Sfoglia per Autore
1,3-diidro-benzimidazoloni analoghi: progettazione, sintesi e SAR di nuovi inibitori non-nucleosidici dell'RT
2007-01-01 Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; Barreca, Maria Letizia; DE CLERCQ, E.; Chimirri, Alba; Monforte, Anna Maria
Rational design, synthesis and SAR of 1,3-dihydro-benzimidazolone analogues as new anti-HIV agents
2007-01-01 Logoteta, Patrizia; Iraci, N; DE LUCA, Laura; Ferro, Stefania; Barreca, Ml; DE CLERCQ, E; Chimirri, Alba; Monforte, Anna Maria
Progettazione, Sintesi e SAR di analoghi 1,3-diidro-benzimidazoloni come nuovi agenti anti-HIV
2007-01-01 Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; Barreca, M. L.; DE CLERCQ, E.; Chimirri, Alba; Monforte, Anna Maria
Structure-Based Pharmacophore Identification of New Chemical Scaffolds as Non –Nucleoside riverse Transcriptase Inhibitors
2007-01-01 DE LUCA, Laura; Barreca, Ml; Iraci, Nunzio; Ferro, Stefania; Monforte, Am; Maga, G; Chimirri, A.
AMPA receptor antagonists: Synthesis and pharmacological evaluation
2007-01-01 Gitto, Rosaria; DE LUCA, Laura; Pagano, B; Ferro, Stefania; DE SARRO, G; Citraro, R; Ciranna, L; Costa, LARA TANIA; Chimirri, Alba
Structure-based pharmacophore identification of new chemical scaffolds as non-nucleoside reverse transcriptase inhibitors
2007-01-01 Barreca, Maria Letizia; DE LUCA, Laura; Iraci, Nunzio; Rao, A; Ferro, Stefania; Maga, G; Chimirri, Alba
HIV-1 integrase inhibitors as anti-AIDS agents: Structure-Activity Relationships (SAR) of new diketo acids and analogs
2007-01-01 Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Rao, A; Manforte, Am; Debyser, Z; Witvrouw, M; Chimirri, Alba
New 4-[(1-benzyl-1H-indol-3-yl)carbonyl]-3-hydroxyfuran-2(5H)-ones, β-diketo acid analogs, as HIV-1 integrase inhibitors
2007-01-01 Ferro, Stefania; Barreca, Ml; DE LUCA, Laura; Rao, A; Monforte, Anna Maria; Chimirri, Alba
PROGETTAZIONE E SINTESI DI NUOVI DKA ANALOGHI COME POTENZIALI INIBITORI DELL’INTEGRASI DELL’HIV-1
2008-01-01 Agnello, Stefano; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Debyser, Z; Chimirri, Alba
MOLECULAR MODELING STUDIES AND SYNTHESIS FOR THE DISCOVERY OF HIV-1 IN-LEDGF/P75 INTERACTION INHIBITORS
2008-01-01 Ferro, Stefania; DE LUCA, Laura; BARRECA M., L; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
Synthesis and SAR of new 1,3-dihydro-benzimidazolone analogues as non-nucleoside reverse transcriptase inhibitors (NNRTIs)
2008-01-01 Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; DE CLERCQ, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria
HIV-1-IN Strand-Transfer Inhibitors: phenyl ring exploration and synthesis of 1H-benzylindole derivative through fluorine substitutions
2008-01-01 Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Iraci, Nunzio; DE GRAZIA, Sara; Debyser, Z; Witvrouw, M; Chimirri, Alba
A refined pharmacophore model and optimization of 1H-benzylindole HIV-1 integrase inhibitors
2008-01-01 DE LUCA, Laura; Barreca, Ml; Ferro, Stefania; Iraci, Nunzio; Debyser, Z; Witvrouw, M; Chimirri, Alba
Combined ligand-based and target-based approach to design NR2B/NMDA receptor antagonists
2008-01-01 Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Gitto, R.
PROGETTAZIONE E SINTESI DI NUOVI DERIVATI ISOCHINOLINICI COME AGENTI ANTICONVULSIVANTI MULTITARGET
2008-01-01 Agnello, Stefano; Ferro, Stefania; DE SARRO, G; Russo, E; Supuran, C; Gitto, Rosaria; Chimirri, Alba
Combined strategies for the discovery of ionotropic glutamate receptor antagonists
2008-01-01 Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; DE SARRO, G; Ciranna, L.; Gitto, Rosaria
New Indole derivatives as NMDA/NR2B rrceptor antagonists: design, synthesis and pharmacological properties
2008-01-01 Ferro, Stefania; Gitto, Rosaria; DE LUCA, Laura; DE SARRO, G; Russo, E; Ciranna, L; Costa, LARA TANIA; Chimirri, Alba
INTEGRASE STRAND TRANSFER INHIBITORS (INSTIs): SYNTHESIS AND ANTIVIRAL EFFETCS OF CHLORO-FLUORO SUBSTITUTIONS
2008-01-01 Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; MARIA LETIZIA, Barreca; Iraci, Nunzio; Frauke, Christ; Zeger, Debyser; Chimirri, Alba
Molecular modeling and synthesis for the discovery of HIV-1 IN-LEDGF/P75 interaction inhibitors.
2008-01-01 Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Iraci, N; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
A refined pharmacophore model for HIV-1 integrase inhibitors: Optimization of potency in the 1H-benzylindole series
2008-01-01 DE LUCA, Laura; Barreca, Maria Letizia; Ferro, Stefania; Iraci, Nunzio; Michiels, M; Christ, F; Debyser, Z; Witvrouw, M; Chimirri, Alba
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1,3-diidro-benzimidazoloni analoghi: progettazione, sintesi e SAR di nuovi inibitori non-nucleosidici dell'RT | 1-gen-2007 | Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; Barreca, Maria Letizia; DE CLERCQ, E.; Chimirri, Alba; Monforte, Anna Maria | |
Rational design, synthesis and SAR of 1,3-dihydro-benzimidazolone analogues as new anti-HIV agents | 1-gen-2007 | Logoteta, Patrizia; Iraci, N; DE LUCA, Laura; Ferro, Stefania; Barreca, Ml; DE CLERCQ, E; Chimirri, Alba; Monforte, Anna Maria | |
Progettazione, Sintesi e SAR di analoghi 1,3-diidro-benzimidazoloni come nuovi agenti anti-HIV | 1-gen-2007 | Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; Barreca, M. L.; DE CLERCQ, E.; Chimirri, Alba; Monforte, Anna Maria | |
Structure-Based Pharmacophore Identification of New Chemical Scaffolds as Non –Nucleoside riverse Transcriptase Inhibitors | 1-gen-2007 | DE LUCA, Laura; Barreca, Ml; Iraci, Nunzio; Ferro, Stefania; Monforte, Am; Maga, G; Chimirri, A. | |
AMPA receptor antagonists: Synthesis and pharmacological evaluation | 1-gen-2007 | Gitto, Rosaria; DE LUCA, Laura; Pagano, B; Ferro, Stefania; DE SARRO, G; Citraro, R; Ciranna, L; Costa, LARA TANIA; Chimirri, Alba | |
Structure-based pharmacophore identification of new chemical scaffolds as non-nucleoside reverse transcriptase inhibitors | 1-gen-2007 | Barreca, Maria Letizia; DE LUCA, Laura; Iraci, Nunzio; Rao, A; Ferro, Stefania; Maga, G; Chimirri, Alba | |
HIV-1 integrase inhibitors as anti-AIDS agents: Structure-Activity Relationships (SAR) of new diketo acids and analogs | 1-gen-2007 | Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Rao, A; Manforte, Am; Debyser, Z; Witvrouw, M; Chimirri, Alba | |
New 4-[(1-benzyl-1H-indol-3-yl)carbonyl]-3-hydroxyfuran-2(5H)-ones, β-diketo acid analogs, as HIV-1 integrase inhibitors | 1-gen-2007 | Ferro, Stefania; Barreca, Ml; DE LUCA, Laura; Rao, A; Monforte, Anna Maria; Chimirri, Alba | |
PROGETTAZIONE E SINTESI DI NUOVI DKA ANALOGHI COME POTENZIALI INIBITORI DELL’INTEGRASI DELL’HIV-1 | 1-gen-2008 | Agnello, Stefano; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Debyser, Z; Chimirri, Alba | |
MOLECULAR MODELING STUDIES AND SYNTHESIS FOR THE DISCOVERY OF HIV-1 IN-LEDGF/P75 INTERACTION INHIBITORS | 1-gen-2008 | Ferro, Stefania; DE LUCA, Laura; BARRECA M., L; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba | |
Synthesis and SAR of new 1,3-dihydro-benzimidazolone analogues as non-nucleoside reverse transcriptase inhibitors (NNRTIs) | 1-gen-2008 | Logoteta, Patrizia; Iraci, Nunzio; DE LUCA, Laura; Ferro, Stefania; DE CLERCQ, E; Maga, G; Chimirri, Alba; Monforte, Anna Maria | |
HIV-1-IN Strand-Transfer Inhibitors: phenyl ring exploration and synthesis of 1H-benzylindole derivative through fluorine substitutions | 1-gen-2008 | Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Iraci, Nunzio; DE GRAZIA, Sara; Debyser, Z; Witvrouw, M; Chimirri, Alba | |
A refined pharmacophore model and optimization of 1H-benzylindole HIV-1 integrase inhibitors | 1-gen-2008 | DE LUCA, Laura; Barreca, Ml; Ferro, Stefania; Iraci, Nunzio; Debyser, Z; Witvrouw, M; Chimirri, Alba | |
Combined ligand-based and target-based approach to design NR2B/NMDA receptor antagonists | 1-gen-2008 | Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Gitto, R. | |
PROGETTAZIONE E SINTESI DI NUOVI DERIVATI ISOCHINOLINICI COME AGENTI ANTICONVULSIVANTI MULTITARGET | 1-gen-2008 | Agnello, Stefano; Ferro, Stefania; DE SARRO, G; Russo, E; Supuran, C; Gitto, Rosaria; Chimirri, Alba | |
Combined strategies for the discovery of ionotropic glutamate receptor antagonists | 1-gen-2008 | Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; DE SARRO, G; Ciranna, L.; Gitto, Rosaria | |
New Indole derivatives as NMDA/NR2B rrceptor antagonists: design, synthesis and pharmacological properties | 1-gen-2008 | Ferro, Stefania; Gitto, Rosaria; DE LUCA, Laura; DE SARRO, G; Russo, E; Ciranna, L; Costa, LARA TANIA; Chimirri, Alba | |
INTEGRASE STRAND TRANSFER INHIBITORS (INSTIs): SYNTHESIS AND ANTIVIRAL EFFETCS OF CHLORO-FLUORO SUBSTITUTIONS | 1-gen-2008 | Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; MARIA LETIZIA, Barreca; Iraci, Nunzio; Frauke, Christ; Zeger, Debyser; Chimirri, Alba | |
Molecular modeling and synthesis for the discovery of HIV-1 IN-LEDGF/P75 interaction inhibitors. | 1-gen-2008 | Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Iraci, N; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba | |
A refined pharmacophore model for HIV-1 integrase inhibitors: Optimization of potency in the 1H-benzylindole series | 1-gen-2008 | DE LUCA, Laura; Barreca, Maria Letizia; Ferro, Stefania; Iraci, Nunzio; Michiels, M; Christ, F; Debyser, Z; Witvrouw, M; Chimirri, Alba |
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