AGNELLO, STEFANO
AGNELLO, STEFANO
1-Aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1H)-sulfonamide derivatives: synthesis and biological evaluation
2009-01-01 Agnello, Stefano; Ferro, Stefania; Gitto, Rosaria; De Sarro, G; Russo, E; Vullo, D; Supuran T., C; Chimirri, Alba
A structure-based approach to ligand discovery for inhibition of HIV-1 IN-LEDGF/p75 interaction: a new target for anti-AIDS therapy
2009-01-01 DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; Gitto, Rosaria; Monforte, Anna Maria; Iraci, Nunzio; Barreca, Ml; Debyser, Z; Chimirri, Alba
Discovery of HIV-1 Integrase and cellular cofactor LEDGF/p75 interaction inhibitors
2009-01-01 Ferro, Stefania; Agnello, Stefano; DE LUCA, Laura; Barreca, Ml; Iraci, N; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
Discovery of potent and selective inhibitors of druggable carbonic anhydrase isoforms
2010-01-01 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; Damiano, FRANCESCA MARIA; Supuran, Ct; Brynda, J; Mader, P; Chimirri, Alba
From 3D-pharmacophore models to synthetic route towards anti-HIV agents
2009-01-01 Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; DE GRAZIA, Sara; Iraci, Nunzio; Barreca, Ml; Debyser, Z.
Identification of 3,4-Dihydroisoquinoline-2(1H)-sulfonamides as Potent Carbonic Anhydrase Inhibitors: Synthesis, Biological Evaluation, and Enzyme−Ligand X-ray Studies
2010-01-01 Gitto, Rosaria; Agnello, Stefano; Ferro, Stefania; DE LUCA, Laura; Vullo, D.; Brynda, J.; Mader, P.; Supuran, C. T.; Chimirri, Alba
Identification of isoquinoline-sulfonamides as potent and selective carbonic anhydrase inhibitors
2010-01-01 Damiano, FRANCESCA MARIA; Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; Supuran, Ct; Mader, P; Chimirri, Alba
Identification of Potent and Selective Human Carbonic Anhydrase VII (hCA VII) Inhibitors
2010-01-01 Gitto R; Agnello S; Ferro S; Vullo D; Supuran CT; Chimirri A.
Identification of potent carbonic anhydrase inhibitors: synthesis, biological evaluation and enzyme-ligand x-ray studies
2009-01-01 Gitto, Rosaria; Agnello, Stefano; Ferro, Stefania; Supuran, Ct; Brynda, J; Mader, P; Chimirri, Alba
New potent and selective carbonic anhydrase inhibitors: synthesis, biological evaluation and X-ray studies
2009-01-01 Ferro, Stefania; Gitto, Rosaria; Agnello, Stefano; Claudiu T., Supuran; Jiri, Brynda; Pavel, Mader; Chimirri, Alba
Novel targets for HIV therapy: small molecules blocking IN-LEDGF/p75 interaction
2009-01-01 Ferro, Stefania; DE LUCA, Laura; Agnello, Stefano; Barreca, Ml; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba
PROGETTAZIONE E SINTESI DI NUOVI DERIVATI ISOCHINOLINICI COME AGENTI ANTICONVULSIVANTI MULTITARGET
2008-01-01 Agnello, Stefano; Ferro, Stefania; DE SARRO, G; Russo, E; Supuran, C; Gitto, Rosaria; Chimirri, Alba
PROGETTAZIONE E SINTESI DI NUOVI DKA ANALOGHI COME POTENZIALI INIBITORI DELL’INTEGRASI DELL’HIV-1
2008-01-01 Agnello, Stefano; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Debyser, Z; Chimirri, Alba
PROGETTAZIONE E SINTESI DI NUOVI DKA ANALOGHI COME POTENZIALI INIBITORI DELL'INTEGRASI DELL'HIV-1
2008-01-01 Agnello, Stefano; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Z., Debyser; Chimirri, Alba
Small Molecules Targeting Protein–Protein Interactions: A Promising Anti-HIV Strategy
2010-01-01 Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Gitto, Rosaria; Monforte, Anna Maria; Agnello, Stefano; Barreca, Ml; Christ, F; Debyser, Z.
Small molecules targeting the interaction between HIV-1 integrase and LEDGF/p75 cofactor.
2010-01-01 DE LUCA, Laura; Ferro, Stefania; Gitto, Rosaria; Barreca, Ml; Agnello, Stefano; Christ, F; Debyser, Z; Chimirri, Alba
Structural basis for the interaction between carbonic anhydrase and 1,2,3,4-tetrahydroisoquinolin-2-ylsulfonamides
2011-01-01 Mader, P.; Brynda, J.; Gitto, Rosaria; Agnello, Stefano; Pachl, P.; Supuran, C. T.; Chimirri, Alba; Řezáčová, P.
Synthesis and evaluation of pharmacological profile of 1-aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1H)-sulfonamides.
2009-01-01 Gitto, Rosaria; Ferro, Stefania; Agnello, Stefano; DE LUCA, Laura; DE SARRO, G; Russo, E; Vullo, D; SUPURAN C., T; Chimirri, Alba
Synthesis and structure-active relationship of 1-aryl-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline anticonvulsants
2010-01-01 Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; Russo, E.; De Sarro, G.; Chimirri, Alba
Synthesis of new pyridazine derivatives as potential anti-HIV-1 agents
2009-01-01 Ferro, Stefania; Agnello, Stefano; Barreca, Ml; DE LUCA, Laura; Christ, F; Gitto, Rosaria
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1-Aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1H)-sulfonamide derivatives: synthesis and biological evaluation | 1-gen-2009 | Agnello, Stefano; Ferro, Stefania; Gitto, Rosaria; De Sarro, G; Russo, E; Vullo, D; Supuran T., C; Chimirri, Alba | |
A structure-based approach to ligand discovery for inhibition of HIV-1 IN-LEDGF/p75 interaction: a new target for anti-AIDS therapy | 1-gen-2009 | DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; Gitto, Rosaria; Monforte, Anna Maria; Iraci, Nunzio; Barreca, Ml; Debyser, Z; Chimirri, Alba | |
Discovery of HIV-1 Integrase and cellular cofactor LEDGF/p75 interaction inhibitors | 1-gen-2009 | Ferro, Stefania; Agnello, Stefano; DE LUCA, Laura; Barreca, Ml; Iraci, N; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba | |
Discovery of potent and selective inhibitors of druggable carbonic anhydrase isoforms | 1-gen-2010 | Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; Damiano, FRANCESCA MARIA; Supuran, Ct; Brynda, J; Mader, P; Chimirri, Alba | |
From 3D-pharmacophore models to synthetic route towards anti-HIV agents | 1-gen-2009 | Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; DE GRAZIA, Sara; Iraci, Nunzio; Barreca, Ml; Debyser, Z. | |
Identification of 3,4-Dihydroisoquinoline-2(1H)-sulfonamides as Potent Carbonic Anhydrase Inhibitors: Synthesis, Biological Evaluation, and Enzyme−Ligand X-ray Studies | 1-gen-2010 | Gitto, Rosaria; Agnello, Stefano; Ferro, Stefania; DE LUCA, Laura; Vullo, D.; Brynda, J.; Mader, P.; Supuran, C. T.; Chimirri, Alba | |
Identification of isoquinoline-sulfonamides as potent and selective carbonic anhydrase inhibitors | 1-gen-2010 | Damiano, FRANCESCA MARIA; Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; Supuran, Ct; Mader, P; Chimirri, Alba | |
Identification of Potent and Selective Human Carbonic Anhydrase VII (hCA VII) Inhibitors | 1-gen-2010 | Gitto R; Agnello S; Ferro S; Vullo D; Supuran CT; Chimirri A. | |
Identification of potent carbonic anhydrase inhibitors: synthesis, biological evaluation and enzyme-ligand x-ray studies | 1-gen-2009 | Gitto, Rosaria; Agnello, Stefano; Ferro, Stefania; Supuran, Ct; Brynda, J; Mader, P; Chimirri, Alba | |
New potent and selective carbonic anhydrase inhibitors: synthesis, biological evaluation and X-ray studies | 1-gen-2009 | Ferro, Stefania; Gitto, Rosaria; Agnello, Stefano; Claudiu T., Supuran; Jiri, Brynda; Pavel, Mader; Chimirri, Alba | |
Novel targets for HIV therapy: small molecules blocking IN-LEDGF/p75 interaction | 1-gen-2009 | Ferro, Stefania; DE LUCA, Laura; Agnello, Stefano; Barreca, Ml; Iraci, Nunzio; Gitto, Rosaria; Monforte, Anna Maria; Christ, F; Debyser, Z; Chimirri, Alba | |
PROGETTAZIONE E SINTESI DI NUOVI DERIVATI ISOCHINOLINICI COME AGENTI ANTICONVULSIVANTI MULTITARGET | 1-gen-2008 | Agnello, Stefano; Ferro, Stefania; DE SARRO, G; Russo, E; Supuran, C; Gitto, Rosaria; Chimirri, Alba | |
PROGETTAZIONE E SINTESI DI NUOVI DKA ANALOGHI COME POTENZIALI INIBITORI DELL’INTEGRASI DELL’HIV-1 | 1-gen-2008 | Agnello, Stefano; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Debyser, Z; Chimirri, Alba | |
PROGETTAZIONE E SINTESI DI NUOVI DKA ANALOGHI COME POTENZIALI INIBITORI DELL'INTEGRASI DELL'HIV-1 | 1-gen-2008 | Agnello, Stefano; Ferro, Stefania; DE LUCA, Laura; Gitto, Rosaria; Z., Debyser; Chimirri, Alba | |
Small Molecules Targeting Protein–Protein Interactions: A Promising Anti-HIV Strategy | 1-gen-2010 | Chimirri, Alba; DE LUCA, Laura; Ferro, Stefania; Gitto, Rosaria; Monforte, Anna Maria; Agnello, Stefano; Barreca, Ml; Christ, F; Debyser, Z. | |
Small molecules targeting the interaction between HIV-1 integrase and LEDGF/p75 cofactor. | 1-gen-2010 | DE LUCA, Laura; Ferro, Stefania; Gitto, Rosaria; Barreca, Ml; Agnello, Stefano; Christ, F; Debyser, Z; Chimirri, Alba | |
Structural basis for the interaction between carbonic anhydrase and 1,2,3,4-tetrahydroisoquinolin-2-ylsulfonamides | 1-gen-2011 | Mader, P.; Brynda, J.; Gitto, Rosaria; Agnello, Stefano; Pachl, P.; Supuran, C. T.; Chimirri, Alba; Řezáčová, P. | |
Synthesis and evaluation of pharmacological profile of 1-aryl-6,7-dimethoxy-3,4-dihydroisoquinoline-2(1H)-sulfonamides. | 1-gen-2009 | Gitto, Rosaria; Ferro, Stefania; Agnello, Stefano; DE LUCA, Laura; DE SARRO, G; Russo, E; Vullo, D; SUPURAN C., T; Chimirri, Alba | |
Synthesis and structure-active relationship of 1-aryl-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline anticonvulsants | 1-gen-2010 | Gitto, Rosaria; DE LUCA, Laura; Ferro, Stefania; Agnello, Stefano; Russo, E.; De Sarro, G.; Chimirri, Alba | |
Synthesis of new pyridazine derivatives as potential anti-HIV-1 agents | 1-gen-2009 | Ferro, Stefania; Agnello, Stefano; Barreca, Ml; DE LUCA, Laura; Christ, F; Gitto, Rosaria |