Sfoglia per Autore
Carbonic anhydrase inhibitors: Design, synthesis and structural characterization of new heteroaryl-N-carbonylbenzenesulfonamides targeting druggable human carbonic anhydrase isoforms
2015-01-01 Buemi, Mariarosa; DE LUCA, Laura; Ferro, Stefania; Bruno, Elvira; Ceruso, Mariangela; Supuran, Claudiu T; Pospíšilová, Klára; Brynda, Jiří; Řezáčová, Pavlína; Gitto, Rosaria
Serendipitous discovery of indole derivatives as potent tyrosinase inhibitors
2015-01-01 Gitto, Rosaria; Buemi, Mariarosa; DE LUCA, Laura; Certo, Giovanna; Germano', Maria Paola; Rapisarda, Antonio; Ferro, Stefania
InVivo Evaluation of Selective Carbonic Anhydrase Inhibitors as Potential Anticonvulsant Agents
2016-01-01 Bruno, Elvira; Buemi, Mariarosa; DE LUCA, Laura; Ferro, Stefania; Monforte, Anna Maria; Supuran, Claudiu T.; Vullo, Daniela; De Sarro, Giovambattista; Russo, Emilio; Gitto, Rosaria
Rational design, synthesis and evaluation of coumarin derivatives as protein-protein interaction inhibitors
2016-01-01 DE LUCA, Laura; Agharbaoui, FATIMA EZZAHRA; Gitto, Rosaria; Buemi, Mariarosa; Christ, Frauke; Debyser, Zeger; Ferro, Stefania
Structure-guided design of new indoles as negative allosteric modulators (NAMs) of N-methyl-d-aspartate receptor (NMDAR) containing GluN2B subunit
2016-01-01 Buemi, Mariarosa; De Luca, Laura; Ferro, Stefania; Russo, Emilio; De Sarro, Giovambattista; Gitto, Rosaria
Computational and synthetic approaches for developing Lavendustin B derivatives as allosteric inhibitors of HIV-1 integrase
2016-01-01 Agharbaoui, Fatima Ezzahra; Hoyte, Ashley C.; Ferro, Stefania; Gitto, Rosaria; Buemi, Mariarosa; Fuchs, James R.; Kvaratskhelia, Mamuka; De Luca, Laura
Chemical exploration of 4-(4-fluorobenzyl)piperidine fragment for the development of new tyrosinase inhibitors
2017-01-01 Ferro, Stefania; DE LUCA, Laura; Germano', Maria Paola; Buemi, Mariarosa; Ielo, Laura; Certo, Giovanna; Kanteev, Margarita; Fishman, Ayelet; Rapisarda, Antonio; Gitto, Rosaria
Searching for novel N1-substituted benzimidazol-2-ones as non-nucleoside HIV-1 RT inhibitors
2017-01-01 Ferro, Stefania; Buemi, Maria Rosa; De Luca, Laura; Agharbaoui, Fatima E.; Pannecouque, Christophe; Monforte, Anna-Maria
Probing Molecular Interactions between Human Carbonic Anhydrases (hCAs) and a Novel Class of Benzenesulfonamides
2017-01-01 BRUNO, ELVIRA; BUEMI, MARIAROSA; Di Fiore, Anna; DE LUCA, Laura; FERRO, Stefania; Angeli, Andrea; Cirilli, Roberto; Sadutto, Daniele; Alterio, Vincenzo; Monti, Simona Maria; Supuran, Claudiu T.; De Simone, Giuseppina; GITTO, Rosaria
Discovery and optimization of isoquinoline-derived inhibitors of human Carbonic Anhydrases (hCAs)
2017-01-01 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Řezáčová, Pavlina; De Simone, Giuseppina; Supuran, Claudiu T.
Identification of influenza PA-Nter endonuclease inhibitors using pharmacophore- and docking-based virtual screening
2018-01-01 Ferro, S; Gitto, R; Buemi M., R; Karamanou, S; Stevaert, A; Naesens, L; Luca, De
Structural optimization of N1-aryl-benzimidazoles for the discovery of new non-nucleoside reverse transcriptase inhibitors active against wild-type and mutant HIV-1 strains
2018-01-01 Monforte, Anna Maria; De Luca, Laura; Buemi, Maria Rosa; Agharbaoui, Fatima E.; Pannecouque, Christophe; Ferro, Stefania
Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases
2018-01-01 De Luca, Laura; Mancuso, Francesca; Ferro, Stefania; Buemi, Maria Rosa; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria
Graphene Quantum Dots Based Systems As HIV Inhibitors
2018-01-01 Iannazzo, Daniela; Pistone, Alessandro; Ferro, Stefania; De Luca, Laura; Monforte, Anna Maria; Romeo, Roberto; Buemi, Mariarosa
Targeting Tyrosinase: Development and Structural Insights of Novel Inhibitors Bearing Arylpiperidine and Arylpiperazine Fragments
2018-01-01 Ferro, Stefania; Deri, Batel; Germanò, Maria Paola; Gitto, Rosaria; Ielo, Laura; Buemi, Maria Rosa; Certo, Giovanna; Vittorio, Serena; Rapisarda, Antonio; Pazy, Yael; Fishman, Ayelet; De Luca, Laura
Discovery of benzimidazole-based Leishmania mexicana cysteine protease CPB2.8ΔCTE inhibitors as potential therapeutics for leishmaniasis
2018-01-01 De Luca, Laura; Ferro, Stefania; Buemi, Maria Rosa; Monforte, Anna-Maria; Gitto, Rosaria; Schirmeister, Tanja; Maes, Louis; Rescifina, Antonio; Micale, Nicola
Exploring structural properties of potent human carbonic anhydrase inhibitors bearing a 4-(cycloalkylamino-1-carbonyl)benzenesulfonamide moiety
2019-01-01 Buemi, Maria Rosa; Di Fiore, Anna; De Luca, Laura; Angeli, Andrea; Mancuso, Francesca; Ferro, Stefania; Monti, Simona Maria; Buonanno, Martina; Russo, Emilio; De Sarro, Giovanbattista; De Simone, Giuseppina; Supuran, Claudiu T; Gitto, Rosaria
Inhibition of HIV-1 RT activity by a new series of 3-(1,3,4-thiadiazol-2-yl)thiazolidin-4-one derivatives
2020-01-01 Buemi, M. R.; Gitto, R.; Ielo, L.; Pannecouque, C.; De Luca, L.
Discovery of a new potent inhibitor of mushroom tyrosinase (Agaricus bisporus) containing 4-(4-hydroxyphenyl)piperazin-1-yl moiety
2020-01-01 De Luca, L.; Germano, M. P.; Fais, A.; Pintus, F.; Buemi, M. R.; Vittorio, S.; Mirabile, S.; Rapisarda, A.; Gitto, R.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Carbonic anhydrase inhibitors: Design, synthesis and structural characterization of new heteroaryl-N-carbonylbenzenesulfonamides targeting druggable human carbonic anhydrase isoforms | 1-gen-2015 | Buemi, Mariarosa; DE LUCA, Laura; Ferro, Stefania; Bruno, Elvira; Ceruso, Mariangela; Supuran, Claudiu T; Pospíšilová, Klára; Brynda, Jiří; Řezáčová, Pavlína; Gitto, Rosaria | |
Serendipitous discovery of indole derivatives as potent tyrosinase inhibitors | 1-gen-2015 | Gitto, Rosaria; Buemi, Mariarosa; DE LUCA, Laura; Certo, Giovanna; Germano', Maria Paola; Rapisarda, Antonio; Ferro, Stefania | |
InVivo Evaluation of Selective Carbonic Anhydrase Inhibitors as Potential Anticonvulsant Agents | 1-gen-2016 | Bruno, Elvira; Buemi, Mariarosa; DE LUCA, Laura; Ferro, Stefania; Monforte, Anna Maria; Supuran, Claudiu T.; Vullo, Daniela; De Sarro, Giovambattista; Russo, Emilio; Gitto, Rosaria | |
Rational design, synthesis and evaluation of coumarin derivatives as protein-protein interaction inhibitors | 1-gen-2016 | DE LUCA, Laura; Agharbaoui, FATIMA EZZAHRA; Gitto, Rosaria; Buemi, Mariarosa; Christ, Frauke; Debyser, Zeger; Ferro, Stefania | |
Structure-guided design of new indoles as negative allosteric modulators (NAMs) of N-methyl-d-aspartate receptor (NMDAR) containing GluN2B subunit | 1-gen-2016 | Buemi, Mariarosa; De Luca, Laura; Ferro, Stefania; Russo, Emilio; De Sarro, Giovambattista; Gitto, Rosaria | |
Computational and synthetic approaches for developing Lavendustin B derivatives as allosteric inhibitors of HIV-1 integrase | 1-gen-2016 | Agharbaoui, Fatima Ezzahra; Hoyte, Ashley C.; Ferro, Stefania; Gitto, Rosaria; Buemi, Mariarosa; Fuchs, James R.; Kvaratskhelia, Mamuka; De Luca, Laura | |
Chemical exploration of 4-(4-fluorobenzyl)piperidine fragment for the development of new tyrosinase inhibitors | 1-gen-2017 | Ferro, Stefania; DE LUCA, Laura; Germano', Maria Paola; Buemi, Mariarosa; Ielo, Laura; Certo, Giovanna; Kanteev, Margarita; Fishman, Ayelet; Rapisarda, Antonio; Gitto, Rosaria | |
Searching for novel N1-substituted benzimidazol-2-ones as non-nucleoside HIV-1 RT inhibitors | 1-gen-2017 | Ferro, Stefania; Buemi, Maria Rosa; De Luca, Laura; Agharbaoui, Fatima E.; Pannecouque, Christophe; Monforte, Anna-Maria | |
Probing Molecular Interactions between Human Carbonic Anhydrases (hCAs) and a Novel Class of Benzenesulfonamides | 1-gen-2017 | BRUNO, ELVIRA; BUEMI, MARIAROSA; Di Fiore, Anna; DE LUCA, Laura; FERRO, Stefania; Angeli, Andrea; Cirilli, Roberto; Sadutto, Daniele; Alterio, Vincenzo; Monti, Simona Maria; Supuran, Claudiu T.; De Simone, Giuseppina; GITTO, Rosaria | |
Discovery and optimization of isoquinoline-derived inhibitors of human Carbonic Anhydrases (hCAs) | 1-gen-2017 | Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Řezáčová, Pavlina; De Simone, Giuseppina; Supuran, Claudiu T. | |
Identification of influenza PA-Nter endonuclease inhibitors using pharmacophore- and docking-based virtual screening | 1-gen-2018 | Ferro, S; Gitto, R; Buemi M., R; Karamanou, S; Stevaert, A; Naesens, L; Luca, De | |
Structural optimization of N1-aryl-benzimidazoles for the discovery of new non-nucleoside reverse transcriptase inhibitors active against wild-type and mutant HIV-1 strains | 1-gen-2018 | Monforte, Anna Maria; De Luca, Laura; Buemi, Maria Rosa; Agharbaoui, Fatima E.; Pannecouque, Christophe; Ferro, Stefania | |
Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases | 1-gen-2018 | De Luca, Laura; Mancuso, Francesca; Ferro, Stefania; Buemi, Maria Rosa; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria | |
Graphene Quantum Dots Based Systems As HIV Inhibitors | 1-gen-2018 | Iannazzo, Daniela; Pistone, Alessandro; Ferro, Stefania; De Luca, Laura; Monforte, Anna Maria; Romeo, Roberto; Buemi, Mariarosa | |
Targeting Tyrosinase: Development and Structural Insights of Novel Inhibitors Bearing Arylpiperidine and Arylpiperazine Fragments | 1-gen-2018 | Ferro, Stefania; Deri, Batel; Germanò, Maria Paola; Gitto, Rosaria; Ielo, Laura; Buemi, Maria Rosa; Certo, Giovanna; Vittorio, Serena; Rapisarda, Antonio; Pazy, Yael; Fishman, Ayelet; De Luca, Laura | |
Discovery of benzimidazole-based Leishmania mexicana cysteine protease CPB2.8ΔCTE inhibitors as potential therapeutics for leishmaniasis | 1-gen-2018 | De Luca, Laura; Ferro, Stefania; Buemi, Maria Rosa; Monforte, Anna-Maria; Gitto, Rosaria; Schirmeister, Tanja; Maes, Louis; Rescifina, Antonio; Micale, Nicola | |
Exploring structural properties of potent human carbonic anhydrase inhibitors bearing a 4-(cycloalkylamino-1-carbonyl)benzenesulfonamide moiety | 1-gen-2019 | Buemi, Maria Rosa; Di Fiore, Anna; De Luca, Laura; Angeli, Andrea; Mancuso, Francesca; Ferro, Stefania; Monti, Simona Maria; Buonanno, Martina; Russo, Emilio; De Sarro, Giovanbattista; De Simone, Giuseppina; Supuran, Claudiu T; Gitto, Rosaria | |
Inhibition of HIV-1 RT activity by a new series of 3-(1,3,4-thiadiazol-2-yl)thiazolidin-4-one derivatives | 1-gen-2020 | Buemi, M. R.; Gitto, R.; Ielo, L.; Pannecouque, C.; De Luca, L. | |
Discovery of a new potent inhibitor of mushroom tyrosinase (Agaricus bisporus) containing 4-(4-hydroxyphenyl)piperazin-1-yl moiety | 1-gen-2020 | De Luca, L.; Germano, M. P.; Fais, A.; Pintus, F.; Buemi, M. R.; Vittorio, S.; Mirabile, S.; Rapisarda, A.; Gitto, R. |
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