Sfoglia per Autore
A refined pharmacophore model for HIV-1 integrase inhibitors: Optimization of potency in the 1H-benzylindole series
2008-01-01 DE LUCA, Laura; Barreca, Maria Letizia; Ferro, Stefania; Iraci, Nunzio; Michiels, M; Christ, F; Debyser, Z; Witvrouw, M; Chimirri, Alba
Computational Studies to Discover a New NR2B/NMDA Receptor Antagonist and Evaluation of Pharmacological Profile
2008-01-01 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Occhiuto, Francesco; Samperi, S; DE SARRO, G; Russo, E; Ciranna, L; Costa, LARA TANIA; Chimirri, Alba
Preclinical evaluation of 1H-benzylindole derivatives as novel human immunodeficiency virus integrase strand transfer inhibitors
2008-01-01 HOMBROUCK A; VAN REMOORTEL B; MICHIELS M; NOPPE W; CHRIST F; ENEROTH A; SAHLBERG BL; BENKESTOCK K; VRANG L; JOHANSSON NG; BARRECA ML; DE LUCA L.; FERRO S; CHIMIRRI A; DEBYSER Z; WITVROUW M
Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside riverse transcriptase inhibitors
2008-01-01 Monforte, Anna Maria; Rao, A; Logoteta, Patrizia; Ferro, Stefania; DE LUCA, Laura; Barreca, Maria Letizia; Iraci, Nunzio; Maga, G; DE CLERCQ, E; Pannecouque, C; Chimirri, Alba
Design, synthesis and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents
2009-01-01 Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; De Clercq, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria
Identification of potent carbonic anhydrase inhibitors: synthesis, biological evaluation and enzyme-ligand x-ray studies
2009-01-01 Gitto, Rosaria; Agnello, Stefano; Ferro, Stefania; Supuran, Ct; Brynda, J; Mader, P; Chimirri, Alba
Antiretroviral strategy using multi-target agents
2009-01-01 Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; Gitto, Rosaria; Monforte, Anna Maria; Barreca, Ml; Christ, F; Chimirri, Alba
Discovery of HIV-1 Integrase and cellular cofactor LEDGF/p75 interaction inhibitors
2009-01-01 Ferro, Stefania; Agnello, Stefano; DE LUCA, Laura; Barreca, Ml; Iraci, N; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
Discovery of rationally designed small molecules as neuroprotectiveagents
2009-01-01 Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; De Sarro, G; Ciranna, L; Gitto, Rosaria
Optimization of indolediketoacids, potent HIV-1 integrase strand transfer inhibitors
2009-01-01 DE LUCA, Laura; DE GRAZIA, Sara; Ferro, Stefania; Barreca, Ml; Debyser, Z; Chimirri, Alba
1-Aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1H)-sulfonamide derivatives: synthesis and biological evaluation
2009-01-01 Agnello, Stefano; Ferro, Stefania; Gitto, Rosaria; De Sarro, G; Russo, E; Vullo, D; Supuran T., C; Chimirri, Alba
Progettazione e sintesi di antagonisti non competitivi del recettore NR2B/NMDA
2009-01-01 Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Scicchitano, F; Maierù, Mt; Gitto, Rosaria
Nuovi ligandi del recettore NR2B/NMDA a struttura indolica
2009-01-01 Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Chimirri, Alba
Discovery of potent HIV-1 integrase strand transfer inhibitors: design and synthetic strategies
2009-01-01 DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Debyser, Z; Chimirri, Alba
From 3D-pharmacophore models to synthetic route towards anti-HIV agents
2009-01-01 Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; DE GRAZIA, Sara; Iraci, Nunzio; Barreca, Ml; Debyser, Z.
New potent and selective carbonic anhydrase inhibitors: synthesis, biological evaluation and X-ray studies
2009-01-01 Ferro, Stefania; Gitto, Rosaria; Agnello, Stefano; Claudiu T., Supuran; Jiri, Brynda; Pavel, Mader; Chimirri, Alba
Novel targets for HIV therapy: small molecules blocking IN-LEDGF/p75 interaction
2009-01-01 Ferro, Stefania; DE LUCA, Laura; Agnello, Stefano; Barreca, Ml; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
Derivati benzimidazolonici ed analoghi come potenti inibitori non-nucleosidici dell'RT dell'HIV-1
2009-01-01 Logoteta, Patrizia; DE LUCA, Laura; Ferro, Stefania; De Clercq, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria
Optimization of a potent HIV-1 integrase strand transfer inhibitor (INSTI): molecular modeling, synthesis and anti-HIV activity
2009-01-01 DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Debyser, Z; Chimirri, Alba
Pharmacophore-based discovery of small-molecule inhibitors of protein-protein interactions between HIV-1 integrase and cellular cofactor LEDGF/p75
2009-01-01 DE LUCA, Laura; Barreca, Ml; Ferro, Stefania; Christ, F; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Debyser, Z; Chimirri, Alba
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A refined pharmacophore model for HIV-1 integrase inhibitors: Optimization of potency in the 1H-benzylindole series | 1-gen-2008 | DE LUCA, Laura; Barreca, Maria Letizia; Ferro, Stefania; Iraci, Nunzio; Michiels, M; Christ, F; Debyser, Z; Witvrouw, M; Chimirri, Alba | |
Computational Studies to Discover a New NR2B/NMDA Receptor Antagonist and Evaluation of Pharmacological Profile | 1-gen-2008 | Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Occhiuto, Francesco; Samperi, S; DE SARRO, G; Russo, E; Ciranna, L; Costa, LARA TANIA; Chimirri, Alba | |
Preclinical evaluation of 1H-benzylindole derivatives as novel human immunodeficiency virus integrase strand transfer inhibitors | 1-gen-2008 | HOMBROUCK A; VAN REMOORTEL B; MICHIELS M; NOPPE W; CHRIST F; ENEROTH A; SAHLBERG BL; BENKESTOCK K; VRANG L; JOHANSSON NG; BARRECA ML; DE LUCA L.; FERRO S; CHIMIRRI A; DEBYSER Z; WITVROUW M | |
Novel N1-substituted 1,3-dihydro-2H-benzimidazol-2-ones as potent non-nucleoside riverse transcriptase inhibitors | 1-gen-2008 | Monforte, Anna Maria; Rao, A; Logoteta, Patrizia; Ferro, Stefania; DE LUCA, Laura; Barreca, Maria Letizia; Iraci, Nunzio; Maga, G; DE CLERCQ, E; Pannecouque, C; Chimirri, Alba | |
Design, synthesis and structure-activity relationships of 1,3-dihydrobenzimidazol-2-one analogues as anti-HIV agents | 1-gen-2009 | Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; De Clercq, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria | |
Identification of potent carbonic anhydrase inhibitors: synthesis, biological evaluation and enzyme-ligand x-ray studies | 1-gen-2009 | Gitto, Rosaria; Agnello, Stefano; Ferro, Stefania; Supuran, Ct; Brynda, J; Mader, P; Chimirri, Alba | |
Antiretroviral strategy using multi-target agents | 1-gen-2009 | Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; Gitto, Rosaria; Monforte, Anna Maria; Barreca, Ml; Christ, F; Chimirri, Alba | |
Discovery of HIV-1 Integrase and cellular cofactor LEDGF/p75 interaction inhibitors | 1-gen-2009 | Ferro, Stefania; Agnello, Stefano; DE LUCA, Laura; Barreca, Ml; Iraci, N; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba | |
Discovery of rationally designed small molecules as neuroprotectiveagents | 1-gen-2009 | Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; De Sarro, G; Ciranna, L; Gitto, Rosaria | |
Optimization of indolediketoacids, potent HIV-1 integrase strand transfer inhibitors | 1-gen-2009 | DE LUCA, Laura; DE GRAZIA, Sara; Ferro, Stefania; Barreca, Ml; Debyser, Z; Chimirri, Alba | |
1-Aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1H)-sulfonamide derivatives: synthesis and biological evaluation | 1-gen-2009 | Agnello, Stefano; Ferro, Stefania; Gitto, Rosaria; De Sarro, G; Russo, E; Vullo, D; Supuran T., C; Chimirri, Alba | |
Progettazione e sintesi di antagonisti non competitivi del recettore NR2B/NMDA | 1-gen-2009 | Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Scicchitano, F; Maierù, Mt; Gitto, Rosaria | |
Nuovi ligandi del recettore NR2B/NMDA a struttura indolica | 1-gen-2009 | Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Chimirri, Alba | |
Discovery of potent HIV-1 integrase strand transfer inhibitors: design and synthetic strategies | 1-gen-2009 | DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Debyser, Z; Chimirri, Alba | |
From 3D-pharmacophore models to synthetic route towards anti-HIV agents | 1-gen-2009 | Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; DE GRAZIA, Sara; Iraci, Nunzio; Barreca, Ml; Debyser, Z. | |
New potent and selective carbonic anhydrase inhibitors: synthesis, biological evaluation and X-ray studies | 1-gen-2009 | Ferro, Stefania; Gitto, Rosaria; Agnello, Stefano; Claudiu T., Supuran; Jiri, Brynda; Pavel, Mader; Chimirri, Alba | |
Novel targets for HIV therapy: small molecules blocking IN-LEDGF/p75 interaction | 1-gen-2009 | Ferro, Stefania; DE LUCA, Laura; Agnello, Stefano; Barreca, Ml; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba | |
Derivati benzimidazolonici ed analoghi come potenti inibitori non-nucleosidici dell'RT dell'HIV-1 | 1-gen-2009 | Logoteta, Patrizia; DE LUCA, Laura; Ferro, Stefania; De Clercq, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria | |
Optimization of a potent HIV-1 integrase strand transfer inhibitor (INSTI): molecular modeling, synthesis and anti-HIV activity | 1-gen-2009 | DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Debyser, Z; Chimirri, Alba | |
Pharmacophore-based discovery of small-molecule inhibitors of protein-protein interactions between HIV-1 integrase and cellular cofactor LEDGF/p75 | 1-gen-2009 | DE LUCA, Laura; Barreca, Ml; Ferro, Stefania; Christ, F; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Debyser, Z; Chimirri, Alba |
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