DE GRAZIA, SARA
DE GRAZIA, SARA
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]1,3-oxazolidin-2-one
2011-01-01 Brancatelli G.; Nicolò F.; De Grazia S.; Monforte A.M.; Chimirri A.
4-[1-(4-Fluorobenzyl)-4-hydroxy-1H-indol-3-yl]-2-hydroxy-4-oxobut-2-enoic acid as a prototype to develop dual inhibitors of HIV-1 integration process.
2011-01-01 DE LUCA, Laura; Gitto, Rosaria; Christ, F; Ferro, Stefania; DE GRAZIA, Sara; Morreale, F; Debyser, Z; Chimirri, Alba
Antiretroviral strategy using multi-target agents
2009-01-01 Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; Gitto, Rosaria; Monforte, Anna Maria; Barreca, Ml; Christ, F; Chimirri, Alba
Antiretroviral strategy: design and synthesis of HIV-1 IN-LEDGF/p75 interaction inhibitors
2009-01-01 Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; Gitto, Rosaria; Monforte, Anna Maria; Barreca, Ml; Christ, F; Chimirri, Alba
Binding mode investigation and SAR studies of HIV-1 integrase inhibitors
2011-01-01 DE GRAZIA, Sara; DE LUCA, Laura; Gitto, Rosaria; Ferro, Stefania; Debyser, Z; Chimirri, Alba
Computational studies and synthetic approaches for the identification of new protein-protein interaction inhibitors (PPI)
2010-01-01 DE LUCA, Laura; DE GRAZIA, Sara; Ferro, Stefania; Gitto, Rosaria; Barreca, L; Debyser, Z; Chimirri, Alba
Design and synthesis of acetylcholinesterase inhibitors
2006-01-01 Gitto, Rosaria; Chimirri, Alba; Pagano, Benedetta; Francica, Eleonora; DE GRAZIA, Sara; DE LUCA, Grazia
Design e Sintesi di composti a struttura 3-Indol-Gliossilamidica come potenziali inibitori dell'integrasi dell'HIV-1.
2007-01-01 DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Monforte, Anna Maria; Witvrouw, M; Debyser, Z; Chimirri, Alba
Discovery of potent HIV-1 integrase strand transfer inhibitors: design and synthetic strategies
2009-01-01 DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Debyser, Z; Chimirri, Alba
Docking studies on a new human immunodeficiency virus integrase-Mg-DNA complex: phenyl ring exploration and synthesis of 1H-benzylindole derivatives through fluorine substitutions
2009-01-01 Ferro, Stefania; DE LUCA, Laura; Barreca, Maria Letizia; Iraci, Nunzio; DE GRAZIA, Sara; Christ, F; Witvrouw, M; Debyser, Z; Chimirri, Alba
From 3D-pharmacophore models to synthetic route towards anti-HIV agents
2009-01-01 Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; DE GRAZIA, Sara; Iraci, Nunzio; Barreca, Ml; Debyser, Z.
Glutamatergic neurotransmission as molecular target of new anticonvulsants.
2012-01-01 Gitto, Rosaria; DE LUCA, Laura; DE GRAZIA, Sara; Chimirri, Alba
HIV-1 integrase strand-transfer inhibitors: design and synthetic strategies in the process of a lead optimization
2010-01-01 DE GRAZIA, Sara; DE LUCA, Laura; Ferro, Stefania; Barreca M., L; Christ, F; Debyser, Z; Chimirri, Alba
HIV-1 integrase strand-transfer inhibitors: Design, synthesis and molecular modeling investigation
2011-01-01 DE LUCA, Laura; DE GRAZIA, Sara; Ferro, Stefania; Gitto, Rosaria; Christ, F; Debyser, Z; Chimirri, Alba
HIV-1-IN Strand-Transfer Inhibitors: phenyl ring exploration and synthesis of 1H-benzylindole derivative through fluorine substitutions
2008-01-01 Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Iraci, Nunzio; DE GRAZIA, Sara; Debyser, Z; Witvrouw, M; Chimirri, Alba
Inhibitors of the Interactions between HIV-1 IN and the Cofactor LEDGF/p75
2011-01-01 De Luca L; Ferro S; Morreale F; De Grazia S; Chimirri A
Insight into the INSTIs binding mode: molecular modeling investigation and SAR studies
2010-01-01 DE LUCA, Laura; DE GRAZIA, Sara; Ferro, Stefania; Debyser, Z.; Chimirri, Alba
INTEGRASE STRAND TRANSFER INHIBITORS (INSTIs): SYNTHESIS AND ANTIVIRAL EFFETCS OF CHLORO-FLUORO SUBSTITUTIONS
2008-01-01 Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; MARIA LETIZIA, Barreca; Iraci, Nunzio; Frauke, Christ; Zeger, Debyser; Chimirri, Alba
Microwave assisted organic synthesis (MAOS) of small molecules as potential HIV-1 integrase inhibitors.
2011-01-01 Ferro, Stefania; DE GRAZIA, Sara; DE LUCA, Laura; Gitto, Rosaria; Faliti, Ce; Debyzer, Z; Chimirri, Alba
Modificazioni strutturali del gruppo dichetoacido (DKA) di potenti inibitori dell'Integrasi dell'HIV-1
2007-01-01 DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; M. L., Barreca; Monforte, Anna Maria; M., Witvrouw; Z., Debyser; Chimirri, Alba
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]1,3-oxazolidin-2-one | 1-gen-2011 | Brancatelli G.; Nicolò F.; De Grazia S.; Monforte A.M.; Chimirri A. | |
| 4-[1-(4-Fluorobenzyl)-4-hydroxy-1H-indol-3-yl]-2-hydroxy-4-oxobut-2-enoic acid as a prototype to develop dual inhibitors of HIV-1 integration process. | 1-gen-2011 | DE LUCA, Laura; Gitto, Rosaria; Christ, F; Ferro, Stefania; DE GRAZIA, Sara; Morreale, F; Debyser, Z; Chimirri, Alba | |
| Antiretroviral strategy using multi-target agents | 1-gen-2009 | Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; Gitto, Rosaria; Monforte, Anna Maria; Barreca, Ml; Christ, F; Chimirri, Alba | |
| Antiretroviral strategy: design and synthesis of HIV-1 IN-LEDGF/p75 interaction inhibitors | 1-gen-2009 | Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; Gitto, Rosaria; Monforte, Anna Maria; Barreca, Ml; Christ, F; Chimirri, Alba | |
| Binding mode investigation and SAR studies of HIV-1 integrase inhibitors | 1-gen-2011 | DE GRAZIA, Sara; DE LUCA, Laura; Gitto, Rosaria; Ferro, Stefania; Debyser, Z; Chimirri, Alba | |
| Computational studies and synthetic approaches for the identification of new protein-protein interaction inhibitors (PPI) | 1-gen-2010 | DE LUCA, Laura; DE GRAZIA, Sara; Ferro, Stefania; Gitto, Rosaria; Barreca, L; Debyser, Z; Chimirri, Alba | |
| Design and synthesis of acetylcholinesterase inhibitors | 1-gen-2006 | Gitto, Rosaria; Chimirri, Alba; Pagano, Benedetta; Francica, Eleonora; DE GRAZIA, Sara; DE LUCA, Grazia | |
| Design e Sintesi di composti a struttura 3-Indol-Gliossilamidica come potenziali inibitori dell'integrasi dell'HIV-1. | 1-gen-2007 | DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Monforte, Anna Maria; Witvrouw, M; Debyser, Z; Chimirri, Alba | |
| Discovery of potent HIV-1 integrase strand transfer inhibitors: design and synthetic strategies | 1-gen-2009 | DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Debyser, Z; Chimirri, Alba | |
| Docking studies on a new human immunodeficiency virus integrase-Mg-DNA complex: phenyl ring exploration and synthesis of 1H-benzylindole derivatives through fluorine substitutions | 1-gen-2009 | Ferro, Stefania; DE LUCA, Laura; Barreca, Maria Letizia; Iraci, Nunzio; DE GRAZIA, Sara; Christ, F; Witvrouw, M; Debyser, Z; Chimirri, Alba | |
| From 3D-pharmacophore models to synthetic route towards anti-HIV agents | 1-gen-2009 | Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; DE GRAZIA, Sara; Iraci, Nunzio; Barreca, Ml; Debyser, Z. | |
| Glutamatergic neurotransmission as molecular target of new anticonvulsants. | 1-gen-2012 | Gitto, Rosaria; DE LUCA, Laura; DE GRAZIA, Sara; Chimirri, Alba | |
| HIV-1 integrase strand-transfer inhibitors: design and synthetic strategies in the process of a lead optimization | 1-gen-2010 | DE GRAZIA, Sara; DE LUCA, Laura; Ferro, Stefania; Barreca M., L; Christ, F; Debyser, Z; Chimirri, Alba | |
| HIV-1 integrase strand-transfer inhibitors: Design, synthesis and molecular modeling investigation | 1-gen-2011 | DE LUCA, Laura; DE GRAZIA, Sara; Ferro, Stefania; Gitto, Rosaria; Christ, F; Debyser, Z; Chimirri, Alba | |
| HIV-1-IN Strand-Transfer Inhibitors: phenyl ring exploration and synthesis of 1H-benzylindole derivative through fluorine substitutions | 1-gen-2008 | Ferro, Stefania; DE LUCA, Laura; Barreca, Ml; Iraci, Nunzio; DE GRAZIA, Sara; Debyser, Z; Witvrouw, M; Chimirri, Alba | |
| Inhibitors of the Interactions between HIV-1 IN and the Cofactor LEDGF/p75 | 1-gen-2011 | De Luca L; Ferro S; Morreale F; De Grazia S; Chimirri A | |
| Insight into the INSTIs binding mode: molecular modeling investigation and SAR studies | 1-gen-2010 | DE LUCA, Laura; DE GRAZIA, Sara; Ferro, Stefania; Debyser, Z.; Chimirri, Alba | |
| INTEGRASE STRAND TRANSFER INHIBITORS (INSTIs): SYNTHESIS AND ANTIVIRAL EFFETCS OF CHLORO-FLUORO SUBSTITUTIONS | 1-gen-2008 | Ferro, Stefania; DE LUCA, Laura; DE GRAZIA, Sara; MARIA LETIZIA, Barreca; Iraci, Nunzio; Frauke, Christ; Zeger, Debyser; Chimirri, Alba | |
| Microwave assisted organic synthesis (MAOS) of small molecules as potential HIV-1 integrase inhibitors. | 1-gen-2011 | Ferro, Stefania; DE GRAZIA, Sara; DE LUCA, Laura; Gitto, Rosaria; Faliti, Ce; Debyzer, Z; Chimirri, Alba | |
| Modificazioni strutturali del gruppo dichetoacido (DKA) di potenti inibitori dell'Integrasi dell'HIV-1 | 1-gen-2007 | DE GRAZIA, Sara; Ferro, Stefania; DE LUCA, Laura; M. L., Barreca; Monforte, Anna Maria; M., Witvrouw; Z., Debyser; Chimirri, Alba |