MANCUSO, Francesca
MANCUSO, Francesca
Dipartimento di Scienze chimiche, biologiche, farmaceutiche e ambientali
4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae
2021-01-01 Mancuso, F.; De Luca, L.; Bucolo, F.; Vrabel, M.; Angeli, A.; Capasso, C.; Supuran, C. T.; Gitto, R.
Effetto in vitro di derivati di 1-(1H-indol-3-il) etanone e propan-1-one su Candida spp. and Aspergillus niger
2021-01-01 Gervasi, Teresa; Ginestra, Giovanna; Mancuso, Francesca; Barreca, Davide; DE LUCA, Laura; Mandalari, Giuseppina
Exploring structural properties of potent human carbonic anhydrase inhibitors bearing a 4-(cycloalkylamino-1-carbonyl)benzenesulfonamide moiety
2019-01-01 Buemi, Maria Rosa; Di Fiore, Anna; De Luca, Laura; Angeli, Andrea; Mancuso, Francesca; Ferro, Stefania; Monti, Simona Maria; Buonanno, Martina; Russo, Emilio; De Sarro, Giovanbattista; De Simone, Giuseppina; Supuran, Claudiu T; Gitto, Rosaria
In Silico-Guided Identification of New Potent Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae
2020-01-01 Mancuso, Francesca; De Luca, Laura; Angeli, Andrea; Berrino, Emanuela; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria
Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases
2018-01-01 De Luca, Laura; Mancuso, Francesca; Ferro, Stefania; Buemi, Maria Rosa; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria
Looking toward the Rim of the Active Site Cavity of Druggable Human Carbonic Anhydrase Isoforms
2020-01-01 Mancuso, F.; Di Fiore, A.; De Luca, L.; Angeli, A.; Monti, S. M.; De Simone, G.; Supuran, C. T.; Gitto, R.
P158-DEVELOPMENT OF FLEXIBLE ARYLSULFONAMIDES AS POTENTIAL MULTITARGET ANTICANCER AGENTS
2020-01-01 Bucolo, Federica; Mancuso, Francesca; DE LUCA, Laura; Angeli, Andrea; Supuran, Claudiu T.; Gitto, Rosaria
Proton transfer mediated recognition of amines by ionizable macrocyclic receptors
2022-01-01 Gattuso, Giuseppe; Crisafulli, Daniele; Milone, Marco; Mancuso, Francesca; Pisagatti, Ilenia; Notti, Anna; Parisi, Melchiorre F.
Seeking new approach for therapeutic treatment of cholera disease via inhibition of bacterial carbonic anhydrases: experimental and theoretical studies for sixteen benzenesulfonamide derivatives
2019-01-01 Gitto, R.; De Luca, L.; Mancuso, Francesca; Del Prete, S.; Vullo, D.; Supuran, CLAUDIU TRANDAFIR; Capasso, C.
Simulated human digestion of N1-aryl-2-arylthioacetamidobenzimidazoles and their activity against Herpes-simplex virus 1 in vitro
2019-01-01 Mandalari, Giuseppina; Bisignano, Carlo; Smeriglio, Antonella; Denaro, Marcella; Musarra-Pizzo, Maria; Pennisi, Rosamaria; Mancuso, Francesca; Ferro, Stefania; Trombetta, Domenico; Monforte, Anna Maria; Sciortino, Maria Teresa; De Luca, Laura
Synthesis and biological evaluation of sulfonamide-based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae
2022-01-01 Mancuso, F.; Angeli, A.; De Luca, V.; Bucolo, F.; De Luca, L.; Capasso, C.; Supuran, C. T.; Gitto, R.
Synthesis, computational studies and assessment of in vitro inhibitory activity of umbelliferon-based compounds against tumour-associated carbonic anhydrase isoforms IX and XII
2020-01-01 Mancuso, Francesca; De Luca, Laura; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria
Targeting Carbonic Anhydrases (CAs): Rational Design, Synthesis, Structural Studies and Biochemical Evaluation
2021-01-08 Mancuso, Francesca
Tetracationic-to-dianionic tetraamino-dihydroxy-tetraoxacalix[4]arene: A paraquat receptor for all seasons
2022-01-01 Mancuso, Francesca; Crisafulli, Daniele; Milone, Marco; Irto, Anna; Cigala, Rosalia Maria; Lando, Gabriele; Pisagatti, Ilenia; Notti, Anna; Gattuso, Giuseppe
The In Vitro Potential of 1-(1H-indol-3-yl) Derivatives against Candida spp. and Aspergillus niger as Tyrosinase Inhibitors
2021-01-01 Gervasi, T.; Ginestra, G.; Mancuso, F.; Barreca, D.; De Luca, L.; Mandalari, G.
The in vitro potential of novel carbonic anhydrase Inhibitors against candida spp
2022-01-01 Gitto, Rosaria; Mancuso, Francesca; Bucolo, Federica; Gervasi, Teresa; Ginestra, Giovanna; DE LUCA, Laura; Mandalari, Giuseppina
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae | 1-gen-2021 | Mancuso, F.; De Luca, L.; Bucolo, F.; Vrabel, M.; Angeli, A.; Capasso, C.; Supuran, C. T.; Gitto, R. | |
Effetto in vitro di derivati di 1-(1H-indol-3-il) etanone e propan-1-one su Candida spp. and Aspergillus niger | 1-gen-2021 | Gervasi, Teresa; Ginestra, Giovanna; Mancuso, Francesca; Barreca, Davide; DE LUCA, Laura; Mandalari, Giuseppina | |
Exploring structural properties of potent human carbonic anhydrase inhibitors bearing a 4-(cycloalkylamino-1-carbonyl)benzenesulfonamide moiety | 1-gen-2019 | Buemi, Maria Rosa; Di Fiore, Anna; De Luca, Laura; Angeli, Andrea; Mancuso, Francesca; Ferro, Stefania; Monti, Simona Maria; Buonanno, Martina; Russo, Emilio; De Sarro, Giovanbattista; De Simone, Giuseppina; Supuran, Claudiu T; Gitto, Rosaria | |
In Silico-Guided Identification of New Potent Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae | 1-gen-2020 | Mancuso, Francesca; De Luca, Laura; Angeli, Andrea; Berrino, Emanuela; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria | |
Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases | 1-gen-2018 | De Luca, Laura; Mancuso, Francesca; Ferro, Stefania; Buemi, Maria Rosa; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria | |
Looking toward the Rim of the Active Site Cavity of Druggable Human Carbonic Anhydrase Isoforms | 1-gen-2020 | Mancuso, F.; Di Fiore, A.; De Luca, L.; Angeli, A.; Monti, S. M.; De Simone, G.; Supuran, C. T.; Gitto, R. | |
P158-DEVELOPMENT OF FLEXIBLE ARYLSULFONAMIDES AS POTENTIAL MULTITARGET ANTICANCER AGENTS | 1-gen-2020 | Bucolo, Federica; Mancuso, Francesca; DE LUCA, Laura; Angeli, Andrea; Supuran, Claudiu T.; Gitto, Rosaria | |
Proton transfer mediated recognition of amines by ionizable macrocyclic receptors | 1-gen-2022 | Gattuso, Giuseppe; Crisafulli, Daniele; Milone, Marco; Mancuso, Francesca; Pisagatti, Ilenia; Notti, Anna; Parisi, Melchiorre F. | |
Seeking new approach for therapeutic treatment of cholera disease via inhibition of bacterial carbonic anhydrases: experimental and theoretical studies for sixteen benzenesulfonamide derivatives | 1-gen-2019 | Gitto, R.; De Luca, L.; Mancuso, Francesca; Del Prete, S.; Vullo, D.; Supuran, CLAUDIU TRANDAFIR; Capasso, C. | |
Simulated human digestion of N1-aryl-2-arylthioacetamidobenzimidazoles and their activity against Herpes-simplex virus 1 in vitro | 1-gen-2019 | Mandalari, Giuseppina; Bisignano, Carlo; Smeriglio, Antonella; Denaro, Marcella; Musarra-Pizzo, Maria; Pennisi, Rosamaria; Mancuso, Francesca; Ferro, Stefania; Trombetta, Domenico; Monforte, Anna Maria; Sciortino, Maria Teresa; De Luca, Laura | |
Synthesis and biological evaluation of sulfonamide-based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae | 1-gen-2022 | Mancuso, F.; Angeli, A.; De Luca, V.; Bucolo, F.; De Luca, L.; Capasso, C.; Supuran, C. T.; Gitto, R. | |
Synthesis, computational studies and assessment of in vitro inhibitory activity of umbelliferon-based compounds against tumour-associated carbonic anhydrase isoforms IX and XII | 1-gen-2020 | Mancuso, Francesca; De Luca, Laura; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Gitto, Rosaria | |
Targeting Carbonic Anhydrases (CAs): Rational Design, Synthesis, Structural Studies and Biochemical Evaluation | 8-gen-2021 | Mancuso, Francesca | |
Tetracationic-to-dianionic tetraamino-dihydroxy-tetraoxacalix[4]arene: A paraquat receptor for all seasons | 1-gen-2022 | Mancuso, Francesca; Crisafulli, Daniele; Milone, Marco; Irto, Anna; Cigala, Rosalia Maria; Lando, Gabriele; Pisagatti, Ilenia; Notti, Anna; Gattuso, Giuseppe | |
The In Vitro Potential of 1-(1H-indol-3-yl) Derivatives against Candida spp. and Aspergillus niger as Tyrosinase Inhibitors | 1-gen-2021 | Gervasi, T.; Ginestra, G.; Mancuso, F.; Barreca, D.; De Luca, L.; Mandalari, G. | |
The in vitro potential of novel carbonic anhydrase Inhibitors against candida spp | 1-gen-2022 | Gitto, Rosaria; Mancuso, Francesca; Bucolo, Federica; Gervasi, Teresa; Ginestra, Giovanna; DE LUCA, Laura; Mandalari, Giuseppina |