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A refined pharmacophore model for HIV-1 integrase inhibitors: Optimization of potency in the 1H-benzylindole series 1-gen-2008 DE LUCA, Laura; Barreca, Maria Letizia; Ferro, Stefania; Iraci, Nunzio; Michiels, M; Christ, F; Debyser, Z; Witvrouw, M; Chimirri, Alba
Computational Studies to Discover a New NR2B/NMDA Receptor Antagonist and Evaluation of Pharmacological Profile 1-gen-2008 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Occhiuto, Francesco; Samperi, S; DE SARRO, G; Russo, E; Ciranna, L; Costa, LARA TANIA; Chimirri, Alba
Preclinical evaluation of 1H-benzylindole derivatives as novel human immunodeficiency virus integrase strand transfer inhibitors 1-gen-2008 HOMBROUCK A; VAN REMOORTEL B; MICHIELS M; NOPPE W; CHRIST F; ENEROTH A; SAHLBERG BL; BENKESTOCK K; VRANG L; JOHANSSON NG; BARRECA ML; DE LUCA L.; FERRO S; CHIMIRRI A; DEBYSER Z; WITVROUW M
Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside riverse transcriptase inhibitors 1-gen-2008 Monforte, Anna Maria; Rao, A; Logoteta, Patrizia; Ferro, Stefania; DE LUCA, Laura; Barreca, Maria Letizia; Iraci, Nunzio; Maga, G; DE CLERCQ, E; Pannecouque, C; Chimirri, Alba
Design, synthesis and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents 1-gen-2009 Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; De Clercq, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria
Identification of potent carbonic anhydrase inhibitors: synthesis, biological evaluation and enzyme-ligand x-ray studies 1-gen-2009 Gitto, Rosaria; Agnello, Stefano; Ferro, Stefania; Supuran, Ct; Brynda, J; Mader, P; Chimirri, Alba
Antiretroviral strategy using multi-target agents 1-gen-2009 Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; Gitto, Rosaria; Monforte, Anna Maria; Barreca, Ml; Christ, F; Chimirri, Alba
Discovery of HIV-1 Integrase and cellular cofactor LEDGF/p75 interaction inhibitors 1-gen-2009 Ferro, Stefania; Agnello, Stefano; DE LUCA, Laura; Barreca, Ml; Iraci, N; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
Discovery of rationally designed small molecules as neuroprotectiveagents 1-gen-2009 Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; De Sarro, G; Ciranna, L; Gitto, Rosaria
Optimization of indolediketoacids, potent HIV-1 integrase strand transfer inhibitors 1-gen-2009 DE LUCA, Laura; DE GRAZIA, Sara; Ferro, Stefania; Barreca, Ml; Debyser, Z; Chimirri, Alba
1-Aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1H)-sulfonamide derivatives: synthesis and biological evaluation 1-gen-2009 Agnello, Stefano; Ferro, Stefania; Gitto, Rosaria; De Sarro, G; Russo, E; Vullo, D; Supuran T., C; Chimirri, Alba
Progettazione e sintesi di antagonisti non competitivi del recettore NR2B/NMDA 1-gen-2009 Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Scicchitano, F; Maierù, Mt; Gitto, Rosaria
Nuovi ligandi del recettore NR2B/NMDA a struttura indolica 1-gen-2009 Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Chimirri, Alba
Discovery of potent HIV-1 integrase strand transfer inhibitors: design and synthetic strategies 1-gen-2009 DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Debyser, Z; Chimirri, Alba
From 3D-pharmacophore models to synthetic route towards anti-HIV agents 1-gen-2009 Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; DE GRAZIA, Sara; Iraci, Nunzio; Barreca, Ml; Debyser, Z.
New potent and selective carbonic anhydrase inhibitors: synthesis, biological evaluation and X-ray studies 1-gen-2009 Ferro, Stefania; Gitto, Rosaria; Agnello, Stefano; Claudiu T., Supuran; Jiri, Brynda; Pavel, Mader; Chimirri, Alba
Novel targets for HIV therapy: small molecules blocking IN-LEDGF/p75 interaction 1-gen-2009 Ferro, Stefania; DE LUCA, Laura; Agnello, Stefano; Barreca, Ml; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
Derivati benzimidazolonici ed analoghi come potenti inibitori non-nucleosidici dell'RT dell'HIV-1 1-gen-2009 Logoteta, Patrizia; DE LUCA, Laura; Ferro, Stefania; De Clercq, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria
Optimization of a potent HIV-1 integrase strand transfer inhibitor (INSTI): molecular modeling, synthesis and anti-HIV activity 1-gen-2009 DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Debyser, Z; Chimirri, Alba
Pharmacophore-based discovery of small-molecule inhibitors of protein-protein interactions between HIV-1 integrase and cellular cofactor LEDGF/p75 1-gen-2009 DE LUCA, Laura; Barreca, Ml; Ferro, Stefania; Christ, F; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Debyser, Z; Chimirri, Alba
Mostrati risultati da 61 a 80 di 173
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