-01 G., DE SARRO; M., Rizzo; Gitto, Rosaria; Zappala', Maria; Chimirri, Alba; A., DE SARRO
Anticonvulsant activity and plasma level of 2,3-benzodiazepin- 4-ones (CFMs) in genetically epilepsy-prone rats
1999-01-01 DE SARRO, G; Rizzo, M; Spagnolo, C; Gitto, Rosaria; DE SARRO, Angelina; Scotto, G; Zappala', Maria; Chimirri, Alba
7,11b-dihydro-9,10-dimethoxy-3,11b- diphenyl[1,2,4]oxadiazolo[5,4-a]-[2,3]benzodiazepin-6(5H)-one
1999-01-01 BRUNO G; CHIMIRRI A; GITTO R; NICOLO' FRANCESCO; SCOPELLITI R
Determination of 2,3-benzodiazepine derivatives in rat plasma by high-performance liquid chromatography
1999-01-01 RIZZO M; DE SARRO G; GITTO R; ZAPPALA M; CHIMIRRI A.
Synthesis and biological activity of novel 1H,3H-thiazolo[3,4- a] benzimidazoles: non-nucleoside human immunodeficiency virus type 1 reverse transcriptase inhibitors
1999-01-01 Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Rao, Angela; Zappala', Maria; Monforte, Anna Maria; Pannecouque, C; Witvrouw, M; Balzarini, J; DE CLERCQ, E.
Synthesis, structural features and anti-HIV activity of TBZ analogues
1999-01-01 Chimirri, Alba; Monforte, Anna Maria; P., Monforte; L., Musumeci; A., Rao; M., Zappal; M., Witvrouw; E., DE CLERCQ
Comparative molecular field analysis (CoMFA) and docking studies of non-nucleoside HIV-1 RT inhibitors (NNIs)
1999-01-01 Barreca, Maria Letizia; Carotti, A; Carrieri, A; Chimirri, Alba; Monforte, Anna Maria; Calace, Mp; Rao, Angela
AMPA receptor antagonists
1999-01-01 Chimirri, Alba; Gitto, Rosaria; Zappala', Maria
Development of 2,3-benzodiazepines and related AMPA receptor antagonists
2000-01-01 Gitto, Rosaria; Chimirri, Alba; Zappala', Maria; Quartarone, S.; Bevacqua, F.; DE SARRO, A.; DE SARRO, G.
Sintesi ed effetti apoptotici di derivati tiazolobenzimidazolici antitumorali
2000-01-01 Chimirri, Alba; P., Monforte; L., Musumeci; A., Rao; M. ZAPPAL A. M., Monforte; V. L., Narayanan
Design and development of 2,3-benzodiazepine (CFM) noncompetitive AMPA receptor antagonists
2000-01-01 Gitto, Rosaria; Zappala', Maria; Chimirri, Alba; G., DE SARRO
Synthesis and pharmacological evaluation of 4-aryl-6,7- dimethoxyphthalazines as anticonvulsant agents
2000-01-01 Gitto, Rosaria; Chimirri, Alba; Zappala', Maria; DE SARRO, G; DE SARRO, Angelina
Synthesis and structural features of new cyclofunctionalized benzimidazoles
2000-01-01 Chimirri, Alba; Monforte, Anna Maria; Monforte, Pietro; Nicolo', Francesco; Rao, Angela; Zappala', Maria
Synthesis and evaluation of pharmacological and pharmacokinetic properties of 11H-[1,2,4]triazolo[4,5-c][2,3]benzodiazepin- 3(2H)-ones
2000-01-01 Zappala', Maria; Gitto, Rosaria; Bevacqua, F; Quartarone, S; Chimirri, Alba; Rizzo, M; DE SARRO, G; DE SARRO, Angelina
Synthesis and metabolic study of 1H,3H-oxazolo[3,4-a]benzimidazoles, a new class of non-nucleoside HIV-1 RT-inhibitors.
2000-01-01 Chimirri, Alba; E., DE CLERCQ; Monforte, Anna Maria; Monforte, Pietro; C., Pannecouque; Rao, Angela; M., Witvrouw; Zappala', Maria
Benzimidazole derivatives: role of cyclofunctionalization on selectivity against HIV-1 or HIV-2
2000-01-01 Chimirri, Alba; Monforte, Anna Maria; P., Monforte; L., Musumeci; A., Rao; M., Zappal; M., Witvrouw; E., DE CLERCQ
New noncompetitive AMPA-receptor antagonists structural analogues of CFMs
2001-01-01 Gitto, Rosaria; G., DE SARRO; Chimirri, Alba; S., Quartarone; V., Orlando; A., Chimirri
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
HIV-1 RT inhibitors containing a cyclofunctionalized benzimidazole system | 1-gen-1999 | Chimirri, Alba; E., DE CLERCQ; Grasso, Silvana; Monforte, Anna Maria; P., Monforte; C., Pannecouque; A., Rao; M., Witvrouw; Zappala', Maria | |
Synthesis and anticonvulsant activity of new 11H-triazolo[4,5- c] [2,3]benzodiazepines | 1-gen-1999 | Chimirri, Alba; Bevacqua, F; Gitto, Rosaria; Quartarone, S; Zappala', Maria; DE SARRO, Angelina; Maciocco, L; Biggio, G; DE SARRO, G. | |
Synthesis and structural features of 11H-tetrazolo[1,5-c][2,3]benzodiazepines | 1-gen-1999 | Chimirri, Alba; Zappala', Maria; Gitto, Rosaria; Quartarone, S.; Bevacqua, F. | |
Anticonvulsant activity and plasma level of 2,3-benzodiazepin-4-ones (CFMs) in genetically epilepsy prone rats | 1-gen-1999 | G., DE SARRO; M., Rizzo; Gitto, Rosaria; Zappala', Maria; Chimirri, Alba; A., DE SARRO | |
Anticonvulsant activity and plasma level of 2,3-benzodiazepin- 4-ones (CFMs) in genetically epilepsy-prone rats | 1-gen-1999 | DE SARRO, G; Rizzo, M; Spagnolo, C; Gitto, Rosaria; DE SARRO, Angelina; Scotto, G; Zappala', Maria; Chimirri, Alba | |
7,11b-dihydro-9,10-dimethoxy-3,11b- diphenyl[1,2,4]oxadiazolo[5,4-a]-[2,3]benzodiazepin-6(5H)-one | 1-gen-1999 | BRUNO G; CHIMIRRI A; GITTO R; NICOLO' FRANCESCO; SCOPELLITI R | |
Determination of 2,3-benzodiazepine derivatives in rat plasma by high-performance liquid chromatography | 1-gen-1999 | RIZZO M; DE SARRO G; GITTO R; ZAPPALA M; CHIMIRRI A. | |
Synthesis and biological activity of novel 1H,3H-thiazolo[3,4- a] benzimidazoles: non-nucleoside human immunodeficiency virus type 1 reverse transcriptase inhibitors | 1-gen-1999 | Chimirri, Alba; Grasso, Silvana; Monforte, Pietro; Rao, Angela; Zappala', Maria; Monforte, Anna Maria; Pannecouque, C; Witvrouw, M; Balzarini, J; DE CLERCQ, E. | |
Synthesis, structural features and anti-HIV activity of TBZ analogues | 1-gen-1999 | Chimirri, Alba; Monforte, Anna Maria; P., Monforte; L., Musumeci; A., Rao; M., Zappal; M., Witvrouw; E., DE CLERCQ | |
Comparative molecular field analysis (CoMFA) and docking studies of non-nucleoside HIV-1 RT inhibitors (NNIs) | 1-gen-1999 | Barreca, Maria Letizia; Carotti, A; Carrieri, A; Chimirri, Alba; Monforte, Anna Maria; Calace, Mp; Rao, Angela | |
AMPA receptor antagonists | 1-gen-1999 | Chimirri, Alba; Gitto, Rosaria; Zappala', Maria | |
Development of 2,3-benzodiazepines and related AMPA receptor antagonists | 1-gen-2000 | Gitto, Rosaria; Chimirri, Alba; Zappala', Maria; Quartarone, S.; Bevacqua, F.; DE SARRO, A.; DE SARRO, G. | |
Sintesi ed effetti apoptotici di derivati tiazolobenzimidazolici antitumorali | 1-gen-2000 | Chimirri, Alba; P., Monforte; L., Musumeci; A., Rao; M. ZAPPAL A. M., Monforte; V. L., Narayanan | |
Design and development of 2,3-benzodiazepine (CFM) noncompetitive AMPA receptor antagonists | 1-gen-2000 | Gitto, Rosaria; Zappala', Maria; Chimirri, Alba; G., DE SARRO | |
Synthesis and pharmacological evaluation of 4-aryl-6,7- dimethoxyphthalazines as anticonvulsant agents | 1-gen-2000 | Gitto, Rosaria; Chimirri, Alba; Zappala', Maria; DE SARRO, G; DE SARRO, Angelina | |
Synthesis and structural features of new cyclofunctionalized benzimidazoles | 1-gen-2000 | Chimirri, Alba; Monforte, Anna Maria; Monforte, Pietro; Nicolo', Francesco; Rao, Angela; Zappala', Maria | |
Synthesis and evaluation of pharmacological and pharmacokinetic properties of 11H-[1,2,4]triazolo[4,5-c][2,3]benzodiazepin- 3(2H)-ones | 1-gen-2000 | Zappala', Maria; Gitto, Rosaria; Bevacqua, F; Quartarone, S; Chimirri, Alba; Rizzo, M; DE SARRO, G; DE SARRO, Angelina | |
Synthesis and metabolic study of 1H,3H-oxazolo[3,4-a]benzimidazoles, a new class of non-nucleoside HIV-1 RT-inhibitors. | 1-gen-2000 | Chimirri, Alba; E., DE CLERCQ; Monforte, Anna Maria; Monforte, Pietro; C., Pannecouque; Rao, Angela; M., Witvrouw; Zappala', Maria | |
Benzimidazole derivatives: role of cyclofunctionalization on selectivity against HIV-1 or HIV-2 | 1-gen-2000 | Chimirri, Alba; Monforte, Anna Maria; P., Monforte; L., Musumeci; A., Rao; M., Zappal; M., Witvrouw; E., DE CLERCQ | |
New noncompetitive AMPA-receptor antagonists structural analogues of CFMs | 1-gen-2001 | Gitto, Rosaria; G., DE SARRO; Chimirri, Alba; S., Quartarone; V., Orlando; A., Chimirri |
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