BUEMI, MARIAROSA

BUEMI, MARIAROSA  

Dipartimento di Scienze chimiche, biologiche, farmaceutiche e ambientali  

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Risultati 1 - 20 di 39 (tempo di esecuzione: 0.08 secondi).
Titolo Data di pubblicazione Autore(i) File
Carbonic anhydrase inhibitors: Design, synthesis and structural characterization of new heteroaryl-N-carbonylbenzenesulfonamides targeting druggable human carbonic anhydrase isoforms 1-gen-2015 Buemi, Mariarosa; DE LUCA, Laura; Ferro, Stefania; Bruno, Elvira; Ceruso, Mariangela; Supuran, Claudiu T; Pospíšilová, Klára; Brynda, Jiří; Řezáčová, Pavlína; Gitto, Rosaria
Chemical exploration of 4-(4-fluorobenzyl)piperidine fragment for the development of new tyrosinase inhibitors 1-gen-2017 Ferro, Stefania; DE LUCA, Laura; Germano', Maria Paola; Buemi, Mariarosa; Ielo, Laura; Certo, Giovanna; Kanteev, Margarita; Fishman, Ayelet; Rapisarda, Antonio; Gitto, Rosaria
Computational and synthetic approaches for developing Lavendustin B derivatives as allosteric inhibitors of HIV-1 integrase 1-gen-2016 Agharbaoui, Fatima Ezzahra; Hoyte, Ashley C.; Ferro, Stefania; Gitto, Rosaria; Buemi, Mariarosa; Fuchs, James R.; Kvaratskhelia, Mamuka; De Luca, Laura
Design and optimization of isoquinoline-sulfonamides as potent and selective inhibitors of human carbonic anhydrase VII 1-gen-2014 Bruno, Elvira; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Ceruso, Mariangela; Supuran, Claudiu T.; Gitto, Rosaria
Design, Synthesis and Biostructural Characterization of Carbonic Anhydrase Inhibitors 1-gen-2013 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Vullo, D; Supuran, Ct; Brynda, J; Rezacova, P; Pospisilova, K; Damiano, F; Chimirri, Alba
Discovery and optimization of isoquinoline-derived inhibitors of human Carbonic Anhydrases (hCAs) 1-gen-2017 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; Řezáčová, Pavlina; De Simone, Giuseppina; Supuran, Claudiu T.
Discovery of a new potent inhibitor of mushroom tyrosinase (Agaricus bisporus) containing 4-(4-hydroxyphenyl)piperazin-1-yl moiety 1-gen-2020 De Luca, L.; Germano, M. P.; Fais, A.; Pintus, F.; Buemi, M. R.; Vittorio, S.; Mirabile, S.; Rapisarda, A.; Gitto, R.
Discovery of benzimidazole-based Leishmania mexicana cysteine protease CPB2.8ΔCTE inhibitors as potential therapeutics for leishmaniasis 1-gen-2018 De Luca, Laura; Ferro, Stefania; Buemi, Maria Rosa; Monforte, Anna-Maria; Gitto, Rosaria; Schirmeister, Tanja; Maes, Louis; Rescifina, Antonio; Micale, Nicola
DISCOVERY OF NEW INDOLE DERIVATES AS NEUROPROTECTIVE AGENTS 1-gen-2011 Buemi, Mariarosa; Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; R., Alajarin; J., ALVAREZ BUILLA; R., Citraro; Chimirri, Alba
Exploring structural properties of potent human carbonic anhydrase inhibitors bearing a 4-(cycloalkylamino-1-carbonyl)benzenesulfonamide moiety 1-gen-2019 Buemi, Maria Rosa; Di Fiore, Anna; De Luca, Laura; Angeli, Andrea; Mancuso, Francesca; Ferro, Stefania; Monti, Simona Maria; Buonanno, Martina; Russo, Emilio; De Sarro, Giovanbattista; De Simone, Giuseppina; Supuran, Claudiu T; Gitto, Rosaria
From NMDA receptor antagonists to discovery of selective σ2 receptor ligands 1-gen-2014 Rosaria Gitto;Laura De Luca;Stefania Ferro;Angela Scala;Simone Ronsisvalle;Carmela Parenti;Orazio Prezzavento;Maria Rosa Buemi;Alba Chimirri
Graphene Quantum Dots Based Systems As HIV Inhibitors 1-gen-2018 Iannazzo, Daniela; Pistone, Alessandro; Ferro, Stefania; De Luca, Laura; Monforte, Anna Maria; Romeo, Roberto; Buemi, Mariarosa
Identification of 3-substituted-1H-indoles as ligands of GluN2B containing N-methyl-D-aspartate receptors 1-gen-2012 Ferro, Stefania; Buemi, Mariarosa; Gitto, Rosaria; DE LUCA, Laura; Russo, E.; Ciranna, L.; Chimirri, Alba
Identification of influenza PA-Nter endonuclease inhibitors using pharmacophore- and docking-based virtual screening 1-gen-2018 Ferro, S; Gitto, R; Buemi M., R; Karamanou, S; Stevaert, A; Naesens, L; Luca, De
Indole derivatives as dual-effective agents for the treatment of neurodegenerative diseases: Synthesis, biological evaluation, and molecular modeling studies 1-gen-2013 Maria Rosa, Buemi; Laura, De Luca; Alba, Chimirri; Stefania, Ferro; Rosaria, Gitto; Julio, Alvarez-Builla; Ramon, Alajarin
Inhibition of HIV-1 RT activity by a new series of 3-(1,3,4-thiadiazol-2-yl)thiazolidin-4-one derivatives 1-gen-2020 Buemi, M. R.; Gitto, R.; Ielo, L.; Pannecouque, C.; De Luca, L.
Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases 1-gen-2018 De Luca, Laura; Mancuso, Francesca; Ferro, Stefania; Buemi, Maria Rosa; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria
InVivo Evaluation of Selective Carbonic Anhydrase Inhibitors as Potential Anticonvulsant Agents 1-gen-2016 Bruno, Elvira; Buemi, Mariarosa; DE LUCA, Laura; Ferro, Stefania; Monforte, Anna Maria; Supuran, Claudiu T.; Vullo, Daniela; De Sarro, Giovambattista; Russo, Emilio; Gitto, Rosaria
New indole derivatives as promising ligands for ifenprodil site of NR2B/NMDA receptors 1-gen-2010 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Buemi, Mariarosa; De Sarro, G; Chimirri, Alba
Nuovi ligandi del recettore NR2B/NMDA a struttura indolica 1-gen-2009 Buemi, Mariarosa; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Chimirri, Alba